LI

Leon M. Smith, II

BS Bristol-Myers Squibb: 36 patents #78 of 3,969Top 2%
AM Amgen: 5 patents #645 of 2,867Top 25%
📍 Raritan, NJ: #10 of 167 inventorsTop 6%
🗺 New Jersey: #1,317 of 69,400 inventorsTop 2%
Overall (All Time): #75,457 of 4,157,543Top 2%
41
Patents All Time

Issued Patents All Time

Showing 1–25 of 41 patents

Patent #TitleCo-InventorsDate
12428421 Pyrimidinones as factor XIA inhibitors Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more 2025-09-30
11053247 Pyrimidinones as factor XIA inhibitors Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more 2021-07-06
10899743 Substituted glycine derived FXIA inhibitors Donald J. P. Pinto 2021-01-26
10829501 Spiroheptane salicylamides and related compounds as inhibitors of ROCK Vladimir Ladziata, Indawati DeLucca, Donald J. P. Pinto, Michael J. Orwat, Andrew K. Dilger +5 more 2020-11-10
10611776 Spiroheptane salicylamides and related compounds as inhibitors of rock Vladimir Ladziata, Indawati De Lucca, Donald J. P. Pinto, Michael J. Orwat, Andrew K. Dilger +5 more 2020-04-07
10336730 Substituted glycine derived FXIA inhibitors James R. Corte, William R. Ewing, Donald J. P. Pinto 2019-07-02
10336754 Pyrimidinones as factor XIa inhibitors Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more 2019-07-02
10273236 Macrocyclic factor XIa inhibitors bearing heterocyclic groups Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more 2019-04-30
10208021 Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, Shefali Srivastava 2019-02-19
10160750 Diamide macrocycles as factor XIa inhibitors Donald J. P. Pinto, James R. Corte, William R. Ewing 2018-12-25
10000466 Substituted 4,5,6,7-tetrahydropyrazolo[3,4-c]pyridines as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, James R. Corte, Shefali Srivastava 2018-06-19
9951071 Dihydropyridone P1 as factor XIa inhibitors Wu-Der Yang, James R. Corte, Paul J. Gilligan, Donald J. P. Pinto, William R. Ewing +4 more 2018-04-24
9944625 Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, Shefali Srivastava 2018-04-17
9902742 Macrocycles as factor XIa inhibitors Donald J. P. Pinto, James R. Corte, Paul J. Gilligan, Tianan Fang, Yufeng Wang +2 more 2018-02-27
9777001 Macrocycles with aromatic P2′ groups as factor xia inhibitors James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang, Yufeng Wang +7 more 2017-10-03
9738655 Tetrahydroisoquinolines containing substituted azoles as factor XIa inhibitors Donald J. P. Pinto, Charles G. Clarke, Michael J. Orwat, Yoon Jeon, James R. Corte 2017-08-22
9725435 Substituted 4,5,6,7-tetrahydropyrazolo[4,3-c]pyridines as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, James R. Corte, Shefali Srivastava 2017-08-08
9611274 Macrocycles as factor XIa inhibitors Donald J. P. Pinto, James R. Corte, Paul J. Gilligan, Tianan Fang, Yufeng Wang +2 more 2017-04-04
9453018 Pyrimidinones as factor XIa inhibitors Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more 2016-09-27
9447110 Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, Shefali Srivastava 2016-09-20
9409908 Dihydropyridone p1 as factor XIa inhibitors Wu-Der Yang, James R. Corte, Paul J. Gilligan, Donald J. P. Pinto, William R. Ewing +4 more 2016-08-09
9403774 Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors Donald J. P. Pinto, Charles G. Clark, Michael J. Orwat, William R. Ewing 2016-08-02
9394276 Substituted 1,2,3,4-tetrahydro-2,6-naphthyridines as factor XIa inhibitors Michael J. Orwat, Donald J. P. Pinto, James R. Corte, Shefali Srivastava 2016-07-19
9315519 Guanidine substituted tetrahydroisoquinoline compounds as factor XIa inhibitors Donald J. P. Pinto, Charles G. Clark, Michael J. Orwat, William R. Ewing 2016-04-19
9221818 Macrocycles as factor XIa inhibitors Donald J. P. Pinto, James R. Corte, Paul J. Gilligan, Tianan Fang, Yufeng Wang +2 more 2015-12-29