AC

Andrew P. Combs

IN Incyte: 115 patents #2 of 356Top 1%
PI Prelude Therapeutics, Incorporated: 7 patents #4 of 25Top 20%
BS Bristol-Myers Squibb: 2 patents #1,811 of 3,969Top 50%
Overall (All Time): #9,051 of 4,157,543Top 1%
125
Patents All Time

Issued Patents All Time

Showing 25 most recent of 125 patents

Patent #TitleCo-InventorsDate
12421197 Aminopyrazine derivatives as PI3K-γ inhibitors Brent Douty, Yanran Ai, David M. Burns, Nikoo Falahatpisheh, Daniel Levy +6 more 2025-09-23
12365668 Aminopyrazine diol compounds as PI3K-y inhibitors Stacey Shepard, Nikoo Falahatpisheh, Lixin Shao 2025-07-22
12227502 1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c] pyridin-7(6H)-ones as inhibitors of BET proteins Thomas P. Maduskuie, Jr., Nikoo Falahatpisheh 2025-02-18
12201636 Heterocyclylamines as PI3K inhibitors Yun-Long Li, Wenqing Yao, Eddy W. Yue, Song Mei, Joseph Glenn +2 more 2025-01-21
12173006 Crystalline forms of a phosphoinositide 3-kinase (PI3K) inhibitor Brent Douty, David M. Burns, Zhongjiang Jia, Daniel Levy, Eddy W. Yue 2024-12-24
12152033 Use of pyrazolopyrimidine derivatives for the treatment of PI3K-δ related disorders Yun-Long Li, Eddy W. Yue, Song Mei, Brent Douty 2024-11-26
12129262 CDK inhibitors and their use as pharmaceuticals Xiaowei Wu, Andrew W. Buesking, Ryan Holmes, Sarah Pawley, Katarina Rohlfing 2024-10-29
12030885 Substituted imidazo[2,1-f][1,2,4]triazines as PI3K-gamma inhibitors Andrew W. Buesking, Richard B. Sparks, Brent Douty, Nikoo Falahatpisheh, Lixin Shao +5 more 2024-07-09
12006320 Heterocyclic derivatives as PI3K inhibitors Stacey Shepard, Yanran Ai, Nikoo Falahatpisheh, Lixin Shao, Artem Shvartsbart 2024-06-11
11999751 Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors Yun-Long Li 2024-06-04
11952367 Pyridine and pyridimine compounds as PI3K-gamma inhibitors Richard B. Sparks, Stacey Shepard, Andrew W. Buesking, Lixin Shao, Haisheng Wang +1 more 2024-04-09
11939340 CDK inhibitors and their use as pharmaceuticals Jincong Zhuo, Xiaowei Wu, Katarina Rohlfing 2024-03-26
11926616 Aminopyrazine diol compounds as PI3K-γ inhibitors Stacey Shepard, Nikoo Falahatpisheh, Lixin Shao 2024-03-12
11926630 Tertiary alcohols as PI3K-γ inhibitors Brent Douty, Andrew W. Buesking, David M. Burns, Nikoo Falahatpisheh, Ravi Kumar Jalluri +7 more 2024-03-12
11819505 Heterocyclylamines as PI3K inhibitors Yun-Long Li, Eddy W. Yue, Brent Douty, Song Mei 2023-11-21
11773102 Heterocyclic compounds as PI3K-γ inhibitors Artem Shvartsbart, Stacey Shepard, Lixin Shao, Nikoo Falahatpisheh, Ge Zou +4 more 2023-10-03
11702416 1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins Thomas P. Maduskuie, Jr., Nikoo Falahatpisheh 2023-07-18
11702423 BRM targeting compounds and associated methods of use Hong-Nien Lin, Philip Pitis, Liang Lu 2023-07-18
11685744 CDK inhibitors and their use as pharmaceuticals Andrew W. Buesking, Jincong Zhuo, Ryan Holmes, Sarah Pawley, Xiaowei Wu 2023-06-27
11673893 CDK inhibitors and their use as pharmaceuticals Liang Lu, Rupa Shetty, Chaofeng Dai, Raul Andrew Leal, Klare Lazor Bersch 2023-06-13
11622970 BCL-2 inhibitors and their use as pharmaceuticals Jincong Zhuo, Peng Wei, Jialiang Wang 2023-04-11
11498926 Tricyclic heterocycles as BET protein inhibitors Richard B. Sparks, Thomas P. Maduskuie, Jr., James D. Rodgers 2022-11-15
11433071 Heterocyclylamines as PI3K inhibitors Yun-Long Li, Wenqing Yao, Eddy W. Yue, Song Mei, Joseph Glenn +4 more 2022-09-06
11401280 Pyrimidinones as PI3K inhibitors Yun-Long Li, Brian W. Metcalf 2022-08-02
11396502 Substituted heterocyclic derivatives as PI3K inhibitors Stacey Shepard 2022-07-26