Patent Leaderboard
USPTO Patent Rankings Data through Sept 30, 2025
MN

Matthias Nettekoven — 130 Patents

Hoffmann-La Roche: 126 patents #1 of 3,238Top 1%
RNRemynd N.V.: 4 patents #11 of 27Top 45%
VLVernalis Research Limited: 1 patents #39 of 57Top 70%
Weil am Rhein, DE: #1 of 1 inventorsTop 100%
Overall (All Time): #8,436 of 4,157,543Top 1%
130 Patents All Time

Issued Patents All Time

Showing 51–75 of 130 patents

Patent #TitleCo-InventorsDate
8067598 Heterofused piperidines as orexin antagonists Luca Gobbi, Henner Knust, Parichehr Malherbe, Emmanuel Pinard, Olivier Roche +1 more 2011-11-29
8063075 Pyrrolidine ether derivatives as NK3 receptor antagonists Philippe Jablonski, Kenichi Kawasaki, Henner Knust, Anja Limberg, Hasane Ratni +1 more 2011-11-22
8022099 N-benzyl pyrrolidine derivatives Caterina Bissantz, Philippe Jablonski, Henner Knust, Hasane Ratni, Claus Riemer 2011-09-20
8017773 Cyclohexyl sulfonamide derivatives Olivier Roche 2011-09-13
8012998 Pyrrolidine aryl-ether as NK-3 receptor antagonists Philippe Jablonski, Kenichi Kawasaki, Henner Knust, Anja Limberg, Hasane Ratni +2 more 2011-09-06
7932269 Sulfonamides as orexin antagonists Henner Knust, Emmanuel Pinard, Olivier Roche, Mark Rogers-Evans 2011-04-26
7923470 Benzooxazoles as orexin antagonists Henner Knust, Emmanuel Pinard, Olivier Roche, Mark Rogers-Evans 2011-04-12
7902184 Piperazinyl pyrimidine derivatives Olivier Roche 2011-03-08
7897627 Heteroaryl derivatives as orexin receptor antagonists Henner Knust, Emmanuel Pinard, Olivier Roche, Mark Rogers-Evans 2011-03-01
7893062 Pyrrolidine derivatives as dual NK1/NK3 receptor antagonists Caterina Bissantz, Torsten Hoffmann, Philippe Jablonski, Henner Knust, Hasane Ratni +1 more 2011-02-22
7829563 Aminoamides as orexin antagonists Luca Gobbi, Henner Knust, Parichehr Malherbe, Emmanuel Pinard, Olivier Roche +1 more 2010-11-09
7812028 3-pyridinecarboxamide derivatives as HDL-cholesterol raising agents Mirjana Andjelkovic, Agnes Benardeau, Evelyne Chaput, Paul Hebeisen, Ulrike Obst Sander +2 more 2010-10-12
7812021 Pyrrolidine aryl-ether as NK3 receptor antagonists Philippe Jablonski, Kenichi Kawasaki, Henner Knust, Anja Limberg, Hasane Ratni +2 more 2010-10-12
7786109 Tricyclic amide derivatives as modulators of H3 receptors Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2010-08-31
7786128 Indole or benzimidazole derivatives as CB1 inverse agonists Konrad Bleicher, Philippe Pflieger, Stephen Roever 2010-08-31
7786143 Thiazolyl piperidine derivatives Olivier Roche 2010-08-31
7754736 5-aminoindole derivatives as H3 inverse agonists Jean-Marc Plancher, Olivier Roche, Rosa Maria Rodriguez-Sarmiento 2010-07-13
7745479 1,5-substituted indol-2-yl amide derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Valerie Runtz-Schmitt, Sven Taylor 2010-06-29
7723325 5-amido-indole-2-carboxamide derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2010-05-25
7691863 Pyrazine-2-carboxamide derivatives as CB2 receptor modulators Michel Dietz, Sabine Gruener, Paul Hebeisen, Sylvie C. Meyer Reigner, Bernd PUELLMANN +2 more 2010-04-06
7648979 5-amido-(1H-indol-2-yl)-piperazin-1-yl-methanone derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2010-01-19
7629346 Pyrazinecarboxamide derivatives as CB1 antagonists Paul Hebeisen, Hans Iding, Ulrike Obst Sander, Stephan Roever, Urs Weiss +1 more 2009-12-08
7622466 Azaindole-2-carboxamide derivatives Jean-Marc Plancher, Hans Richter, Olivier Roche, Sven Taylor 2009-11-24
7612076 Piperazinyl-pyridine derivatives Olivier Roche, Rosa Maria Rodriguez-Sarmiento 2009-11-03
7608617 Naphthaline derivatives as H3 inverse agonists Silvia Gatti McArthur, Cornelia Hertel, Jean-Marc Plancher, Susanne Raab, Olivier Roche +2 more 2009-10-27