Issued Patents All Time
Showing 25 most recent of 85 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12428421 | Pyrimidinones as factor XIA inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2025-09-30 |
| 12077558 | Phosphorus (V)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophosphorus (V) compounds | Michael Schmidt, Bin Zheng, Kyle Knouse, Justine deGruyter, Martin D. Eastgate +3 more | 2024-09-03 |
| 12065505 | Antibodies and antigen binding peptides for factor XIa inhibitors and uses thereof | Joseph M. Luettgen, Lumelle Schneeweis, Ginger Rakestraw, Christina Terragni, Andrew K. Dilger +6 more | 2024-08-20 |
| 11613554 | Phosphorous (V)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (V) compounds | Michael Schmidt, Bin Zheng, Kyle Knouse, Justine deGruyter, Martin D. Eastgate +3 more | 2023-03-28 |
| 11192891 | Diazaspiro ROCK inhibitors | Yeheng Zhu, Sunita V. Dewnani | 2021-12-07 |
| 11083704 | Method of administering nitroxyl donating compounds | Paul D. Kessler, Maria Borentain, Tushar Garimella, Elyse G. Stock | 2021-08-10 |
| 11053247 | Pyrimidinones as factor XIA inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2021-07-06 |
| 10752641 | Diamide macrocycles having factor XIa inhibiting activity | Jun Shi, Donald J. P. Pinto | 2020-08-25 |
| 10676477 | Factor XIa macrocycle inhibitors bearing a non-aromatic P2' group | Yeheng Zhu, Andrew K. Dilger, Michael J. Orwat, Donald J. P. Pinto | 2020-06-09 |
| 10336754 | Pyrimidinones as factor XIa inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2019-07-02 |
| 10336730 | Substituted glycine derived FXIA inhibitors | James R. Corte, Donald J. P. Pinto, Leon M. Smith, II | 2019-07-02 |
| 10287288 | Factor XIa macrocyclic inhibitors bearing alkyl or cycloalkyl P2' moieties | Kumar Balashanmuga Pabbisetty, James R. Corte, Andrew K. Dilger, Yeheng Zhu | 2019-05-14 |
| 10273236 | Macrocyclic factor XIa inhibitors bearing heterocyclic groups | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2019-04-30 |
| 10208068 | Macrocycles as factor XIa inhibitors | Donald J. P. Pinto, James R. Corte, Wu-Der Yang | 2019-02-19 |
| 10160750 | Diamide macrocycles as factor XIa inhibitors | Leon M. Smith, II, Donald J. P. Pinto, James R. Corte | 2018-12-25 |
| 10081623 | Diamide macrocycles that are FXIa inhibitors | Jun Shi, Laura Nielsen, Zilun Hu, Mimi L. Quan | 2018-09-25 |
| 9951071 | Dihydropyridone P1 as factor XIa inhibitors | Wu-Der Yang, James R. Corte, Paul J. Gilligan, Donald J. P. Pinto, Andrew K. Dilger +4 more | 2018-04-24 |
| 9902742 | Macrocycles as factor XIa inhibitors | Donald J. P. Pinto, James R. Corte, Paul J. Gilligan, Tianan Fang, Leon M. Smith, II +2 more | 2018-02-27 |
| 9777001 | Macrocycles with aromatic P2′ groups as factor xia inhibitors | James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang, Yufeng Wang +7 more | 2017-10-03 |
| 9714231 | Pyrrolidine GPR40 modulators | Bruce A. Ellsworth, Elizabeth A. Jurica, Jun Shi, Xiang-Yang Ye, Ximao Wu +2 more | 2017-07-25 |
| 9656963 | Dihydropyrazole GPR40 modulators | Andres Hernandez, Bruce A. Ellsworth, Bin Chen | 2017-05-23 |
| 9611274 | Macrocycles as factor XIa inhibitors | Donald J. P. Pinto, James R. Corte, Paul J. Gilligan, Tianan Fang, Leon M. Smith, II +2 more | 2017-04-04 |
| 9604964 | Dihydropyrazole GPR40 modulators | Bruce A. Ellsworth, Jun Shi, Elizabeth A. Jurica, Andres Hernandez, Ximao Wu +3 more | 2017-03-28 |
| 9453018 | Pyrimidinones as factor XIa inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2016-09-27 |
| 9409908 | Dihydropyridone p1 as factor XIa inhibitors | Wu-Der Yang, James R. Corte, Paul J. Gilligan, Donald J. P. Pinto, Andrew K. Dilger +4 more | 2016-08-09 |