Patent Leaderboard
USPTO Patent Rankings Data through Sept 30, 2025
MN

Matthias Nettekoven — 130 Patents

Hoffmann-La Roche: 126 patents #1 of 3,238Top 1%
RNRemynd N.V.: 4 patents #11 of 27Top 45%
VLVernalis Research Limited: 1 patents #39 of 57Top 70%
Weil am Rhein, DE: #1 of 1 inventorsTop 100%
Overall (All Time): #8,436 of 4,157,543Top 1%
130 Patents All Time

Issued Patents All Time

Showing 76–100 of 130 patents

Patent #TitleCo-InventorsDate
7605163 Benzoyl-piperazine derivatives Synese Jolidon, Robert Narquizian, Roger Norcross, Emmanuel Pinard, Henri Stalder 2009-10-20
7601711 5-amido-indole-2-carboxamide derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2009-10-13
7595314 Benzoyl-piperazine derivatives Daniela Alberati-Giani, Synese Jolidon, Robert Narquizian, Roger Norcross, Emmanuel Pinard +1 more 2009-09-29
7592345 Piperazine and [1,4]diazepan derivatives as NK antagonists Henner Knust, Hasane Ratni, Xihan Wu 2009-09-22
7579351 Tricyclic amide derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2009-08-25
7557101 4,5,6,7-tetrahydro-thieno[3,2-c] pyridine derivatives Li Chen, Wayne Wen Lai, Olivier Roche, Deye Zheng 2009-07-07
7557108 (Indol-4-yl) or (indol-5-yl)-piperazinylmethanones Olivier Roche 2009-07-07
7544683 Cyclohexyl derivatives Delphine Gaufreteau, Jean-Marc Plancher, Olivier Roche, Sebastien Schmitt, Tadakatsu Takahashi 2009-06-09
7538132 Isoxazolo derivatives Bernd Buettelmann, Bo Han, Henner Knust, Andrew Thomas 2009-05-26
7538101 1,1-dioxo-thiomorpholinyl indolyl methanone derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Rosa Maria Rodriguez Sarmiento, Sven Taylor 2009-05-26
7534788 Benzofuran and benzothiophene-2-carboxylic acid amide derivatives Peter Mohr, Jean-Marc Plancher, Hans Richter, Olivier Roche, Tadakatsu Takahashi +1 more 2009-05-19
7534891 Quinoline derivatives as H3R inverse agonists Silvia Gatti McArthur, Cornelia Hertel, Susanne Raab, Hans Richter, Olivier Roche +2 more 2009-05-19
7528135 Pyridine derivatives as H3 antagonists Olivier Roche, Rosa Maria Rodriguez-Sarmiento 2009-05-05
7528136 Prolinamide derivatives as NK3 antagonists Bo Han, Henner Knust, Hasane Ratni, Xihan Wu 2009-05-05
7514433 1H-indole-6-yl-piperazin-1-yl-methanone derivatives Olivier Roche 2009-04-07
7507736 Indol-2-yl-piperazin-1-yl-methanone derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2009-03-24
7501422 Prolinamide-tetrazole derivatives as NK3 receptor antagonists Bo Han, Henner Knust, Hasane Ratni, Xihan Wu 2009-03-10
7501541 Malonamides as orexin antagonists Luca Gobbi, Henner Knust, Parichehr Malherbe, Emmanuel Pinard, Olivier Roche +1 more 2009-03-10
7470684 Spiropiperidine derivatives as NK3 antagonists Joanie Marie Caroon, Michael Patrick Dillon, Bo Han, Hasane Ratni, Walter Vifian 2008-12-30
7462617 Substituted acylpiperazine derivatives Daniela Alberati-Giani, Synese Jolidon, Robert Narquizian, Roger Norcross, Emmanuel Pinard +1 more 2008-12-09
7459480 Benzodioxepine derivatives Luca Gobbi, Marcel Gubler, Werner Neidhart 2008-12-02
7456175 Piperazinyl-pyridine derivatives Olivier Roche, Rosa Maria Rodriguez-Sarmiento 2008-11-25
7456174 5-aminoindole derivatives as H3 inverse agonists Jean-Marc Plancher, Olivier Roche, Rosa Maria Rodriguez-Sarmiento 2008-11-25
7432255 1H-indol-5-yl-piperazin-1-yl-methanone derivatives Olivier Roche 2008-10-07
7427612 Benzoyl-piperazine derivatives Daniela Alberati-Giani, Synese Jolidon, Robert Narquizian, Roger Norcross, Emmanuel Pinard +1 more 2008-09-23