Issued Patents All Time
Showing 25 most recent of 70 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 9440952 | Compounds inhibiting leucine-rich repeat kinase enzyme activity | Michael Miller, Kallol Basu, Duane DeMong, Jack D. Scott, Hong Liu +9 more | 2016-09-13 |
| 8822480 | Bicyclic heterocycle derivatives and use thereof as GPR119 modulators | Santhosh F. Neelamkavil, Craig D. Boyle, Samuel Chackalamannil, William J. Greenlee, Andrew Stamford | 2014-09-02 |
| 8815876 | Bicyclic heterocycle derivatives and methods of use thereof | Santhosh F. Neelamkavil, Craig D. Boyle, Samuel Chackalamannil, William J. Greenlee | 2014-08-26 |
| 8722882 | Pyrimidine derivatives as GPCR modulators for use in the treatment of obesity and diabetes | Andrew Stamford, Jinsong Hao, Charles Lee Jayne, Yan Xia | 2014-05-13 |
| 8435994 | Substituted [1,2,4]triazolo[4,3-alpha]quinoxalines as adenosine A2a receptor antagonists | Joel M. Harris, Andrew Stamford | 2013-05-07 |
| RE44205 | Adenosine A2a receptor antagonists | Neil A. Lindo, William J. Greenlee, Deen Tulshian, Lisa S. Silverman, Yan Xia +2 more | 2013-05-07 |
| 8415353 | Amino-quinoxaline and amino-quinoline compounds for use as adenosine A2a receptor antagonists | Joel M. Harris, Hong Liu, Jinsong Hao, Andrew Stamford | 2013-04-09 |
| 8410122 | Bicyclic heterocycle derivatives and methods of use thereof | Joel M. Harris, Andrew Stamford, Hong Liu | 2013-04-02 |
| 8318751 | Pyrimidinone derivatives and methods of use thereof | Craig D. Boyle, Samuel Chackalamannil, Claire M. Lankin, Unmesh Shah, Hong Liu +1 more | 2012-11-27 |
| 8222259 | 1,2,4-triazolo[4,3-c]pyrimidin-3-one and pyrazolo[4,3-e]-1,2,4-triazolo[4,3-c]pyrimidin-3-one compounds for use as adenosine A2a receptor antagonists | Joel M. Harris, Jinsong Hao, Andrew Stamford | 2012-07-17 |
| 8114879 | Piperazine derivatives useful as CCR5 antagonists | Bahige M. Baroudy, John W. Clader, Hubert Josien, Stuart W. McCombie, Brian McKittrick +9 more | 2012-02-14 |
| 7790474 | p53 modulators | Bimalendu Dasmahapatra, Mark Demma, Alan K. Mallams, Henry A. Vaccaro, Jonathan A. Pachter | 2010-09-07 |
| 7741318 | Pyrazolo [1,5-A]pyrimidine adenosine A2a receptor antagonists | Martin C. Clasby, Samuel Chackalamannil, Xiaobang Gao | 2010-06-22 |
| 7709492 | Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists | Jinsong Hao, Hong Liu, Craig D. Boyle, Samuel Chackalamannil, Unmesh Shah +2 more | 2010-05-04 |
| 7465740 | 2-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists | Craig D. Boyle, Samuel Chackalamannil, Joel M. Harris, Claire M. Lankin, Hong Liu +2 more | 2008-12-16 |
| 7384944 | Piperazine derivatives useful as CCR5 antagonists | Bahige M. Baroudy, John W. Clader, Hubert Josien, Stuart W. McCombie, Brian McKittrick +9 more | 2008-06-10 |
| 7368449 | 2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists | Jinsong Hao, Hong Liu, Craig D. Boyle, Samuel Chackalamannil, Unmesh Shah +1 more | 2008-05-06 |
| 7078408 | [1,2,4]-Triazole bicyclic adenosine A2a receptor antagonists | Hong Liu | 2006-07-18 |
| 7067655 | Adenosine A2a receptor antagonists | Neil A. Lindo | 2006-06-27 |
| 7041666 | Adenosine A2a receptor antagonists | Julius J. Matasi, John P. Caldwell, Deen Tulshian, Lisa S. Silverman | 2006-05-09 |
| 6897217 | 2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists | Jinsong Hao, Hong Liu, Craig D. Boyle, Samuel Chackalamannil, Unmesh Shah +1 more | 2005-05-24 |
| 6897216 | Adenosine A2a receptor antagonists | Neil A. Lindo, William J. Greenlee, Deen Tulshian, Lisa S. Silverman, Yan Xia +2 more | 2005-05-24 |
| 6875772 | [1,2,4]-Triazole bicyclic adeonsine A2a receptor antagonists | Hong Liu | 2005-04-05 |
| 6689765 | Piperazine derivatives useful as CCR5 antagonists | Bahige M. Baroudy, John W. Clader, Hubert Josien, Stuart W. McCombie, Brian McKittrick +9 more | 2004-02-10 |
| 6630475 | Adenosine A2a receptor antagonists | Neil A. Lindo, William J. Greenlee, Deen Tulshian, Lisa S. Silverman, Yan Xia +2 more | 2003-10-07 |