| 12509447 |
Small molecule compound |
Guanqun Li, Xinyu Wang, Yufeng Cai, Xiang Jiang, Xianfeng Pan +3 more |
2025-12-30 |
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| 12384795 |
Pyrimido[5,4-b]pyrrolizin compound, optical isomer thereof, preparation method therefor and use thereof |
Ao Zhang, Jian Ding, Hua Xie, Zilan Song, Yu-Yi Xue +2 more |
2025-08-12 |
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| 12129256 |
Pyrazolo[1,5-a]pyrazin-4-yl derivatives |
Matthew Frank Brown, Alpay Dermenci, Andrew Fensome, Brian Stephen Gerstenberger, Matthew Merrill Hayward +3 more |
2024-10-29 |
$505,385,000 |
| 11834432 |
Substituted amino six-membered nitric heterocyclic ring compound and preparation and use thereof |
Ao Zhang, Meiyu Geng, Jing Ai, Zilan Song, Xia Peng +2 more |
2023-12-05 |
|
| 11472809 |
Pyrazolo[1,5-a]pyrazin-4-yl derivatives |
Matthew Frank Brown, Alpay Dermenci, Andrew Fensome, Brian Stephen Gerstenberger, Matthew Merrill Hayward +3 more |
2022-10-18 |
$393,425,000 |
| 11254668 |
Pyrazolo[1,5-A]pyrazin-4-yl and related derivatives |
Brian Stephen Gerstenberger, Andrew Fensome, Dafydd Rhys Owen, Matthew Frank Brown, Matthew Merrill Hayward +2 more |
2022-02-22 |
$482,573,000 |
| 11197867 |
Aminopyrimidinyl compounds |
Andrew Fensome, Ariamala Gopalsamy, Brian Stephen Gerstenberger, Ivan Viktorovich Efremov, Zhao-Kui Wan +5 more |
2021-12-14 |
$1,320,244,000 |
| 11001592 |
DNA polymerase IIIC inhibitors and use thereof |
Xiang Yu, Minghua Wang, Casey Cameron McComas, Michael SILVERMAN, Richard Soll |
2021-05-11 |
|
| 10980815 |
Aminopyrimidinyl compounds |
Andrew Fensome, Ariamala Gopalsamy, Brian Stephen Gerstenberger, Ivan Viktorovich Efremov, Zhao-Kui Wan +5 more |
2021-04-20 |
$674,734,000 |
| 10836772 |
DNA polymerase IIIC inhibitors and use thereof |
Xiang Yu, Minghua Wang, Casey Cameron McComas, Michael SILVERMAN, Richard Soll |
2020-11-17 |
|
| 10822341 |
Pyrazolo[1,5-a]pyrazin-4-yl derivatives |
Matthew Frank Brown, Alpay Dermenci, Andrew Fensome, Brian Stephen Gerstenberger, Matthew Merrill Hayward +3 more |
2020-11-03 |
$385,583,000 |
| 10815213 |
Bruton's tyrosine kinase inhibitors |
John Robert Springer, Balekudru Devadas, Danny James Garland, Margaret L. Grapperhaus, Seungil Han +9 more |
2020-10-27 |
$309,700,000 |
| 10723741 |
DNA polymerase IIIC inhibitors and use thereof |
Xiang Yu, Minghua Wang, Casey Cameron McComas, Michael SILVERMAN, Richard Soll |
2020-07-28 |
|
| 10493129 |
Use of fibroblast growth factor 2 |
Xiliang Wang, Chengyu JIANG, Penghui Yang, Xin Liu, Yueqiang Duan +1 more |
2019-12-03 |
|
| 10463675 |
Aminopyrimidinyl compounds |
Andrew Fensome, Ariamala Gopalsamy, Brian Stephen Gerstenberger, Ivan Viktorovich Efremov, Zhao-Kui Wan +5 more |
2019-11-05 |
$427,991,000 |
| 10426135 |
Methyl- and trifluromethyl-substituted pyrrolopyridine modulators of RORC2 and methods of use thereof |
Mark Edward Schnute, Andrew Christopher Flick, Peter Jones, Neelu Kaila, Scot Richard Mente +6 more |
2019-10-01 |
$298,967,000 |
| 10385036 |
Sulfonamide-substituted indole modulators of RORC2 and methods of use thereof |
Mark Edward Schnute, Andrew Christopher Flick, Peter Jones, Neelu Kaila, Scot Richard Mente +6 more |
2019-08-20 |
$837,148,000 |
| 10336748 |
Methyoxy-substituted pyrrolopyridine modulators of RORC2 and methods of use thereof |
Mark Edward Schnute, Andrew Christopher Flick, Peter Jones, Neelu Kaila, Scot Richard Mente +6 more |
2019-07-02 |
$980,917,000 |
| 10308615 |
Heterocyclic compounds as inhibitors of Vanin-1 enzyme |
Agustin Casimiro-Garcia, Jeffrey Scott Condon, Andrew Christopher Flick, Ariamala Gopalsamy, Steven J. Kirincich +4 more |
2019-06-04 |
$869,926,000 |
| 10266513 |
Bruton's tyrosine kinase inhibitors |
John Robert Springer, Balekudru Devadas, Danny James Garland, Margaret L. Grapperhaus, Seungil Han +9 more |
2019-04-23 |
$877,937,000 |
| 10227346 |
Methyl- and trifluoromethyl-substituted pyrrolopyridine modulators of RORC2 and methods of use therof |
Mark Edward Schnute, Andrew Christopher Flick, Peter Jones, Neelu Kaila, Scot Richard Mente +6 more |
2019-03-12 |
$419,848,000 |
| 10144738 |
Pyrazolo[1,5-A]PYRAZIN-4-YL derivatives |
Matthew Frank Brown, Alpay Dermenci, Andrew Fensome, Brian Stephen Gerstenberger, Matthew Merrill Hayward +3 more |
2018-12-04 |
$489,814,000 |
| 9670201 |
Methyl- and trifluoromethyl-substituted pyrrolopyridine modulators of RORC2 and methods of use thereof |
Mark Edward Schnute, Andrew Christopher Flick, Peter Jones, Neelu Kaila, Scot Richard Mente +5 more |
2017-06-06 |
$303,831,000 |
| 9663526 |
Aminopyrimidinyl compounds |
Andrew Fensome, Ariamala Gopalsamy, Brian Stephen Gerstenberger, Ivan Viktorovich Efremov, Zhao-Kui Wan +5 more |
2017-05-30 |
$667,472,000 |
| 9284283 |
Macrocyclic compounds for modulating IL-17 |
Michael D. Taylor, Nicholas K. Terrett, William H. Connors, Cheri Snedeker, Kelley C. Shortsleeves +8 more |
2016-03-15 |
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