Issued Patents All Time
Showing 1–25 of 82 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12404274 | Macrocycles as factor xia inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2025-09-02 |
| 12187699 | GSPT1 compounds and methods of use of the novel compounds | Joshua Hansen | 2025-01-07 |
| 11136327 | Macrocycles as factor XIA inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2021-10-05 |
| 10730858 | Lactam, cyclic urea and carbamate, and triazolone derivatives as potent and selective rock inhibitors | Zilun Hu, Cailan Wang, Peter W. Glunz | 2020-08-04 |
| 10487086 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2019-11-26 |
| 10385026 | Phthalazinones and isoquinolinones as rock inhibitors | Peter W. Glunz, Yan Zou, Vladimir Ladziata | 2019-08-20 |
| 10112936 | Five-membered heterocycles useful as serine protease inhibitors | Jon J. Hangeland, Joanne M. Smallheer, Gregory S. Bisacchi, James R. Corte, Todd J. Friends +3 more | 2018-10-30 |
| 10112939 | Tied-back benzamide derivatives as potent rock inhibitors | Zilun Hu, Doree F. Sitkoff | 2018-10-30 |
| 10081623 | Diamide macrocycles that are FXIa inhibitors | Jun Shi, William R. Ewing, Laura Nielsen, Zilun Hu | 2018-09-25 |
| 9926282 | Phthalazinones and isoquinolinones as rock inhibitors | Peter W. Glunz, Yan Zou, Vladimir Ladziata | 2018-03-27 |
| 9914740 | Tricyclic pyrido-carboxamide derivatives as rock inhibitors | Zilun Hu, Cailan Wang, Sharanabasappa Patil | 2018-03-13 |
| 9828345 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Zilun Hu | 2017-11-28 |
| 9802939 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2017-10-31 |
| 9745313 | Macrocycles as factor XIa inhibitors | Carl P. Decicco, James R. Corte, Cailan Wang | 2017-08-29 |
| 9663529 | Tricyclic pyrido-carboxamide derivatives as rock inhibitors | Zilun Hu, Cailan Wang | 2017-05-30 |
| 9617224 | Five-membered heterocycles useful as serine protease inhibitors | Jon J. Hangeland, Joanne M. Smallheer, Gregory S. Bisacchi, James R. Corte, Todd J. Friends +3 more | 2017-04-11 |
| 9458110 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Zilun Hu, Cailan Wang, Peter W. Glunz | 2016-10-04 |
| 9453029 | Macrocycles as factor XIa inhibitors | Carl P. Decicco, James R. Corte, Cailan Wang | 2016-09-27 |
| 9221767 | Substituted phthalazinones as rock inhibitors | Peter W. Glunz, Yan Zou | 2015-12-29 |
| 9126944 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Zilun Hu, Cailan Wang | 2015-09-08 |
| 9079860 | Five-membered heterocycles useful as serine protease inhibitors | Jon J. Hangeland, Joanne M. Smallheer, Gregory S. Bisacchi, James R. Corte, Todd J. Friends +3 more | 2015-07-14 |
| 9079918 | Macrocycles as factor XIa inhibitors | Carl P. Decicco, James R. Corte, Cailan Wang | 2015-07-14 |
| 8940720 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2015-01-27 |
| 8828983 | Macrocycles as factor XIa inhibitors | Carl P. Decicco, James R. Corte, Cailan Wang | 2014-09-09 |
| 8716492 | Five-membered heterocycles useful as serine protease inhibitors | Jon J. Hangeland, Joanne M. Smallheer, Gregory S. Bisacchi, James R. Corte, Todd J. Friends +3 more | 2014-05-06 |