Issued Patents All Time
Showing 1–25 of 29 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12187725 | Tricyclic urea compounds as JAK2 V617F inhibitors | Yanran Ai, Yu Sheng Bai, Joseph Barbosa, Hao Feng, Leah C. Konkol +5 more | 2025-01-07 |
| 11952367 | Pyridine and pyridimine compounds as PI3K-gamma inhibitors | Richard B. Sparks, Stacey Shepard, Andrew P. Combs, Andrew W. Buesking, Lixin Shao +1 more | 2024-04-09 |
| 11780840 | Tricyclic urea compounds as JAK2 V617F inhibitors | Yanran Ai, Onur Atasoylu, Yu Sheng Bai, Joseph Barbosa, David M. Burns +11 more | 2023-10-10 |
| 11352340 | Pyridine and pyridimine compounds as PI3K-gamma inhibitors | Richard B. Sparks, Stacey Shepard, Andrew P. Combs, Andrew W. Buesking, Lixin Shao +1 more | 2022-06-07 |
| 11091484 | Tricyclic heterocycles as BET protein inhibitors | James D. Rodgers, Stacey Shepard, Lixin Shao | 2021-08-17 |
| 10975085 | Process for preparing a composition comprising an enantiomeric excess of greater than or equal to 90% of the (R)-enantiomer of a compound of formula III | Jiacheng Zhou, James D. Rodgers | 2021-04-13 |
| 10442803 | Tricyclic heterocycles as bet protein inhibitors | James D. Rodgers, Stacey Shepard, Lixin Shao | 2019-10-15 |
| 10364248 | Processes for preparing 4-chloro-7H-pyrrolo[2,3-d]pyrimidine | Jiacheng Zhou, James D. Rodgers | 2019-07-30 |
| 9908888 | Processes for preparing pyrazolyl-substituted pyrrolo[2,3-d]pyrimidines | Jiacheng Zhou, Pingli Liu, Qiyan Lin, Brian W. Metcalf, David Meloni +5 more | 2018-03-06 |
| 9879010 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b] pyrimidin-5-yl-amines as Janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2018-01-30 |
| 9777003 | Tricyclic heterocycles as bet protein inhibitors | Stacey Shepard, Lixin Shao | 2017-10-03 |
| 9580419 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2017-02-28 |
| 9334274 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Stacey Shepard, Argyrios G. Arvanitis, Louis Storace, Beverly Folmer +3 more | 2016-05-10 |
| 9309246 | Tricyclic heterocycles as BET protein inhibitors | James D. Rodgers, Stacey Shepard, Lixin Shao | 2016-04-12 |
| 9249145 | Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Yun-Long Li, Stacey Shepard | 2016-02-02 |
| 9090611 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2015-07-28 |
| 8741895 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2014-06-03 |
| 8716303 | N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors | James D. Rodgers, Stacey Shepard, Argyrios G. Arvanitis, Louis Storace, Beverly Folmer +3 more | 2014-05-06 |
| 8445488 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2013-05-21 |
| 8415362 | Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | James D. Rodgers, Stacey Shepard, Thomas P. Maduskuie, Jr., Nikoo Falahatpisheh, Maria Rafalski +3 more | 2013-04-09 |
| 8410265 | Processes for preparing JAK inhibitors and related intermediate compounds | Jiacheng Zhou, Pingli Liu, Qiyan Lin, Brian W. Metcalf, David Meloni +5 more | 2013-04-02 |
| 8053433 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2011-11-08 |
| 7335667 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-4-yl-amines as Janus kinase inhibitors | James D. Rodgers, Andrew P. Combs, Richard B. Sparks | 2008-02-26 |
| 6969721 | Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors | James D. Rodgers, Mona Patel, Argyrios G. Arvanitis, Anthony J. Cocuzza | 2005-11-29 |
| 6809109 | 2, 4-disubstituted-pyridine N-oxides useful as HIV reverse transcriptase inhibitors | James D. Rodgers | 2004-10-26 |