Issued Patents All Time
Showing 1–25 of 28 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 11673886 | 5-membered and bicyclic heterocyclic amides as inhibitors of ROCK | Vladimir Ladziata, Indawati De Lucca, George O. Tora, Tarun Kumar Maishal, Raghuram Tangirala +1 more | 2023-06-13 |
| 11078197 | 5-membered and bicyclic heterocyclic amides as inhibitors of rock | Vladimir Ladziata, Indawati De Lucca, George O. Tora, Tarun Kumar Maishal, Raghuram Tangirala +1 more | 2021-08-03 |
| 10829501 | Spiroheptane salicylamides and related compounds as inhibitors of ROCK | Leon M. Smith, II, Vladimir Ladziata, Indawati DeLucca, Donald J. P. Pinto, Michael J. Orwat +5 more | 2020-11-10 |
| 10787450 | Spiro-fused cyclic ureas as inhibitors of rock | Rajeev S. Bhide, Mandar Shrikrishna Bodas, Pravin S. Shirude, Sharanabasappa Patil, Tarun Kumar Maishal +2 more | 2020-09-29 |
| 10730858 | Lactam, cyclic urea and carbamate, and triazolone derivatives as potent and selective rock inhibitors | Zilun Hu, Cailan Wang, Mimi L. Quan | 2020-08-04 |
| 10696674 | Spirolactams as inhibitors of ROCK | Indawati DeLucca, Andrew K. Dilger | 2020-06-30 |
| 10654860 | Tricyclic rho kinase inhibitors | Wu-Der Yang, Rajeev S. Bhide, Kamalraj Thiyagarajan | 2020-05-19 |
| 10611776 | Spiroheptane salicylamides and related compounds as inhibitors of rock | Leon M. Smith, II, Vladimir Ladziata, Indawati De Lucca, Donald J. P. Pinto, Michael J. Orwat +5 more | 2020-04-07 |
| 10562887 | Triazolones and tetrazolones as inhibitors of ROCK | Natesan Murugesan, Mandar Shrikrishna Bodas, Navnath Dnyanoba Yadav, Venu Alla | 2020-02-18 |
| 10385026 | Phthalazinones and isoquinolinones as rock inhibitors | Yan Zou, Mimi L. Quan, Vladimir Ladziata | 2019-08-20 |
| 10123993 | Cyclic ureas as inhibitors of rock | Doree F. Sitkoff, Navnath Dnyanoba Yadav, Mandar Shrikrishna Bodas, Rajeev S. Bhide, Sharanabasappa Patil +3 more | 2018-11-13 |
| 10112929 | Lactams as inhibitors of rock | Doree F. Sitkoff, Mandar Shrikrishna Bodas, Navnath Dnyanoba Yadav, Sharanabasappa Patil, Prasanna Savanor Maddu Rao | 2018-10-30 |
| 9926282 | Phthalazinones and isoquinolinones as rock inhibitors | Yan Zou, Mimi L. Quan, Vladimir Ladziata | 2018-03-27 |
| 9902702 | Spirocycloheptanes as inhibitors of rock | Vladimir Ladziata, Zilun Hu, Yufeng Wang | 2018-02-27 |
| 9458110 | Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors | Mimi L. Quan, Zilun Hu, Cailan Wang | 2016-10-04 |
| 9221767 | Substituted phthalazinones as rock inhibitors | Yan Zou, Mimi L. Quan | 2015-12-29 |
| 9174974 | Macrocyclic factor VIIa inhibitors | Xiaojun Zhang, Eldon Scott Priestley, James A. Johnson, Nicholas R. Wurtz, Vladimir Ladziata | 2015-11-03 |
| 8420830 | Macrocyclic factor VIIa inhibitors useful as anticoagulants | Nicholas R. Wurtz, Eldon Scott Priestley, Daniel L. Cheney, Xiaojun Zhang, Brandon Parkhurst +2 more | 2013-04-16 |
| 7592331 | Macrocyclic factor VIIa inhibitors useful as anticoagulants | Eldon Scott Priestley, Daniel L. Cheney, Nicholas R. Wurtz | 2009-09-22 |
| 7576098 | Heterocyclic compounds as inhibitors of factor VIIa | Nicolas Wurtz, Xuhong Cheng | 2009-08-18 |
| 7550146 | Glycopeptide conjugates and uses thereof | Samuel J. Danishefsky, Dalibor Sames, Samuel Hintermann, Govindaswami Ragupathi, Philip O. Livingston +2 more | 2009-06-23 |
| 7160856 | α-O-linked glycoconjugates, methods of preparation and uses thereof | Samuel J. Danishefsky, Dalibor Sames, Samuel Hintermann, Xiao-Tao Chen, Jacob Bradley Schwarz +4 more | 2007-01-09 |
| 7122559 | Phenylglycine derivatives useful as serine protease inhibitors | Gregory S. Bisacchi, George C. Morton, Alexandra Holubec, E. Scott Priestley, Xiaojun Zhang +1 more | 2006-10-17 |
| 7112601 | Cycloalkyl heterocycles for treating hepatitis C virus | Brent Douty, Scott W. Martin, Jeffrey Lee Romine | 2006-09-26 |
| 7094783 | Bicyclic pyrimidinones as coagulation cascade inhibitors | — | 2006-08-22 |