| 12286400 |
Isofagomine salts, methods of use and formulations |
Helge Alfred Reisch, Jeffrey S. DePue, Jennifer Robin, Michael Hahn, Gaozhong Zhu +1 more |
2025-04-29 |
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| 12221445 |
Crystalline salts of 5-methyl-(6S)-tetrahydrofolic acid and amino ethyl esters |
Rudolf Moser, Viola Groehn, Ruth Boehni Stamm, Martin Szelagiewicz |
2025-02-11 |
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| 12221446 |
Crystalline salt of 5-methyl-(6S)-tetrahydrofolic acid and L-isoleucine ethyl ester |
Rudolf Moser, Viola Groehn, Ruth Boehni Stamm, Martin Szelagiewicz |
2025-02-11 |
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| 12116344 |
Crystalline forms of a pharmaceutical compound |
Robert Hett, Jennifer Robin, Kyle Landskroner |
2024-10-15 |
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| 12048700 |
Crystalline monosodium salt of 5-methyl-(6S)-tetrahydrofolic acid |
Rudolf Moser, Viola Groehn, Martin Szelagiewicz, Ruth Boehni Stamm, Markus Ruettimann +1 more |
2024-07-30 |
$232,799,000 |
| 11992491 |
Crystalline salts of 5-methyl-(6S)-tetrahydrofolic acid and L-valine ethyl ester |
Rudolf Moser, Viola Groehn, Ruth Boehni Stamm, Martin Szelagiewicz |
2024-05-28 |
$153,549,000 |
| 11925644 |
Crystalline salts of 5-methyl-(6S)-tetrahydrofolic acid and l-leucine ethyl ester |
Rudolf Moser, Viola Groehn, Ruth Boehni Stamm, Martin Szelagiewicz |
2024-03-12 |
$345,937,000 |
| 11820777 |
Crystal forms of (s)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide |
Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa, Jerry Evarts |
2023-11-21 |
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| 11633400 |
Crystalline salt comprising 5-methyl-(6S)-tetrahydrofolic acid and 4-(2-hydroxyethyl)-morpholine |
Rudolf Moser, Viola Groehn, Ruth Boehni Stamm, Martin Szelagiewicz |
2023-04-25 |
$617,771,000 |
| 11377448 |
Crystalline sodium salt of 5-methyl-(6S)-tetrahydrofolic acid |
Rudolf Moser, Viola Groehn, Martin Szelagiewicz, Ruth Boehni Stamm, Markus Ruettimann |
2022-07-05 |
$309,260,000 |
| 11185545 |
Crystalline monosodium salt of 5-methyl-(6S)-tetrahydrofolic acid |
Rudolf Moser, Viola Groehn, Martin Szelagiewicz, Ruth Boehni Stamm, Markus Ruettimann +1 more |
2021-11-30 |
$230,654,000 |
| 11129820 |
Ferroportin-inhibitor salts |
Collin D. Morris, Giuseppe Lapadula, Stefan Reim, Michael Burgert, Erik Philipp |
2021-09-28 |
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| 11066408 |
Crystalline binary sodium salts of 5-methyl-(6S)-tetrahydrofolic acid with organic bases |
Rudolf Moser, Viola Groehn, Martin Szelagiewicz, Ruth Boehni Stamm, Markus Ruettimann +1 more |
2021-07-20 |
$167,720,000 |
| 11059829 |
Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide maleate |
Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa, Jerry Evarts |
2021-07-13 |
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| 10640509 |
Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide for treating diffuse large B-cell lymphoma |
Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa, Jerry Evarts |
2020-05-05 |
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| 10167291 |
Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl) pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide |
Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa, Jerry Evarts |
2019-01-01 |
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| 10045998 |
Solid form of abiraterone acetate |
Tiziana Chiodo, Beate Salvador, Marcus Vossen, Andreas Hafner, Tobias Hintermann +3 more |
2018-08-14 |
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| 9993481 |
Methods and compositions for the treatment of metabolic disorders |
Daniel I. Oppenheimer, Emil D. Kakkis, Fredric D. Price, Alejandro Dorenbaum, Rudolf Moser +2 more |
2018-06-12 |
$98,548,000 |
| 9884857 |
Salts of dasatinib in amorphous form |
Andreas Hafner, Martin Szelagiewicz, Bernd Siebenhaar, Tiziana Chiodo, Tobias Hintermann +2 more |
2018-02-06 |
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| 9796721 |
Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide |
Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa, Jerry Evarts |
2017-10-24 |
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| 9567317 |
Multicomponent crystalline system comprising nilotinib and selected co-crystal formers |
Tiziana Chiodo, Andreas Hafner, Tobias Hintermann, Beate Salvador, Martin Szelagiewicz +2 more |
2017-02-14 |
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| 9556164 |
Salts of Dasatinib in crystalline form |
Andreas Hafner, Martin Szelagiewicz, Bernd Siebenhaar, Tiziana Chiodo, Tobias Hintermann +2 more |
2017-01-31 |
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| 9433624 |
Methods and compositions for the treatment of metabolic disorders |
Daniel I. Oppenheimer, Emil D. Kakkis, Fredric D. Price, Alejandro Dorenbaum, Rudolf Moser +2 more |
2016-09-06 |
$179,906,000 |
| 9394328 |
Crystalline dapagliflozin hydrate |
Katharina Reichenbaecher |
2016-07-19 |
$13,205,000 |
| 9340536 |
Multicomponent crystals comprising dasatinib and selected co-crystal formers |
Tiziana Chiodo, Andreas Hafner, Tobias Hintermann, Beate Salvador, Martin Szelagiewicz +2 more |
2016-05-17 |
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