| 10967078 |
Radiolabelled mGluR2 PET ligands |
Michiel Luc Maria Van Gool, José Ignacio Andrés-Gil, Guy Maurits R. Bormans, Sofie Jeanne Leopoldine Celen, Joost Verbeek |
2021-04-06 |
| 10072014 |
6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one compounds and their use as negative allosteric modulators of MGLUR2 receptors |
Michiel Luc Maria Van Gool, Sergio-Alvar Alonso-de Diego, Ana Isabel De Lucas Olivares |
2018-09-11 |
| 9029366 |
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors |
P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide +4 more |
2015-05-12 |
| 8901125 |
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulators of mGluR5 receptors |
P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide +4 more |
2014-12-02 |
| 8592422 |
Bicyclic triazole and pyrazole lactams as allosteric modulators of mGluR5 receptors |
P. Jeffrey Conn, Craig W. Lindsley, Shaun R. Stauffer, José Manuel Bartolomé-Nebreda, Susana Conde-Ceide +5 more |
2013-11-26 |
| 8329704 |
Substituted pyrazinone derivatives for use in MCH-1 mediated diseases |
José Ignacio Andrés-Gil, Rosa Maria Alvarez-Escobar, Julen Oyarzabal Santamarina, Frank Matthias Dautzenberg, Jacqueline Anne Macritchie +2 more |
2012-12-11 |
| 8158643 |
Substituted diaza-spiro-pyridinone derivatives for use in MCH-1 mediated diseases |
José Ignacio Andrés-Gil, Frank Matthias Dautzenberg, Joannes Theodorus Maria Linders |
2012-04-17 |
| 7732437 |
Use of anti-histaminics for acute reduction of elevated intracranial pressure |
Frank Tegtmeier, Frans Eduard Janssens, Joseph Elisabeth Leenaerts, Koenraad Arthur van Rossem, Pedro Martinez-Jimenez +4 more |
2010-06-08 |
| 7635696 |
Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic activity |
José Ignacio Andrés-Gil, José Manuel Bartolomé-Nebreda, Maria de las Mercedes Garcia-Martin, Antonius Adrianus Hendrikus Petrus Megens |
2009-12-22 |
| 7501418 |
Fused heterocyclic isoxazoline derivatives and their use as anti-depressants |
José Ignacio Andrés-Gil, José Manuel Bartolomé -Nebreda, Francisco Javier Fernandez-Gadea, Margaretha Henrica Maria Bakker, Antonius Adrianus Hendrikus Petrus Megens |
2009-03-10 |
| 7476662 |
Substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine |
Frans Eduard Janssens, Joseph Elisabeth Leenaerts, Koenraad Arthur van Rossem, Pedro Martinez-Jimenez, José Manuel Bartolomé-Nebreda +3 more |
2009-01-13 |
| 7462717 |
C6-and C9-substituted chromeno[4,3-c]isoxazoline derivatives and their use as anti-depressants |
José Ignacio Andrés-Gil, Maria Encarnacion Matesanz-Ballesteros, Margaretha Henrica Maria Bakker, Antonius Adrianus Hendrikus Petrus Megens |
2008-12-09 |
| 7423048 |
Compounds for treating fundic disaccomodation |
Kristol Van Emelen, Marcel Frans Leopold De Bruyn, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea, Maria Encamacion Matesanz-Ballesteros +1 more |
2008-09-09 |
| 7265103 |
Substituted amino isoxazoline derivatives and their use as anti-depressants |
José Ignacio Andrés-Gil, Margaretha Henrica Maria Bakker, Ana Isabel De Lucas Olivares |
2007-09-04 |
| 7169786 |
Isoxazoline derivatives as anti-depressants |
José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea, Jose Maria Cid-Nunez, Joaquin Pastor-Fernández, Antonius Adrianus Hendrikus Petrus Megens +4 more |
2007-01-30 |
| 7081453 |
Compounds for treating impaired fundic relaxation |
Kristof Van Emelen, Marcel Frans Leopold De Bruyn, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea, Maria Encarnacion Matesanz-Ballesteros +1 more |
2006-07-25 |