Issued Patents All Time
Showing 1–25 of 27 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12024520 | Processes for the preparation of 4-{8-amino-3-[(2S)-1-(but-2-ynoyl)-pyrrolidin-2-yl]imidazo[1,5-a]-pyrazin-1-yl}N-(pyridin-2-yl)-benzamide | Paul Allen Bethel, Lai Chun CHAN, Katie Grace COOPER, Robert John COX, Michael David Golden +15 more | 2024-07-02 |
| 11820777 | Crystal forms of (s)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa | 2023-11-21 |
| 11059829 | Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide maleate | Fritz Blatter, Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa | 2021-07-13 |
| 10954199 | Process methods for phosphatidylinositol 3-kinase inhibitors | Stacy Bremner, Keiko Sujino, Duong Tran, Dragos Vizitiu | 2021-03-23 |
| 10858364 | Imidazopyrazine inhibitors of Bruton's tyrosine kinase | Terry Podoll, Allard Kaptein | 2020-12-08 |
| 10730879 | Polymorphic forms of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one | Ernest A. Carra, Michael J. Gerber, Bing Shi, Keiko Sujino, Duong Tran +1 more | 2020-08-04 |
| 10640509 | Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide for treating diffuse large B-cell lymphoma | Fritz Blatter, Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa | 2020-05-05 |
| 10442805 | Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one | Suzanne BUTTAR, Ernest A. Carra, Tracy Ehiwe, Duong Tran, Fang Wang +1 more | 2019-10-15 |
| 10414737 | Process methods for phosphatidylinositol 3-kinase inhibitors | Stacy Bremner, Keiko Sujino, Duong Tran, Dragos Vizitiu | 2019-09-17 |
| 10308639 | Phosphatidylinositol 3-kinase inhibitors | Joshua A. Kaplan, Leena Patel, Stephane Perreault, Barton W. Phillips, Gary Phillips +2 more | 2019-06-04 |
| 10221197 | Phosphatidylinositol 3-kinase inhibitors | Zhimin Du, Joshua A. Kaplan, Musong Kim, Devan Naduthambi, Leena Patel +8 more | 2019-03-05 |
| 10167291 | Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl) pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa | 2019-01-01 |
| 10059677 | Process for preparing phosphatidylinositol 3-kinase inhibitors and intermediates thereof | Stacy Bremner, Keiko Sujino, Duong Tran, Dragos Vizitiu | 2018-08-28 |
| 10047060 | Process methods for phosphatidylinositol 3-kinase inhibitors | Stacy Bremner, Keiko Sujino, Duong Tran, Dragos Vizitiu | 2018-08-14 |
| 9796721 | Crystal forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide | Fritz Blatter, Tim Ingallinera, Tjeerd Barf, Edwin Aret, Cecile M. Krejsa | 2017-10-24 |
| 9765060 | Phosphatidylinositol 3-kinase inhibitors | Joshua A. Kaplan, Musong Kim, Devan Naduthambi, Leena Patel, Stephane Perreault +4 more | 2017-09-19 |
| 9708327 | Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one | Suzanne BUTTAR, Ernest A. Carra, Tracy Ehiwe, Duong Tran, Fang Wang +1 more | 2017-07-18 |
| 9567337 | Process methods for phosphatidylinositol 3-kinase inhibitors | Stacy Bremner, Keiko Sujino, Duong Tran, Dragos Vizitiu | 2017-02-14 |
| 9469643 | Polymorphic forms of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one | Ernest A. Carra, Michael J. Gerber, Bing Shi, Keiko Sujino, Duong Tran +1 more | 2016-10-18 |
| 9266878 | Phosphatidylinositol 3-kinase inhibitors | Leena Patel, Jennifer Treiberg, Stephane Perreault, Arthur Yeung, Lafe J. Purvis, II +1 more | 2016-02-23 |
| 9221795 | Phosphatidylinositol 3-kinase inhibitors | Joshua A. Kaplan, Musong Kim, Leena Patel, Stephane Perreault, Gary Phillips +2 more | 2015-12-29 |
| 9029384 | Phosphatidylinositol 3-kinase inhibitors | Leena Patel, Joshua A. Kaplan, Jennifer Treiberg, Stephane Perreault, Gary Phillips | 2015-05-12 |
| 9018221 | Phosphatidylinositol 3-kinase inhibitors | Leena Patel, Jennifer Treiberg, Stephane Perreault, Arthur Yeung, Lafe J. Purvis, II +1 more | 2015-04-28 |
| 8865730 | Polymorphic forms of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one | Ernest A. Carra, Michael J. Gerber, Bing Shi, Keiko Sujino, Duong Tran +1 more | 2014-10-21 |
| 8546409 | Methods of treatment for solid tumors | Kamal D. Puri, Brian Lannutti, Neill A. Giese | 2013-10-01 |