Issued Patents All Time
Showing 26–50 of 58 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 10639310 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | James D. Rodgers | 2020-05-05 |
| 10479795 | Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors | Andrew W. Buesking, Richard B. Sparks, Andrew P. Combs, Brent Douty, Nikoo Falahatpisheh +5 more | 2019-11-19 |
| 10472368 | Heterocyclic compounds as PI3K-γ inhibitors | Artem Shvartsbart, Andrew P. Combs, Lixin Shao, Nikoo Falahatpisheh, Ge Zou +4 more | 2019-11-12 |
| 10463667 | Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | James D. Rodgers, Argyrios G. Arvanitis, Jack Guoen Shi | 2019-11-05 |
| 10442803 | Tricyclic heterocycles as bet protein inhibitors | James D. Rodgers, Haisheng Wang, Lixin Shao | 2019-10-15 |
| 10398699 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors | James D. Rodgers | 2019-09-03 |
| 10138248 | Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-γ inhibitors | Andrew W. Buesking, Richard B. Sparks, Andrew P. Combs, Brent Douty, Nikoo Falahatpisheh +2 more | 2018-11-27 |
| 10065963 | Heterocyclic compounds as PI3K-γ inhibitors | Artem Shvartsbart, Andrew P. Combs, Lixin Shao, Nikoo Falahatpisheh, Ge Zou +2 more | 2018-09-04 |
| 9974790 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors | James D. Rodgers | 2018-05-22 |
| 9814722 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors | James D. Rodgers | 2017-11-14 |
| 9777003 | Tricyclic heterocycles as bet protein inhibitors | Lixin Shao, Haisheng Wang | 2017-10-03 |
| 9662335 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as janus kinase inhibitors | James D. Rodgers | 2017-05-30 |
| 9512161 | Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-D]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | James D. Rodgers, Adam Shilling, Argyrios G. Arvanitis, Laurine G. Galya, Mei Li +1 more | 2016-12-06 |
| 9334274 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Argyrios G. Arvanitis, Haisheng Wang, Louis Storace, Beverly Folmer +3 more | 2016-05-10 |
| 9309246 | Tricyclic heterocycles as BET protein inhibitors | James D. Rodgers, Haisheng Wang, Lixin Shao | 2016-04-12 |
| 9249145 | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Yun-Long Li, Haisheng Wang | 2016-02-02 |
| 9206187 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase | James D. Rodgers, Jordan S. Fridman, Krishna Vaddi | 2015-12-08 |
| 9193733 | Piperidinylcyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors | James D. Rodgers, Wenyu Zhu, Lixin Shao, Joseph Glenn | 2015-11-24 |
| 9079912 | Heteroaryl substituted pyrrolo[2,3-B] pyridines and pyrrolo[2,3-B] pyrimidines as Janus kinase inhibitors | James D. Rodgers | 2015-07-14 |
| 8946245 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | James D. Rodgers, Jordan S. Fridman, Krishna Vaddi | 2015-02-03 |
| 8933086 | Heteroaryl substituted pyrrolo[2,3-B]pyridines and pyrrolo[2,3-B]pyrimidines as Janus kinase inhibitors | James D. Rodgers, Jordan S. Fridman, Krishna Vaddi | 2015-01-13 |
| 8933085 | Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors | James D. Rodgers, Wenyu Zhu, Lixin Shao, Joseph Glenn | 2015-01-13 |
| 8889697 | Metabolites of the janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | James D. Rodgers, Argyrios G. Arvanitis, Jack Guoen Shi | 2014-11-18 |
| 8748401 | Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | James D. Rodgers, Adam Shilling, Argyrios G. Arvanitis, Laurine G. Galya, Mei Li +1 more | 2014-06-10 |
| 8716303 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Argyrios G. Arvanitis, Haisheng Wang, Louis Storace, Beverly Folmer +3 more | 2014-05-06 |