Issued Patents All Time
Showing 1–25 of 43 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12428421 | Pyrimidinones as factor XIA inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2025-09-30 |
| 11306081 | Phenylacetamides as inhibitors of rock | Donald J. P. Pinto | 2022-04-19 |
| 11053247 | Pyrimidinones as factor XIA inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2021-07-06 |
| 10829501 | Spiroheptane salicylamides and related compounds as inhibitors of ROCK | Leon M. Smith, II, Vladimir Ladziata, Indawati DeLucca, Donald J. P. Pinto, Andrew K. Dilger +5 more | 2020-11-10 |
| 10676477 | Factor XIa macrocycle inhibitors bearing a non-aromatic P2' group | Yeheng Zhu, Andrew K. Dilger, William R. Ewing, Donald J. P. Pinto | 2020-06-09 |
| 10611776 | Spiroheptane salicylamides and related compounds as inhibitors of rock | Leon M. Smith, II, Vladimir Ladziata, Indawati De Lucca, Donald J. P. Pinto, Andrew K. Dilger +5 more | 2020-04-07 |
| 10336754 | Pyrimidinones as factor XIa inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2019-07-02 |
| 10273236 | Macrocyclic factor XIa inhibitors bearing heterocyclic groups | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2019-04-30 |
| 10208021 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2019-02-19 |
| 10000466 | Substituted 4,5,6,7-tetrahydropyrazolo[3,4-c]pyridines as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, James R. Corte, Shefali Srivastava | 2018-06-19 |
| 9944625 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2018-04-17 |
| 9777001 | Macrocycles with aromatic P2′ groups as factor xia inhibitors | James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang, Yufeng Wang +7 more | 2017-10-03 |
| 9738655 | Tetrahydroisoquinolines containing substituted azoles as factor XIa inhibitors | Donald J. P. Pinto, Charles G. Clarke, Leon M. Smith, II, Yoon Jeon, James R. Corte | 2017-08-22 |
| 9725435 | Substituted 4,5,6,7-tetrahydropyrazolo[4,3-c]pyridines as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, James R. Corte, Shefali Srivastava | 2017-08-08 |
| 9453018 | Pyrimidinones as factor XIa inhibitors | Andrew K. Dilger, James R. Corte, Indawati De Lucca, Tianan Fang, Wu-Der Yang +7 more | 2016-09-27 |
| 9447110 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2016-09-20 |
| 9403774 | Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors | Donald J. P. Pinto, Charles G. Clark, Leon M. Smith, II, William R. Ewing | 2016-08-02 |
| 9394276 | Substituted 1,2,3,4-tetrahydro-2,6-naphthyridines as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, James R. Corte, Shefali Srivastava | 2016-07-19 |
| 9315519 | Guanidine substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Charles G. Clark, Leon M. Smith, II, William R. Ewing | 2016-04-19 |
| 9192607 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2015-11-24 |
| 9108951 | Substituted 5,6,7,8-tetrahydro-1,6-naphthyridines as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, James R. Corte, Shefali Srivastava | 2015-08-18 |
| 9079929 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2015-07-14 |
| 9000172 | Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors | Donald J. P. Pinto, Leon M. Smith, II, Shefali Srivastava | 2015-04-07 |
| 8367709 | Dipeptide analogs as coagulation factor inhibitors | Donald J. P. Pinto, Mimi L. Quan, Leon M. Smith, II, Paul J. Gilligan | 2013-02-05 |
| 7371761 | Lactam-containing compounds and derivatives thereof as factor Xa inhibitors | Donald J. P. Pinto, Mimi L. Quan, Yun-Long Li, Wei Han, Jennifer X. Qiao +2 more | 2008-05-13 |