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2-pyrazine carboxamides as spleen tyrosine kinase inhibitors |
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2017-10-03 |
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Thiazole-substituted aminoheteroaryls as spleen tyrosine kinase inhibitors |
Neville J. Anthony, Brian M. Andresen, Alan B. Northrup, Kaleen Konrad Childers, Anthony Donofrio +14 more |
2017-08-29 |
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Purine inhibitors of human phosphatidylinositol 3-kinase delta |
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2017-08-15 |
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Thiazole-substituted aminoheteroaryls as Spleen Tyrosine Kinase inhibitors |
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2017-06-06 |
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Substituted pyrrolopyrimidines as HDM2 inhibitors |
Christopher J. Dinsmore, Francesc Xavier Fradera Llinas, Amit Ashokro Kudale, Michelle R. Machacek, Michael H. Reutershan +6 more |
2017-05-02 |
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Thiazole-substituted aminopyridines as spleen tyrosine kinase inhibitors |
Brian M. Andresen, Kenneth L. Arrington, Kaleen Konrad Childers, Maria Emilia Di Francesco, John Michael Ellis +8 more |
2017-03-21 |
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Triazolyl derivatives as Syk inhibitors |
Michelle R. Machacek, Eric T. Romeo, Solomon D. Kattar, Matthew Christopher, Alan B. Northrup +17 more |
2017-03-07 |
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Imidazolyl analogs as syk inhibitors |
Jongwon Lim, Michael H. Reutershan, John Michael Ellis, Kaleen Konrad Childers, Anthony Donofrio +11 more |
2016-11-08 |
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Substituted diazine and triazine spleen tyrosine kinease (Syk) inhibitors |
Andrew M. Haidle, Solomon D. Kattar, Matthew Christopher, John Michael Ellis, Christian Fischer +2 more |
2016-08-16 |
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Substituted pyridine spleen tyrosine kinase (SYK) inhibitors |
Andrew M. Haidle, Sandra Lee Knowles, Solomon D. Kattar, Denis Deschenes, Jason Burch +12 more |
2016-06-28 |
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Aminopyrimidines as Syk inhibitors |
Kaleen Konrad Childers, Maria Emilia Di Francesco, John Michael Ellis, Christian Fischer, Jonathan B. Grimm +7 more |
2016-03-22 |
| 9242984 |
Pyrazolyl derivatives as Syk inhibitors |
Michelle R. Machacek, Eric T. Romeo, Dilrukshi Vitharana, Brandon D. Cash, Tony Siu +21 more |
2016-01-26 |
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Aminopyrimidinones as interleukin receptor-associated kinase inhibitors |
W. Michael Seganish, Stephanie Nicole Brumfield, Jongwon Lim, Julius J. Matasi, William T. McElroy +6 more |
2015-12-29 |
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2-Pyridyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors |
Corey E. Bienstock, John W. Butcher, Kaleen Konrad Childers, Maria Emilia Di Francesco, Anthony Donofrio +9 more |
2015-12-22 |
| 9169260 |
Amidopyrazole inhibitors of interleukin receptor-associated kinases |
William T. McElroy, Guoqing Li, Ginny D. Ho, Zheng Tan, Sunil Paliwal +6 more |
2015-10-27 |
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Bipyridylaminopyridines as Syk inhibitors |
Denis Deschenes, John Michael Ellis, Christian Fischer, Andrew M. Haidle, Solomon D. Kattar +14 more |
2015-09-29 |
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Pyridyl aminopyridines as Syk inhibitors |
Maria Emilia Di Francesco, Andrew M. Haidle, Ryan D. Otte, John Michael Ellis, Kaleen Konrad Childers +2 more |
2015-09-01 |
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Phenyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors |
Maria Emilia Di Francesco, John Michael Ellis, Sandra Lee Knowles, Alan B. Northrup |
2015-04-14 |
| 8987456 |
3-pyridyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors |
Kaleen Konrad Childers, Anthony Donofrio, John Michael Ellis, Sandra Lee Knowles, Alan B. Northrup |
2015-03-24 |
| 8962611 |
Substituted imidazopyridines as HDM2 inhibitors |
Matthew Christopher, Francesc Xavier Fradera Llinas, Michelle R. Machacek, Michelle Martinez, Michael H. Reutershan +7 more |
2015-02-24 |
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Pyrazolo[1,5-A]pyrimidines as mark inhibitors |
Jongwon Lim, Brandon M. Taoka, Sandra Lee, Alan B. Northrup, David L. Sloman +2 more |
2015-02-03 |
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Substituted imidazopyridines as HDM2 inhibitors |
Matthew Christopher, Francesc Xavier Fradera Llinas, Michelle R. Machacek, Michelle Martinez, Michael H. Reutershan +7 more |
2014-09-30 |
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Aminopyrimidines as Syk inhibitors |
Kenneth L. Arrington, Jason Burch, Bernard Cote, Jean-Francois Fournier, Jacques Yves Gauthier +9 more |
2014-05-27 |
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Imidazo[1,2-a]pyridines and imidazo[1,2-b]pyridazines as mark inhibitors |
Mark T. Bilodeau, Jongwon Lim, Alan B. Northrup, Matthew G. Stanton, Brandon M. Taoka |
2013-11-26 |
| 8551984 |
Aminopyrimidines as SYK inhibitors |
Brian M. Andresen, Kenneth L. Arrington, Jason Burch, Kaleen Konrad Childers, Bernard Cote +24 more |
2013-10-08 |