| 10519137 |
Pyrazolyl quinoxaline kinase inhibitors |
Gordon Saxty, Christopher William Murray, Valerio Berdini, Gilbert Ebai Besong, Steven John Woodhead +12 more |
2019-12-31 |
| 10208062 |
Macrocyclic quinazole derivatives and their use as MTKI |
Marc Willems, Peter Ten Holte, Alexandra Papanikos, Werner Constant Johan Embrechts, Pierre-Henri Storck +1 more |
2019-02-19 |
| 9850228 |
Pyrazolyl quinoxaline kinase inhibitors |
Gordon Saxty, Christopher William Murray, Valerio Berdini, Gilbert Ebai Besong, Christopher Charles Frederick Hamlett +20 more |
2017-12-26 |
| 9688691 |
Macrocyclic quinazole derivatives and their use as MTKI |
Marc Willems, Peter Ten Holte, Alexandra Papanikos, Werner Constant Johan Embrechts, Pierre-Henri Storck +1 more |
2017-06-27 |
| 9464071 |
Pyrazolyl quinoxaline kinase inhibitors |
Gordon Saxty, Christopher William Murray, Valerio Berdini, Gilbert Ebai Besong, Christopher Charles Frederick Hamlett +20 more |
2016-10-11 |
| 9365517 |
3-cyano-quinoline derivatives with antiproliferative activity |
Peter Jacobus Johannes Antonius Buijnsters, Kristof Van Emelen, Werner Constant Johan Embrechts, Timothy Pietro Suren Perera |
2016-06-14 |
| 9273013 |
Quinazoline derivatives |
Timothy Pietro Suren Perera, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Gaston Stanislas Marcella Diels, Werner Constant Johan Embrechts +3 more |
2016-03-01 |
| 9040511 |
3-cyano-quinoline derivatives with antiproliferative activity |
Peter Jacobus Johannes Antonius Buijnsters, Kristof Van Emelen, Werner Constant Johan Embrechts, Timothy Pietro Suren Perera |
2015-05-26 |
| 8933067 |
Pyrido and pyrimidopyrimidine derivatives as anti-profilerative agents |
Marc Willems, Pierre-Henri Storck, Virginie Sophie Poncelet, Kristof Van Emelen, Peter Jacobus Johannes Antonius +2 more |
2015-01-13 |
| 8895601 |
Pyrazolyl quinoxaline kinase inhibitors |
Gordon Saxty, Christopher William Murray, Valerio Berdini, Gilbert Ebai Besong, Christopher Charles Frederick Hamlett +17 more |
2014-11-25 |
| 8796244 |
Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases |
Valerio Berdini, Maria Grazia Carr, Miles Stuart Congreve, Martyn Frederickson, Charlotte Mary Griffiths-Jones +11 more |
2014-08-05 |
| 8778966 |
Quinolinone derivatives as PARP and tank inhibitors |
Jorge Eduardo Vialard, Patrick René Angibaud, Laurence Anne Mevellec, Christophe Meyer, Isabelle Noëlle Constance Pilatte +10 more |
2014-07-15 |
| 8778920 |
3-cyano-quinoline derivatives with antiproliferative activity |
Peter Jacobus Johannes Antonius Buijnsters, Kristof Van Emelem, Werner Constant Johan Embrechts, Timothy Pietro Suren Perera |
2014-07-15 |
| 8772272 |
Pyrido-and pyrimidopyrimidine derivatives as anti-proliferative agents |
Marc Willems, Pierre-Henri Storck, Virginie Sophie Poncelet, Kristof Van Emelen, Peter Jacobus Johannes Antonius Buijnsters +2 more |
2014-07-08 |
| 8722687 |
Imidazo [1,2-A]pyridine derivatives as FGFR kinase inhibitors for use in therapy |
Gordon Saxty, Valerio Berdini, Christopher William Murray, Yannick Aime Eddy Ligny, Pascal Bonnet +2 more |
2014-05-13 |
| 8492377 |
MTKI quinazoline derivatives |
Alexandra Papanikos, Peter Ten Holte, Marc Willems, Werner Constant Johan Embrechts, Laurence Anne Mevellec +1 more |
2013-07-23 |
| 8481531 |
Bicyclic heterocyclyl derivatives as FGFR kinase inhibitors for therapeutic use |
Gordon Saxty, Valerio Berdini, Alexandra Papanikos, Pascal Benderitter, Werner Constant Johan Embrechts +2 more |
2013-07-09 |
| 8476289 |
Aza-bicyclohexyl substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylace |
Isabelle Noëlle Constance Pilatte, Patrick René Angibaud |
2013-07-02 |
| 8394786 |
Quinazoline derivatives |
Timothy Pietro Suren Perera, Peter Jacobus Johannes Antonius Buijnsters, Marc Willems, Gaston Stanislas Marcella Diels, Werner Constant Johan Embrechts +3 more |
2013-03-12 |
| 8394955 |
2,4 (4,6) pyrimidine derivatives |
Marc Willems, Werner Constant Johan Embrechts, Kristof Van Emelen, Sven Franciscus Anna Van Brandt, Frederik Jan Rita Rombouts |
2013-03-12 |
| 8318731 |
Pyrrolopyrimidines |
Gaston Stanislas Marcella Diels, Peter Ten Holte, Thierry Andre Regis Grand-Perret, Kristof Van Emelen, Werner Constant Johan Embrechts +1 more |
2012-11-27 |
| 8299256 |
Quinolinone derivatives as PARP and TANK inhibitors |
Jorge Eduardo Vialard, Patrick René Angibaud, Laurence Anne Mevellec, Christophe Meyer, Isabelle Noëlle Constance Pilatte +10 more |
2012-10-30 |
| 8168644 |
Quinazolinone derivatives as tubulin polymerization inhibitors |
Laurence Anne Mevellec, Jorge Eduardo Vialard, Christophe Meyer, Elisabeth Therese Jeanne Pasquier, Xavier Marc Bourdrez +1 more |
2012-05-01 |
| 8148388 |
2,4 (4,6) pyrimidine derivatives |
Marc Willems, Werner Constant Johan Embrechts, Kristof Van Emelen, Sven Franciscus Anna Van Brandt, Frederik Jan Rita Rombouts |
2012-04-03 |
| 7947695 |
5-membered annelated heterocyclic pyrimidines as kinase inhibitors |
Jean Fernand Armand Lacrampe, Timothy Pietro Suren Perera, Peter Ten Holte, Yannick Aime Eddy Ligny, Delphine Yvonne Raymonde Lardeau +1 more |
2011-05-24 |