Issued Patents All Time
Showing 1–25 of 26 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12404274 | Macrocycles as factor xia inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2025-09-02 |
| 11136327 | Macrocycles as factor XIA inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2021-10-05 |
| 10730858 | Lactam, cyclic urea and carbamate, and triazolone derivatives as potent and selective rock inhibitors | Cailan Wang, Mimi L. Quan, Peter W. Glunz | 2020-08-04 |
| 10487086 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2019-11-26 |
| 10112939 | Tied-back benzamide derivatives as potent rock inhibitors | Doree F. Sitkoff, Mimi L. Quan | 2018-10-30 |
| 10081623 | Diamide macrocycles that are FXIa inhibitors | Jun Shi, William R. Ewing, Laura Nielsen, Mimi L. Quan | 2018-09-25 |
| 9914740 | Tricyclic pyrido-carboxamide derivatives as rock inhibitors | Mimi L. Quan, Cailan Wang, Sharanabasappa Patil | 2018-03-13 |
| 9902702 | Spirocycloheptanes as inhibitors of rock | Vladimir Ladziata, Peter W. Glunz, Yufeng Wang | 2018-02-27 |
| 9828345 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Mimi L. Quan | 2017-11-28 |
| 9802939 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2017-10-31 |
| 9663529 | Tricyclic pyrido-carboxamide derivatives as rock inhibitors | Mimi L. Quan, Cailan Wang | 2017-05-30 |
| 9458110 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Mimi L. Quan, Cailan Wang, Peter W. Glunz | 2016-10-04 |
| 9126944 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Mimi L. Quan, Cailan Wang | 2015-09-08 |
| 8940720 | Macrocycles as factor XIa inhibitors | James R. Corte, Tianan Fang, Carl P. Decicco, Donald J. P. Pinto, Karen A. Rossi +5 more | 2015-01-27 |
| 8604056 | Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors | Donald J. P. Pinto, Joanne M. Smallheer, James R. Corte, Cullen L. Cavallaro, Paul J. Gilligan +2 more | 2013-12-10 |
| 8324199 | Pyridazine derivatives as factor xia inhibitors | James R. Corte, Mimi L. Quan | 2012-12-04 |
| 8252830 | Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors | Donald J. P. Pinto, Joanne M. Smallheer, James R. Corte, Cullen L. Cavallaro, Paul J. Gilligan +2 more | 2012-08-28 |
| 7842708 | Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor XIa inhibitors | Donald J. P. Pinto, Joanne M. Smallheer, James R. Corte, Cullen L. Cavallaro, Paul J. Gilligan +2 more | 2010-11-30 |
| 7626039 | Arylpropionamide, arylacrylamide, ayrlpropynamide, or arylmethylurea analogs as factor XIa inhibitors | Donald J. P. Pinto, Joanne M. Smallheer, James R. Corte, Cullen L. Cavallaro, Paul J. Gilligan +2 more | 2009-12-01 |
| 7524863 | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors | Joanne M. Smallheer, Donald J. P. Pinto, Shuaige Wang, Jennifer X. Qiao, Wei Han | 2009-04-28 |
| 7507730 | Substituted pyrazolo[1,5-a]pyrimidines as potassium channel activators | Wei Han | 2009-03-24 |
| 7312218 | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors | Wei Han, Timur Gungor | 2007-12-25 |
| 7199149 | Monocyclic and bicyclic lactams as factor Xa inhibitors | Wei Han, Jennifer X. Qiao | 2007-04-03 |
| 7169795 | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors | Wei Han, Timur Gungor | 2007-01-30 |
| 7157470 | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors | Joanne M. Smallheer, Donald J. P. Pinto, Shuaige Wang, Jennifer X. Qiao, Wei Han | 2007-01-02 |