Issued Patents All Time
Showing 26–50 of 125 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 11352340 | Pyridine and pyridimine compounds as PI3K-gamma inhibitors | Richard B. Sparks, Stacey Shepard, Andrew W. Buesking, Lixin Shao, Haisheng Wang +1 more | 2022-06-07 |
| 11306079 | 3-(5-amino-pyrazin-2-yl)-benzenesulfonamide derivatives and related compounds as PI3K-gamma kinase inhibitors | Artem Shvartsbart, Nikoo Falahatpisheh, Padmaja Polam, Lixin Shao, Stacey Shepard | 2022-04-19 |
| 11225486 | Tertiary alcohols as PI3K-γ inhibitors | Brent Douty, Andrew W. Buesking, David M. Burns, Nikoo Falahatpisheh, Ravi Kumar Jalluri +7 more | 2022-01-18 |
| 11207302 | 1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase | Eddy W. Yue, Richard B. Sparks, Wenyu Zhu, Jiacheng Zhou, Qiyan Lin +3 more | 2021-12-28 |
| 11192868 | Modulators of indoleamine 2,3-dioxygenase and methods of using the same | Eddy W. Yue | 2021-12-07 |
| 11186580 | Crystalline forms of a phosphoinositide 3-kinase (PI3K) inhibitor | Brent Douty, David M. Burns, Zhongjiang Jia, Daniel Levy, Eddy W. Yue | 2021-11-30 |
| 11161838 | Heterocyclic derivatives as PI3K inhibitors | Stacey Shepard, Yanran Ai, Artem Shvartsbart | 2021-11-02 |
| 11130767 | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors | Yun-Long Li | 2021-09-28 |
| 11130769 | Spiro-sulfonamide derivatives as inhibitors of myeloid cell leukemia-1 (MCL-1) protein | Jincong Zhuo, Raul Andrew Leal, Rupa Shetty, Juan Luengo, Peng Wei | 2021-09-28 |
| 11091491 | Heterocyclic compounds as PI3K-y inhibitors | Artem Shvartsbart, Stacey Shepard, Lixin Shao, Nikoo Falahatpisheh, Ge Zou +4 more | 2021-08-17 |
| 11078204 | Heterocyclic derivatives as PI3K inhibitors | Stacey Shepard, Yanran Ai, Nikoo Falahatpisheh, Lixin Shao, Artem Shvartsbart | 2021-08-03 |
| 11059821 | 1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins | Thomas P. Maduskuie, Jr., Nikoo Falahatpisheh | 2021-07-13 |
| 11046658 | Aminopyrazine derivatives as PI3K-γ inhibitors | Brent Douty, Yanran Ai, David M. Burns, Nikoo Falahatpisheh, Daniel Levy +6 more | 2021-06-29 |
| 10975088 | Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors | Andrew W. Buesking, Richard B. Sparks, Brent Douty, Nikoo Falahatpisheh, Lixin Shao +5 more | 2021-04-13 |
| 10919912 | Tricyclic heterocycles as BET protein inhibitors | Richard B. Sparks, Thomas P. Maduskuie, Jr., James D. Rodgers | 2021-02-16 |
| 10829502 | Pyrimidinones as PI3K inhibitors | Yun-Long Li, Brian W. Metcalf | 2020-11-10 |
| 10781209 | 1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins | Thomas P. Maduskuie, Jr., Nikoo Falahatpisheh | 2020-09-22 |
| 10738057 | Tertiary alcohols as PI3K-γ inhibitors | Brent Douty, Andrew W. Buesking, David M. Burns, Nikoo Falahatpisheh, Ravi Kumar Jalluri +7 more | 2020-08-11 |
| 10669262 | Aminopyrazine diol compounds as PI3K-γ inhibitors | Stacey Shepard, Nikoo Falahatpisheh, Lixin Shao | 2020-06-02 |
| 10653677 | 1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase | Eddy W. Yue, Richard B. Sparks, Wenyu Zhu | 2020-05-19 |
| 10646492 | Heterocyclylamines as PI3K inhibitors | Yun-Long Li, Wenqing Yao, Song Mei, Joseph Glenn, Thomas P. Maduskuie, Jr. +1 more | 2020-05-12 |
| 10618910 | Tricyclic heterocycles as BET protein inhibitors | Richard B. Sparks | 2020-04-14 |
| 10596184 | Aza-heteroaryl compounds as PI3K-gamma inhibitors | Ge Zou | 2020-03-24 |
| 10479795 | Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors | Andrew W. Buesking, Richard B. Sparks, Brent Douty, Nikoo Falahatpisheh, Lixin Shao +5 more | 2019-11-19 |
| 10479803 | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors | Yun-Long Li | 2019-11-19 |