DB

Douglas C. Beshore

Merck: 34 patents #209 of 9,382Top 3%
Overall (All Time): #100,928 of 4,157,543Top 3%
34
Patents All Time

Issued Patents All Time

Showing 25 most recent of 34 patents

Patent #TitleCo-InventorsDate
12310945 Cyclohexylglycine derivatives as selective cytotoxic agents Keith P. Moore, Rajan Anand, Remond Moningka, William D. Shipe 2025-05-27
10526336 Fused heteroaryl derivatives as orexin receptor antagonists Scott D. Kuduk, Nigel Liverton, Na Meng, Yunfu Luo 2020-01-07
10017504 Piperidine isoxazole and isothiazole orexin receptor antagonists Nigel J. Liverton, Scott D. Kuduk, Yunfu Luo, Na Meng, Tingting Yu 2018-07-10
10010539 Pyrazole, triazole and tetrazole orexin receptor antagonists Nigel J. Liverton, Scott D. Kuduk, Yunfu Luo, Na Meng 2018-07-03
9862716 TRKA kinase inhibitors, compositions and methods thereof Helen J. Mitchell, Mark E. Fraley, Andrew Cooke, Craig A. Stump, Yi-Heng Chen +10 more 2018-01-09
9828368 Oxazole orexin receptor antagonists Nigel J. Liverton, Scott D. Kuduk, Yunfu Luo, Na Meng, Tingting Yu 2017-11-28
9708273 Aryl methyl benzoquinazolinone M1 receptor positive allosteric modulators Scott D. Kuduk, Christina Ng DiMarco, Thomas J. Greshock 2017-07-18
9695163 Thiazole orexin receptor antagonists Nigel Liverton, Scott D. Kuduk, Yunfu Luo, Na Meng, Tingting Yu 2017-07-04
9365562 1,3 substituted azetidine PDE10 inhibitors Christopher D. Cox, June J. Kim, Scott D. Kuduk, Carol A. McVean, Thomas S. Reger +1 more 2016-06-14
9359348 Cyclopropyl imidazopyridine PDE10 inhibitors Scott D. Kuduk, Thomas S. Reger 2016-06-07
9206200 N-linked lactam M1 receptor positive allosteric mogulators Scott D. Kuduk, Zhi-Qiang Yang, Youheng Shu, Daniel L. Pitts 2015-12-08
9139576 Aminomethyl biaryl benzotriazole derivatives Robert M. Garbaccio, Scott D. Kuduk, Adam W. Johnson, Jason W. Skudlarek 2015-09-22
8975286 Ether benzotriazole derivatives Vadim Dudkin, Mark E. Fraley, Cheng Wang, Robert M. Garbaccio, Scott K. Kuduk +1 more 2015-03-10
8895580 Quinolinone-pyrazolone M1 receptor positive allosteric modulators Scott D. Kuduk, Robert M. DiPardo 2014-11-25
8883810 Aryl methyl benzoquinazolinone M1 receptor positive allosteric modulators Scott D. Kuduk, Christina Ng Di Marco, Thomas J. Greshock 2014-11-11
8883850 Naphthalene carboxamide M1 receptor positive allosteric modulators Christina Ng DiMarco, Scott D. Kukuk 2014-11-11
8785482 Cyclohexene benzotriazole derivatives Scott D. Kuduk 2014-07-22
8785481 Ether benzotriazole derivatives Vadim Dudkin, Robert M. Garbaccio, Adam W. Johnson, Scott D. Kuduk, Jason W. Skudlarek +2 more 2014-07-22
8697690 Isoindolone M1 receptor positive allosteric modulators Scott D. Kuduk, Youheng Shu, Zhi-Qiang Yang 2014-04-15
8653079 Pyrazolo [4,3-C] cinnolin-3-one M1 receptor positive allosteric modulators Scott D. Kuduk 2014-02-18
8557832 Aryl methyl benzoquinazolinine M1 receptor positive allosteric modulators Scott D. Kuduk, Christina Ng Di Marco, Thomas J. Greshock 2013-10-15
8507494 Heterocyclic quinolizine derived M1 receptor positive allosteric modulators Scott D. Kuduk 2013-08-13
8486946 Pyrazolo [4,3-c] cinnolin-3-one M1 receptor positive allosteric modulators Scott D. Kuduk 2013-07-16
8426438 Heterocyclic-fused pyrazolo[4,3-c]pyridin-3-one M1 receptor positive allosteric modulators Scott D. Kuduk 2013-04-23
8383638 Aminobenzoquinazolinone M1 receptor positive allosteric modulators Scott D. Kuduk, Christina Ng DiMarco, Thomas J. Greshock 2013-02-26