| 5710275 |
7.beta.-substituted-4-aza-5.alpha.-androstan-3-ones as 5.alpha.-reductase inhibitors |
Raman K. Bakshi, Gary H. Rasmusson, Richard L. Tolman, Gool F. Patel, Georgianna Harris +1 more |
1998-01-20 |
$89,344,000 |
| 5693809 |
Substituted 4-aza-5.alpha.-androstan-ones as 5.alpha.-reductase inhibitors |
Philippe L. Durette, William K. Hagmann, Gary H. Rasmusson, Richard L. Tolman, Ihor E. Kopka +4 more |
1997-12-02 |
$56,997,000 |
| 5639741 |
17-amino substituted 4-azasteroid 5.alpha.-reductase inhibitors |
Jeffrey P. Bergman, Richard L. Tolman |
1997-06-17 |
$146,641,000 |
| 5620986 |
17 urea, thiourea, thiocarbamyl and carbamyl4-azasteroid 5-reductase inhibitors useful in the prevention and treatment of hyperandrogenic disorders |
Richard L. Tolman |
1997-04-15 |
$57,611,000 |
| 5610162 |
Ester derivatives of 4-aza-steroids |
Gary H. Rasmusson, Richard L. Tolman, Shu S. Yang |
1997-03-11 |
$104,011,000 |
| 5536727 |
17-Ethers and thioethers of 4-aza-steroids |
Richard L. Tolman, Gary H. Rasmusson, Raman K. Bakshi, Shu S. Yang |
1996-07-16 |
$47,913,000 |
| 5068248 |
N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors |
Allan N. Tischler, Philippe L. Durette, Kathleen M. Rupprecht, Timothy Francis Gallagher, Marvin M. Goldenberg +1 more |
1991-11-26 |
$28,877,000 |
| 4999436 |
Aryl-substituted thiophene 3-ols, derivatives and analogs useful as lipoxgenase inhibitors |
Debra L. Allison, Charles G. Caldwell, Kathleen M. Rupprecht |
1991-03-12 |
$157,211,000 |
| 4885276 |
"Cyclosporin analogs with modified ""C-9 amino acids""" |
— |
1989-12-05 |
$27,146,000 |
| 4814501 |
Process for preparing N,N-dimethyl 2-(methylthio) benzamides and analogs |
Robert K. Baker, Philippe L. Durette, Robert A. Frankshun |
1989-03-21 |
$13,520,000 |
| 4800211 |
5-methylthio-3-hydroxybenzo [b]thiophene-2-carboxamide derivatives as cyclooxygenase and lipoxygenase inhibitors |
Allan N. Tischler, Philippe L. Durette, Thomas J. Lanza, Jr. |
1989-01-24 |
$14,093,000 |
| 4798823 |
"New cyclosporin analogs with modified ""C-9 amino acids""" |
— |
1989-01-17 |
$15,401,000 |
| 4782080 |
N-alkenyl-2-hydroxybenzo(b)thiophene-3-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors |
— |
1988-11-01 |
$12,833,000 |
| 4760086 |
N-alkenyl-3-hydroxybenzo[b]thiophene-2-carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors |
Allan N. Tischler, Philippe L. Durette, Kathleen M. Rupprecht, Timothy Francis Gallagher, Debra L. Allison +1 more |
1988-07-26 |
$13,870,000 |
| 4720503 |
N-substituted fused-heterocyclic carboxamide derivatives as dual cyclooxygenase and lipoxygenase inhibitors |
Allan N. Tischler, Debra L. Allison |
1988-01-19 |
$26,198,000 |
| 4663344 |
Anti-inflammatory and analgesic 3-hydroxybenzo[b]thiophene derivatives, compositions, and method of use therefor |
Philippe L. Durette, Kathleen M. Rupprecht, Allan N. Tischler, Timothy Francis Gallagher |
1987-05-05 |
$13,409,000 |
| 4536512 |
5-(2,3-Dihydro-1H-pyrrolizin-5-oyl)-2,3-dihyd ro-1H-pyrrolizine-1-alkanoic or carboxylic acids and use thereof as anti-inflammatory and analgesic agents |
Tesfaye Biftu, Peter L. Barker |
1985-08-20 |
$5,757,000 |
| 4533671 |
5-(2,3-Dihydro-1H-pyrrolizin-5-oyl)-2-alkanoic or carboxylic acids and analogs as anti-inflammatory and analgesic agents |
Tesfaye Biftu, Peter L. Barker |
1985-08-06 |
$9,164,000 |
| 4440779 |
Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents |
James B. Doherty, Conrad P. Dorn, Debra L. Allison, Tsung-Ying Shen |
1984-04-03 |
$4,370,000 |
| 4431655 |
2,4-Disubstituted-1,2,5-thiadiazol-3(2H)-one antimicrobials |
Richard A. Dybas, Nathaniel Grier |
1984-02-14 |
$4,328,000 |
| 4402959 |
Antimicrobial compositions |
Richard A. Dybas |
1983-09-06 |
$7,583,000 |
| 4391812 |
2-(Substitutedpiperidylmethyl) propane nitriles and compositions thereof |
Richard A. Dybas, Nathaniel Grier |
1983-07-05 |
$17,208,000 |
| 4380645 |
Process for preparing Benzoxepino- or Benzthiapino[4,3-b]pyrrole-2-acetic acids |
Paul E. Finke, Debra L. Allison |
1983-04-19 |
$28,102,000 |
| 4362877 |
2,4-Disubstituted-1,2,5-thiadiazol-3(2H)-one antimicrobials |
Richard A. Dybas, Nathaniel Grier |
1982-12-07 |
$6,185,000 |
| 4342872 |
2-(Substitutedpiperidylmethyl) propene and propane nitriles |
Nathaniel Grier, Richard A. Dybas |
1982-08-03 |
$2,025,000 |
