VS

Vladimir Simov

Merck: 13 patents #850 of 9,382Top 10%
LY Lycera: 8 patents #7 of 35Top 20%
Overall (All Time): #363,907 of 4,157,543Top 9%
13
Patents All Time

Issued Patents All Time

Patent #TitleCo-InventorsDate
12319671 1-pyrazolyl, 5-, 6-disubstituted indazole derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof Hua Zhou, John J. Acton, III, Michael J. Ardolino, Yi-Heng Chen, Peter H. Fuller +15 more 2025-06-03
12030872 N-heteroaryl indazole derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof William P. Kaplan, John J. Acton, III, Michael J. Ardolino, Joanna L. Chen, Peter H. Fuller +10 more 2024-07-09
11174248 Indazolyl-spiro[2.3]hexane-carbonitrile derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof John J. Acton, III, David A. Candito, J. Michael Ellis, Peter H. Fuller, Hakan Gunaydin +6 more 2021-11-16
11161854 Indazolyl-spiro[2.2]pentane-carbonitrile derivatives as LRRK2 inhibitors, pharmaceutical compositions, and uses thereof David A. Candito, Thomas H. Graham, John J. Acton, III, Ryan Chau, Joanna L. Chen +13 more 2021-11-02
10745364 Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Chad A. VanHuis, William D. Thomas, John MacLean, Brian M. Andresen +9 more 2020-08-18
10377768 Tetrahydronaphthyridine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Kenneth J. Barr, Blair T. Lapointe, Karin Ann Stein, William D. Thomas +3 more 2019-08-13
10221146 Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Chad A. VanHuis, William D. Thomas, John MacLean, Brian M. Andresen +9 more 2019-03-05
10221142 Substituted pyrazole compounds as RORgammaT inhibitors and uses thereof Blair T. Lapointe, Peter H. Fuller, Hakan Gunaydin, Kun Liu, Nunzio Sciammetta +5 more 2019-03-05
9809561 Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Chad A. VanHuis, William D. Thomas, John MacLean, Brian M. Andresen +9 more 2017-11-07
9783511 Carbamate benzoxazine propionic acids and acid derivatives for modulation of RORgamma activity and the treatment of disease Thomas D. Aicher, Chad A. VanHuis, John MacLean, Brian M. Andresen, Kenneth J. Barr +6 more 2017-10-10
9663502 2-Acylamidomethyl and sulfonylamidomethyl benzoxazine carbamates for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Chad A. VanHuis, John MacLean, Brian M. Andresen, Kenneth J. Barr +9 more 2017-05-30
9657033 Tetrahydronaphthyridine and related bicyclic compounds for inhibition of RORγ activity and the treatment of disease Thomas D. Aicher, Kenneth J. Barr, Blair T. Lapointe, Karin Ann Stein, William D. Thomas +3 more 2017-05-23
9266827 Bicyclic sulfone compounds for inhibition of RORgamma activity and the treatment of disease Thomas D. Aicher, Kenneth J. Barr, William D. Thomas, Peter L. Toogood, Chad A. Van Huis 2016-02-23