Patent Leaderboard
USPTO Patent Rankings Data through Dec 31, 2025
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Malcolm MacCoss — 117 Patents

Merck: 103 patents #14 of 9,382Top 1%
USUcb Biopharma Srl: 9 patents #33 of 349Top 10%
CPCardurion Pharmaceuticals: 2 patents #8 of 59Top 15%
SASanofi: 2 patents #699 of 1,881Top 40%
PTPtc Therapeutics: 2 patents #88 of 160Top 60%
IPIsis Pharmaceuticals: 2 patents #179 of 400Top 45%
SISouthern Research Institute: 1 patents #135 of 244Top 60%
DEDepartment Of Energy: 1 patents #41 of 740Top 6%
Seabrook Island, SC: #1 of 3 inventorsTop 35%
South Carolina: #16 of 15,501 inventorsTop 1%
Overall (All Time): #10,533 of 4,157,543Top 1%
117 Patents All Time
Malcolm MacCoss has been granted 117 US patents while listed as an inventor at Merck. The first was granted in 1984 and the most recent in February 2024. Malcolm MacCoss ranks #10,533 of 4,157,543 US inventors in our database (top 0.25%). Patent records list Malcolm MacCoss in Seabrook Island, SC, US.

Issued Patents All Time

Showing 1–25 of 117 patents

Patent #TitleCo-InventorsDateApprox Value ⓘ
11912721 Fused pentacyclic imidazole derivatives Teresa De Haro Garcia, Michael Deligny, Jag Paul Heer, Joanna Rachel Quincey, Mengyang Xuan +14 more 2024-02-27 $28,908,000
11795172 Substituted imidazo[1,2-b]pyridazines and [1,2,4]triazolo[4,3-b]pyridazines as CaMKII inhibitors Nobuyuki Matsunaga, Junya Shirai, Tomohiro Okawa, Yasufumi Miyamoto, Zenyu Shiokawa +3 more 2023-10-24
11479546 Antimalarial hexahydropyrimidine analogues Teresa De Haro Garcia, Lloyd Malcolm King, Martin Alexander Lowe, Richard David Taylor, Zhaoning Zhu 2022-10-25
11136310 Iminotetrahydropyrimidinone derivatives as plasmepsin V inhibitors Rebecca Louise Charlton, Teresa De Haro Garcia, Martin Alexander Lowe, Trevor Morgan, Richard David Taylor +1 more 2021-10-05
11130752 Aminopyrimidine compound Nobuyuki Matsunaga, Yasufumi Miyamoto, Junya Shirai, Takashi Nakahata, Zenyu Shiokawa +2 more 2021-09-28
11091474 Alkoxy bis-heteroaryl derivatives as modulators of protein aggregation Adrian Hall 2021-08-17
10980814 Fused pentacyclic imidazole derivatives as modulators of TNF activity Daniel Christopher Brookings, Teresa De Haro Garcia, Yann Foricher, Helen Tracey Horsley, Martin Clive Hutchings +3 more 2021-04-20 $33,688,000
10975066 Bis-heteroaryl derivatives as modulators of protein aggregation Wolfgang Wrasidlo, Emily M. Stocking, Adrian Hall 2021-04-13
10889584 Bicyclic bis-heteroaryl derivatives as modulators of protein aggregation Adrian Hall, Laurent Provins 2021-01-12
10464932 Iminothiadiazinane dioxide derivatives as plasmepsin V inhibitors Teresa De Haro Garcia, Martin Alexander Lowe, Richard David Taylor, Zhaoning Zhu 2019-11-05
10087179 Fused tricyclic imidazole derivatives as modulators of TNF activity Rikki Peter Alexander, Gareth Neil Brace, Julien Alistair Brown, Mark Daniel Calmiano, Prafulkumar Tulshibhai Chovatia +11 more 2018-10-02
9593108 Compounds and methods for antiviral treatment F. George Njoroge, Amin Nomeir, Guangming Chen, Gary Mitchell Karp, William Jospeh Lennox +6 more 2017-03-14 $11,490,000
9433621 Substituted pyridine and pyrimidine derivatives and their use in treating viral infections Ashok Arasappan, F. George Njoroge, Cecil D. Kwong, Subramaniam Ananthan, Frank Bennett +15 more 2016-09-06 $101,652,000
8859776 Substituted piperidines that increase p53 activity and the uses thereof Stephane L. Bogen, Yao-Dong Ma, Yaolin Wang, Brian Robert Lahue, Latha G. Nair +15 more 2014-10-14 $39,553,000
8809318 Gamma secretase modulators Zhaoning Zhu, William J. Greenlee, Hongmei Li, Monica L. Vicarel, Jun Qin +11 more 2014-08-19 $104,285,000
8735414 Indole derivatives and methods for antiviral treatment F. George Njoroge, Amin Nomeir, Guangming Chen, Song Huang, Ramesh Kakarla +14 more 2014-05-27 $13,443,000
8440668 Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment of type 2 diabetes Scott D. Edmondson, Michael H. Fisher, Dooseop Kim, Emma R. Parmee, Ann E. Weber +1 more 2013-05-14 $107,206,000
8168637 Beta-amino heterocyclic dipeptidyl peptidase inhibitors for the treatment of diabetes Scott D. Edmondson, Dooseop Kim, Emma R. Parmee, Ann E. Weber, Jinyou Xu 2012-05-01 $48,747,000
7879815 Nucleoside aryl phosphoramidates for the treatment of RNA-dependent RNA viral infection David B. Olsen, Monica Donghi, Cristina Gardelli, Steven Harper, Malte Meppen +2 more 2011-02-01 $44,131,000
7632821 Ribonucleoside cyclic acetal derivatives for the treatment of RNA-dependent RNA viral infection Gabor Butora, Kenneth Alan Koeplinger, Daniel R. McMasters, David B. Olsen, Lihu Yang 2009-12-15 $106,751,000
7534767 C-purine nucleoside analogs as inhibitors of RNA-dependent RNA viral polymerase Gabor Butora, Balkrishen Bhat, Anne B. Eldrup 2009-05-19 $73,688,000
7125887 Pyrrolidine modulators of CCR5 chemokine receptor activity Jeffrey J. Hale, Charles G. Caldwell, Dooseop Kim, Dong-Ming Shen, Sander G. Mills +5 more 2006-10-24 $43,547,000
7125873 Beta-amino tetrahydroimidazo (1, 2-a) pyrazines and tetrahydrotrioazolo (4, 3-a) pyrazines as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes Scott D. Edmondson, Michael H. Fisher, Dooseop Kim, Emma R. Parmee, Ann E. Weber +1 more 2006-10-24 $43,547,000
7125855 Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Balkrishen Bhat, Neelima M. Bhat, Anne B. Eldrup, Thazha P. Prakash, Marija Prhavc +4 more 2006-10-24 $43,547,000
7105499 Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Steven Carroll, David B. Olsen, Balkrishen Bhat, Phillip Dan Cook, Anne B. Eldrup +1 more 2006-09-12