Patent Leaderboard
USPTO Patent Rankings Data through Sept 30, 2025
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Gregor James MacDonald — 72 Patents

Johnson & Johnson: 51 patents #100 of 7,810Top 2%
ASAddex Pharma, S.A.: 17 patents #3 of 38Top 8%
GLGlaxo Group Limited: 11 patents #73 of 1,368Top 6%
VUVanderbilt University: 8 patents #84 of 1,609Top 6%
CLCellzome Limited: 3 patents #18 of 59Top 35%
SPSmithkline Beeacham P.L.C.: 2 patents #217 of 690Top 35%
Beerse, BE: #2 of 178 inventorsTop 2%
Overall (All Time): #27,897 of 4,157,543Top 1%
72 Patents All Time

Issued Patents All Time

Showing 26–50 of 72 patents

Patent #TitleCo-InventorsDate
8946205 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors Jose Maria Cid-Nunez, Ana Isabel De Lucas Olivares, Andrés Avelino Trabanco-Suárez 2015-02-03
8946426 Substituted bicyclic heterocyclic compounds as gamma secretase modulators Henricus Jacobus Maria Gijsen, Adriana Ingrid Velter, François Paul Bischoff, Tongfei Wu, Sven Franciscus Anna Van Brandt +6 more 2015-02-03
8940743 Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists Marcel Frans Leopold De Bruyn, Ludo Edmond Josephine Kennis, Xavier Jean Michel Langlois, Frans Alfons Maria Van den Keybus, Yves Emiel Maria Van Roosbroeck 2015-01-27
8937060 1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the treatment of prevention of neurological and psychiatric disorders Jose Maria Cid-Nunez, Daniel Oehlrich, Andrés Avelino Trabanco-Suárez, Gary John Tresadern, Juan Antonio Vega Ramiro 2015-01-20
8933101 Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists José Manuel Bartolomé-Nebreda, Michiel Luc Maria Van Gool 2015-01-13
8906939 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives Jose Maria Cid-Nunez, Andrés Avelino Trabanco-Suárez, Guillaume Albert Jacques Duvey 2014-12-09
8906921 4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists José Manuel Bartolomé-Nebreda 2014-12-09
8901125 Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide +4 more 2014-12-02
8895562 Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists José Manuel Bartolomé-Nebreda, Michiel Luc Maria Van Gool 2014-11-25
8865725 Substituted imidazopyrimidin-5(6H)-ones as allosteric modulators of MGLUR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide +3 more 2014-10-21
8859543 Imidazo[1,2-a]pyrazine derivatives and their use for the prevention or treatment of neurological, psychiatric and metabolic disorders and diseases José Manuel Bartolomé-Nebreda, Susana Conde-Ceide, Joaquin Pastor-Fernández, Michiel Luc Maria Van Gool, María Luz Martín-Martín +1 more 2014-10-14
8853237 Naphthyridinone analogs as mGluR5 positive allosteric modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Jason Manka, Jon Jacobs +4 more 2014-10-07
8841323 1, 4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of MGLUR2-receptors Hassan Imogai, Jose Maria Cid-Nunez, José Ignacio Andrés-Gil, Andrés Avelino Trabanco-Suárez, Julen Oyarzabal Santamarina +7 more 2014-09-23
8829011 2-aminopyrimidine compounds as serotonin receptor modulators Nicholas I. Carruthers, Brock T. Shireman, Vi T. Tran 2014-09-09
8791120 Fast-dissociating dopamine 2 receptor antagonists Xavier Jean Michel Langlois, José Manuel Bartolomé-Nebreda, Michiel Luc Maria Van Gool 2014-07-29
8791144 Substituted N-phenyl-1-(4-Pyridinyl)-1H-pyrazol-3-amines Johannes Wilhelmus John F. Thuring, Frans Alfons Maria Van den Keybus, Yves Emiel Maria Van Roosbroeck 2014-07-29
8778974 Trisubstituted 1,2,4 triazoles Johannes Wilhelmus John F. Thuring, Pauline Stanislawski, Wei Zhuang, Yves Emiel Maria Van Roosbroeck, Frans Alfons Maria Van den Keybus 2014-07-15
8779158 Trisubstituted pyrazoles as acetylcholine receptor modulators Johannes Wilhelmus John F. Thuring, Wei Zhuang 2014-07-15
8772504 Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators Henricus Jacobus Maria Gijsen, François Paul Bischoff, Wei Zhuang, Sven Franciscus Anna Van Brandt, Michel Surkyn +4 more 2014-07-08
8748621 1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones Jose Maria Cid-Nunez, Andrés Avelino Trabanco-Suárez, Guillaume Albert Jacques Duvey, Robert Johannes Lutjens, Patrick Terry Finn 2014-06-10
8722894 1,3-disubstituted-4-phenyl-1H-pyridin-2-ones Jose Maria Cid-Nunez, Andrés Avelino Trabanco-Suárez, Guillaume Albert Jacques Duvey, Robert Johannes Lutjens, Patrick Terry Finn 2014-05-13
8716480 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors Jose Maria Cid-Nunez, Ana Isabel De Lucas Olivares, Andrés Avelino Trabanco-Suárez 2014-05-06
8716282 Imidazo[1,2-b]pyridazine derivatives and their use as PDE10 inhibitors Joaquin Pastor-Fernández, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide, Óscar Delgado-González, Greta Constantia Peter Vanhoof +7 more 2014-05-06
8710074 Dihydronaphthyridinyl(organo)methanone analogs as positive allosteric mGluR5 modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Jason Manka, Jon Jacobs +4 more 2014-04-29
8691813 Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors Jose Maria Cid-Nunez, Andrés Avelino Trabanco-Suárez 2014-04-08