Issued Patents All Time
Showing 1–25 of 30 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12263164 | Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2025-04-01 |
| 11820777 | Crystal forms of (s)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Edwin Aret, Cecile M. Krejsa, Jerry Evarts | 2023-11-21 |
| 11771696 | Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2023-10-03 |
| 11654143 | Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor, a JAK-2 inhibitor, and/or a BCL-2 inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2023-05-23 |
| 11166951 | Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor, a JAK-2 inhibitor, and/or a BCL-2 inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2021-11-09 |
| 11110088 | Imidazopyrazine inhibitors of Bruton's tyrosine kinase | Edwin de Zwart, Saskia Verkaik, Niels Hoogenboom, Dennis Demont | 2021-09-07 |
| 11090302 | Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2021-08-17 |
| 11059829 | Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide maleate | Fritz Blatter, Tim Ingallinera, Edwin Aret, Cecile M. Krejsa, Jerry Evarts | 2021-07-13 |
| 10934296 | 4-imidazopyridazin-1-yl-benzamides as Btk inhibitors | Christiaan Gerardus Johannes Maria Jans, Adrianus Petrus Antonius De Man, Arthur A. Oubrie, Hans C. A. Raaijmakers, Johannes Bernardus Maria Rewinkel +2 more | 2021-03-02 |
| 10736893 | Imidazopyrazine inhibitors of Bruton's tyrosine kinase | Edwin de Zwart, Saskia Verkaik, Niels Hoogenboom, Dennis Demont | 2020-08-11 |
| 10640509 | Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide for treating diffuse large B-cell lymphoma | Fritz Blatter, Tim Ingallinera, Edwin Aret, Cecile M. Krejsa, Jerry Evarts | 2020-05-05 |
| 10328080 | Therapeutic combination of PI3K inhibitor and a BTK inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2019-06-25 |
| 10272083 | Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2019-04-30 |
| 10239883 | 4-imidazopyridazin-1-yl-benzamides as BTK inhibitors | Christiaan Gerardus Johannes Maria Jans, Adrianus Petrus Antonius De Man, Arthur A. Oubrie, Hans C. A. Raaijmakers, Johannes Bernardus Maria Rewinkel +2 more | 2019-03-26 |
| 10167291 | Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl) pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Edwin Aret, Cecile M. Krejsa, Jerry Evarts | 2019-01-01 |
| 9949971 | Therapeutic combinations of a BTK inhibitor, a PI3K inhibitor and/or a JAK-2 inhibitor | Ahmed Hamdy, Wayne Rothbaum, Raquel Izumi, Brian Lannutti, Todd Covey +3 more | 2018-04-24 |
| 9796721 | Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Edwin Aret, Cecile M. Krejsa, Jerry Evarts | 2017-10-24 |
| 9790226 | 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as BtK inhibitors | Christiaan Gerardus Johannes Maria Jans, Adrianus Petrus Antonius De Man, Arthur A. Oubrie, Hans C. A. Raaijmakers, Johannes Bernardus Maria Rewinkel +2 more | 2017-10-17 |
| 9758524 | 4-imidazopyridazin-1-yl-benzamides as Btk inhibitors | Christiaan Gerardus Johannes Maria Jans, Adrianus Petrus Antonius De Man, Arthur A. Oubrie, Hans C. A. Raaijmakers, Johannes Bernardus Maria Rewinkel +2 more | 2017-09-12 |
| 9718828 | BTK Inhibitors | Adrianus Petrus Antonius De Man, Jan Gerard Sterrenburg, Hans C.A. Raaijmakers, Allard Kaptein, Arthur A. Oubrie +18 more | 2017-08-01 |
| 9290504 | 4-imidazopyridazin-1-yl-benzamides and 4-imidazotriazin-1-yl-benzamides as Btk inhibitors | Christiaan Gerardus Johannes Maria Jans, Petrus Antonius De Adrianus Man, Arthur A. Oubrie, Hans C. A. Raaijmakers, Johannes Bernardus Maria Rewinkel +2 more | 2016-03-22 |
| 9102676 | MK2 inhibitors | Arthur A. Oubrie, Carsten Schultz-Fadermrecht, Eduard Willem Zwart, Niels Hoogenboom, Sander Martijn De Wilde +1 more | 2015-08-11 |
| 8772286 | MK2 inhibitors | Arthur A. Oubrie, Carsten Schultz-Fademrecht, Eduard Willem Zwart, Niels Hoogenboom, Sander Martijn De Wilde +1 more | 2014-07-08 |
| 7671051 | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 | Rikard Emond, Jerk Vallgarda, Guido Kurz, Marianne Nilsson, Lian Zhang | 2010-03-02 |
| 7618961 | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 | Rikard Emond, Guido Kurz, Jerk Vallgarda, Marianne Nilsson | 2009-11-17 |