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Crystalline polymorphs of a 1-thiazol-2-yl-pyrazole-5-carboxylic acid derivative |
Zheqiong Wu, Shanming Kuang |
2025-08-05 |
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Methods for making thiazolypyrazole carboxylic acids and intermediates therefor |
Paul O'Shea, Narayanan Anantha |
2025-07-15 |
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Methods of using substituted pyrazole and pyrazole compounds and for treatment of hyperproliferative diseases |
Arshad Siddiqui, Stephane Ciblat, Lea Constantineau-Forget, Chantal Grand-Maitre, Xiangyu Guo +6 more |
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Substituted pyrazole and pyrrole compounds and methods for using them for inhibition of initiation of translation and treatment of diseases and disorders relating thereto |
M. Arshad Siddiqui, Stephane Ciblat, Martin Dery, Lea Constantineau-Forget, Chantal Grand-Maitre +5 more |
2023-03-14 |
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Substituted pyrazole compounds and methods of using them for treatment of hyperproliferative diseases |
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2022-05-10 |
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Substituted pyrazole and pyrrole compounds and methods for using them for inhibition of initiation of translation and treatment of diseases and disorders relating thereto |
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BTK Inhibitors |
Adrianus Petrus Antonius De Man, Jan Gerard Sterrenburg, Hans C.A. Raaijmakers, Allard Kaptein, Arthur A. Oubrie +18 more |
2017-08-01 |
$68,609,000 |
| 9351965 |
Indazole derivatives useful as ERK inhibitors |
Gerald W. Shipps, Jr., Xiaohua Huang, Yongqi Deng, Liang Zhu, Binyuan Sun +2 more |
2016-05-31 |
$68,752,000 |
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Fused pyrazole derivatives as novel ERK inhibitors |
Gerald W. Shipps, Jr., Yongqi Deng, Xiaolei Gao, Binyuam Sun, James Wang +1 more |
2016-01-26 |
$42,047,000 |
| 8999957 |
Heterocyclic compounds as ERK inhibitors |
Yongqi Deng, Liang Zhu, Gerald W. Shipps, Jr., Sie-Mun Lo, Binyuan Sun +16 more |
2015-04-07 |
$36,039,000 |
| 8999966 |
Compounds that are ERK inhibitors |
Sobhana Babu Boga, Joseph M. Kelly, Hugh Y. Zhu, Abdul-Basit Alhassan, Xin Yao +8 more |
2015-04-07 |
$36,039,000 |
| 8946216 |
Indazole derivatives useful as ERK inhibitors |
Yonqi Deng, Gerald W. Shipps, Jr., Sie-Mun Lo, Liang Zhu, Kiran Muppalla |
2015-02-03 |
$56,549,000 |
| 8716483 |
Compounds that are ERK inhibitors |
Yang Nan, Yongqi Deng, Gerald W. Shipps, Jr., Neng-Yang Shih, Hugh Y. Zhu +9 more |
2014-05-06 |
$63,658,000 |
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Compounds that are ERK inhibitors |
Hugh Y. Zhu, Jagdish A. Desai, Ronald J. Doll |
2014-02-25 |
$94,969,000 |
| 8546404 |
Compounds that are ERK inhibitors |
Yongqi Deng, Gerald W. Shipps, Jr., Neng-Yang Shih, Hugh Y. Zhu, Robert Sun +21 more |
2013-10-01 |
$68,208,000 |
| 7807672 |
Compounds that are ERK inhibitors |
Yongqi Deng, Gerald W. Shipps, Jr., Yang Nan, Tong Wang, M. Arshad Siddiqui +11 more |
2010-10-05 |
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Farnesyl protein transferase inhibitors as antitumor agents |
Hugh Y. Zhu, Jagdish A. Desai, James Wang, Ronald J. Doll, F. George Njoroge +1 more |
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Substituted 5-carboxyamide pyrazoles and [1,2,4]triazoles as antiviral agents |
Hugh Y. Zhu, James Wang, Jagdish A. Desai, Gerald W. Shipps, Jr., Patrick J. Curran +3 more |
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Farnesyl protein transferase inhibitors as antitumor agents |
Hugh Y. Zhu, F. George Njoroge, Timothy J. Guzi, Dinanath F. Rane, Keith P. Minor +13 more |
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Substituted 5-oxo pyrazoles and [1,2,4]triazoles as antiviral agents |
Gerald W. Shipps, Jr., Tong Wang, Kristin E. Rosner, Patrick J. Curran, Viyyoor M. Girijavallabhan |
2006-10-03 |
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Farnesyl protein transferase inhibitors |
Timothy J. Guzi, Dinanath F. Rane, Alan K. Mallams, Ronald J. Doll, Viyyoor M. Girijavallabhan +4 more |
2004-10-05 |
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Arthur G. Taveras, Ronald J. Doll, Johan Ferreira, Timothy J. Guzi, Alan K. Mallams +11 more |
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Compounds useful for inhibition of farnesyl protein transferase |
Ronald J. Doll, Anil K. Saksena, Viyyoor M. Girijavallabhan |
2004-02-10 |
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Inhibitors of farnesyl-protein transferase |
Ronald J. Doll, Johan Ferreira, Ashit K. Ganguly, Viyyoor M. Girijavallabhan, Arthur G. Taveras +4 more |
2002-08-13 |
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Farnesyl protein transferase inhibitors |
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2002-04-16 |
$81,480,000 |
