JB

José Manuel Bartolomé-Nebreda

Johnson & Johnson: 16 patents #613 of 7,810Top 8%
VU Vanderbilt University: 10 patents #62 of 1,609Top 4%
📍 Toledo, ES: #3 of 68 inventorsTop 5%
Overall (All Time): #146,609 of 4,157,543Top 4%
27
Patents All Time

Issued Patents All Time

Showing 1–25 of 27 patents

Patent #TitleCo-InventorsDate
9550784 Inhibitors of phosphodiesterase 10 enzyme Laurent Christian L. Leclercq, Susana Conde-Ceide, Michiel Luc Maria Van Gool 2017-01-24
9422296 Fast-dissociating dopamine 2 receptor antagonists Gregor James MacDonald, Xavier Jean Michel Langlois, Michiel Luc Maria Van Gool 2016-08-23
9255103 Substituted pyrazolo[1,5-a]pyrazines as mGluR5 receptor modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Susana Conde-Ceide, Gregor James MacDonald +2 more 2016-02-09
9090632 Bicyclic oxazole and thiazole compounds and their use as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Carrie K. Jones, Susana Conde-Ceide +2 more 2015-07-28
9040707 Bicyclic thiazoles as allosteric modulators of mGluR5 receptors Gregor James MacDonald, Andrés Avelino Trabanco-Suárez, Susana Conde-Ceide, Gary John Tresadern, Joaquin Pastor-Fernández 2015-05-26
9029366 Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Susana Conde-Ceide, Gregor James MacDonald +4 more 2015-05-12
8969389 Substituted 6-methylnicotinamides as mGluR5 positive allosteric modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Ya Zhou, Jason Manka +1 more 2015-03-03
8933101 Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists Gregor James MacDonald, Michiel Luc Maria Van Gool 2015-01-13
8906921 4-alkoxypyridazine derivatives as fast dissociating dopamine 2 receptor antagonists Gregor James MacDonald 2014-12-09
8901125 Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Susana Conde-Ceide, Gregor James MacDonald +4 more 2014-12-02
8895562 Piperazin-1-yl-trifluoromethyl-substituted-pyridines as fast dissociating dopamine 2 receptor antagonists Gregor James MacDonald, Michiel Luc Maria Van Gool 2014-11-25
8865725 Substituted imidazopyrimidin-5(6H)-ones as allosteric modulators of MGLUR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Gregor James MacDonald, Susana Conde-Ceide +3 more 2014-10-21
8859543 Imidazo[1,2-a]pyrazine derivatives and their use for the prevention or treatment of neurological, psychiatric and metabolic disorders and diseases Susana Conde-Ceide, Gregor James MacDonald, Joaquin Pastor-Fernández, Michiel Luc Maria Van Gool, María Luz Martín-Martín +1 more 2014-10-14
8853237 Naphthyridinone analogs as mGluR5 positive allosteric modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Jason Manka, Jon Jacobs +4 more 2014-10-07
8791120 Fast-dissociating dopamine 2 receptor antagonists Gregor James MacDonald, Xavier Jean Michel Langlois, Michiel Luc Maria Van Gool 2014-07-29
8716282 Imidazo[1,2-b]pyridazine derivatives and their use as PDE10 inhibitors Joaquin Pastor-Fernández, Gregor James MacDonald, Susana Conde-Ceide, Óscar Delgado-González, Greta Constantia Peter Vanhoof +7 more 2014-05-06
8710074 Dihydronaphthyridinyl(organo)methanone analogs as positive allosteric mGluR5 modulators P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Jason Manka, Jon Jacobs +4 more 2014-04-29
8703946 Substituted pyrazolo[1,5-A]pyrazine compounds as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Carrie K. Jones, Shaun R. Stauffer, Gregor McDonald +2 more 2014-04-22
8592422 Bicyclic triazole and pyrazole lactams as allosteric modulators of mGluR5 receptors P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, Susana Conde-Ceide, Gregor James MacDonald +5 more 2013-11-26
8530474 Substituted 6-(1-piperazinyl)-pyridazines as 5-HT6 receptor antagonists Gregor James MacDonald, Michiel Luc Maria Van Gool, Susana Conde-Ceide, Francisca Delgado-Jiménez 2013-09-10
8466153 Piperidinylamino-pyridazines and their use as fast dissociating dopamine 2 receptor antagonists Gregor James MacDonald, José Ignacio Andrés-Gil, Frans Alfons Maria Van den Keybus, Michiel Luc Maria Van Gool 2013-06-18
7732437 Use of anti-histaminics for acute reduction of elevated intracranial pressure Frank Tegtmeier, Frans Eduard Janssens, Joseph Elisabeth Leenaerts, Koenraad Arthur van Rossem, Manuel Jesús Alcázar-Vaca +4 more 2010-06-08
7635696 Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic activity José Ignacio Andrés-Gil, Manuel Jesús Alcázar-Vaca, Maria de las Mercedes Garcia-Martin, Antonius Adrianus Hendrikus Petrus Megens 2009-12-22
7476662 Substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine Frans Eduard Janssens, Joseph Elisabeth Leenaerts, Koenraad Arthur van Rossem, Manuel Jesús Alcázar-Vaca, Pedro Martinez-Jimenez +3 more 2009-01-13
7465741 C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants José Ignacio Andrés-Gil, Rosa Maria Alvarez-Escobar, Margaretha Henrica Maria Bakker, Antonius Adrianus Hendrikus Petrus Megens 2008-12-16