GD

Gaston Stanislas Marcella Diels

📍 Turnhout, BE: #3 of 146 inventorsTop 3%
Overall (All Time): #75,414 of 4,157,543Top 2%
41
Patents All Time

Issued Patents All Time

Showing 1–25 of 41 patents

Patent #TitleCo-InventorsDate
12404260 Pyridine rings containing derivatives as MALT1 inhibitors Johannes Wilhelmus John F. Thuring, Tianbao Lu, Tongfei Wu, Didier Jean-Claude Berthelot, Berthold Wroblowski 2025-09-02
12077521 Pyrazole derivatives as MALT1 inhibitors Tianbao Lu, Brett D. Allison, Joseph Kent Barbay, Peter J. Connolly, Maxwell D. Cummings +7 more 2024-09-03
11993614 Monocyclic and bicyclic ring system substituted carbanucleoside analogues for use as PRMT5 inhibitors Tongfei Wu, Dirk Brehmer, Lijs Beke, An Boeckx, Edward C. Lawson +7 more 2024-05-28
11883367 6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors Tongfei Wu, Dirk Brehmer, Lijs Beke, An Boeckx, Ronaldus Arnodus Hendrika Joseph Gilissen +8 more 2024-01-30
11318157 6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors Tongfei Wu, Dirk Brehmer, Lijs Beke, An Boeckx, Ronaldus Arnodus Hendrika Joseph Gilissen +8 more 2022-05-03
11098062 Monocyclic and bicyclic ring system substituted carbanucleoside analogues for use as PRMT5 inhibitors Tongfei Wu, Dirk Brehmer, Lijs Beke, An Boeckx, Edward C. Lawson +7 more 2021-08-24
11040031 Pyrazole derivatives as MALT1 inhibitors Tianbao Lu, Peter J. Connolly, Maxwell D. Cummings, Joseph Kent Barbay, Kevin D. Kreutter +5 more 2021-06-22
10954214 Pyrazole derivatives as MALT1 inhibitors Tianbao Lu, Brett D. Allison, Joseph Kent Barbay, Peter J. Connolly, Maxwell D. Cummings +7 more 2021-03-23
10898504 Substituted nucleoside analogues for use as PRMT5 inhibitors Didier Jean-Claude Berthelot, Dirk Brehmer, Lijs Beke, An Boeckx, Ronaldus Arnodus Hendrika Joseph Gilissen +10 more 2021-01-26
10888550 Pyrazole derivatives as MALT1 inhibitors Tianbao Lu, Peter J. Connolly, Maxwell D. Cummings, Jan Willem Thuring, Ulrike PHILIPPAR +3 more 2021-01-12
10653711 6-6 bicyclic aromatic ring substituted nucleoside analogues for use as PRMT5 inhibitors Tongfei Wu, Dirk Brehmer, Lijs Beke, An Boeckx, Ronaldus Arnodus Hendrika Joseph Gilissen +8 more 2020-05-19
10017509 Macrocylic pyrimidine derivatives Bruno Schoentjes, Matthias VERSELE, Didier Jean-Claude Berthelot, Marc Willems, Marcel Viellevoye +3 more 2018-07-10
9273013 Quinazoline derivatives Eddy Jean Edgard Freyne, Timothy Pietro Suren Perera, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Werner Constant Johan Embrechts +3 more 2016-03-01
8394786 Quinazoline derivatives Eddy Jean Edgard Freyne, Timothy Pietro Suren Perera, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Werner Constant Johan Embrechts +3 more 2013-03-12
7648975 Macrocyclic quinazoline derivatives as antiproliferative agents Eddy Jean Edgard Freyne, Timothy Pietro Suren Perera, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Werner Constant Johan Embrechts 2010-01-19
7514445 Heteroaryl amines as glycogen synthase kinase 3β inhibitors (GSK3 inhibitors) Eddy Jean Edgard Freyne, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Werner Constant Johan Embrechts, Christopher John Love +7 more 2009-04-07
7410970 Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists Frans Eduard Janssens, François Maria Sommen, Benoît Christian Albert Ghislain De Boeck, Joseph Elisabeth Leenaerts, Yves Emiel Maria Van Roosbroeck 2008-08-12
7138403 2,4,5-trisubstituted thiazolyl derivatives and their antiinflammatory activity Christopher John Love, Jean Pierre Frans Van Wauwe, Marc De Brabander, Roger Clive Moses, Mykhalyo Goncharenko +4 more 2006-11-21
6951857 6-Azauracil derivatives as IL-5 inhibitors Eddy Jean Edgard Freyne, Gustaaf Maria Boeckx, Jean Pierre Frans Van Wauwe 2005-10-04
6743792 6-azauracil derivatives as IL-5 inhibitors Eddy Jean Edgard Freyne, Gustaaf Maria Boeckx, Jean Pierre Frans Van Wauwe 2004-06-01
6656959 PDE IV inhibiting pyridine derivatives Eddy Jean Edgard Freyne, Maria Encarnacion Matesanz-Ballesteros, Adolfo Diaz-Martinez 2003-12-02
6403805 1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one derivatves Eddy Jean Edgard Freyne, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea 2002-06-11
5994376 1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one compounds and their use for treating allergic, atopic or inflammatory diseases Eddy Jean Edgard Freyne, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea 1999-11-30
5952510 1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives having PDE IV and cytokine inhibiting activity Eddy Jean Edgard Freyne, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea 1999-09-14
5869515 1,3-dihydro-2H-imidazol-2-one compounds Eddy Jean Edgard Freyne, José Ignacio Andrés-Gil, Francisco Javier Fernandez-Gadea 1999-02-09