Issued Patents All Time
Showing 51–75 of 87 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 8563541 | Azepine inhibitors of Janus kinases | Argyrios G. Arvanitis, Andrew P. Combs, Richard B. Sparks, Darius J. Robinson | 2013-10-22 |
| 8541425 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Stacey Shepard, Jordan S. Fridman, Krishna Vaddi | 2013-09-24 |
| 8530485 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Stacey Shepard | 2013-09-10 |
| 8513270 | Substituted heterocycles as Janus kinase inhibitors | Argyrios G. Arvanitis, Louis Storace, Beverly Folmer | 2013-08-20 |
| 8486902 | Hydroxyl, keto, and glucuronide derivatives of 3-(4-(7H-pyrrolo[2,3-d] pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Adam Shilling, Argyrios G. Arvanitis, Stacey Shepard, Laurine G. Galya, Mei Li +1 more | 2013-07-16 |
| 8445488 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors | Haisheng Wang, Andrew P. Combs, Richard B. Sparks | 2013-05-21 |
| 8420629 | Azetidine and cyclobutane derivatives as JAK inhibitors | Stacey Shepard | 2013-04-16 |
| 8415362 | Pyrazolyl substituted pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors | Stacey Shepard, Thomas P. Maduskuie, Jr., Haisheng Wang, Nikoo Falahatpisheh, Maria Rafalski +3 more | 2013-04-09 |
| 8410265 | Processes for preparing JAK inhibitors and related intermediate compounds | Jiacheng Zhou, Pingli Liu, Qiyan Lin, Brian W. Metcalf, David Meloni +5 more | 2013-04-02 |
| 8309718 | 4-pyrazolyl-N-arylpyrimidin-2-amines and 4-pyrazolyl-N-heteroarylpyrimidin-2-amines as janus kinase inhibitors | Yun-Long Li, Wenqing Yao | 2012-11-13 |
| 8158616 | Azetidine and cyclobutane derivatives as JAK inhibitors | Stacey Shepard | 2012-04-17 |
| 8053433 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as janus kinase inhibitors | Haisheng Wang, Andrew P. Combs, Richard B. Sparks | 2011-11-08 |
| 7834022 | Metabolites of the Janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile | Argyrios G. Arvantis, Jack Guoen Shi, Stacey Shepard | 2010-11-16 |
| 7598257 | Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors | Stacey Shepard | 2009-10-06 |
| 7335667 | Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-4-yl-amines as Janus kinase inhibitors | Haisheng Wang, Andrew P. Combs, Richard B. Sparks | 2008-02-26 |
| 6969721 | Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors | Haisheng Wang, Mona Patel, Argyrios G. Arvanitis, Anthony J. Cocuzza | 2005-11-29 |
| 6946469 | Cyanamide, alkoxyamino, and urea derivatives of 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones as HIV reverse transcriptase inhibitors | Jeffery W. Corbett | 2005-09-20 |
| 6825210 | Tricyclic compounds useful as HIV reverse transcriptase inhibitors | Barry Johnson, Qiyan Lin, Anurag S. Srivastava | 2004-11-30 |
| 6809109 | 2, 4-disubstituted-pyridine N-oxides useful as HIV reverse transcriptase inhibitors | Haisheng Wang | 2004-10-26 |
| 6596729 | Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors | Haisheng Wang, Mona Patel, Argyrios G. Arvanitis, Anthony J. Cocuzza | 2003-07-22 |
| 6593337 | Tricyclic compounds useful as HIV reverse transcriptase inhibitors | Barry Johnson, Mona Patel, Christine M. Tarby, Rajagopal Bakthavatchalam | 2003-07-15 |
| 6503898 | Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors | Patrick Lam, Prabhakar Kondaji Jadhav, Charles Joseph Eyermann, Carl Nicholas Hodge, George V. De Lucca | 2003-01-07 |
| 6489320 | 5, 5-disubstituted-1, 5-dihydro-4, 1-benzoxazepin-2 (3H)-ones useful as HIV reverse transcriptase inhibitors | Anthony J. Cocuzza | 2002-12-03 |
| 6462037 | 1,4-benzodiazepin-2-ones useful as HIV reverse transcriptase inhibitors | Barry Johnson, Haisheng Wang | 2002-10-08 |
| 6451999 | 1-(3-aminoindazol-5-yl)-3-butyl-cyclic urea useful as a HIV protease inhibitor | Patrick Lam | 2002-09-17 |