CB

Craig D. Boyle

SC Schering: 18 patents #131 of 2,442Top 6%
Merck: 11 patents #1,033 of 9,382Top 15%
Overall (All Time): #132,013 of 4,157,543Top 4%
29
Patents All Time

Issued Patents All Time

Showing 25 most recent of 29 patents

Patent #TitleCo-InventorsDate
9301929 Substituted biaryl derivatives and methods of use thereof Claire M. Lankin, William J. Greenlee, Joel M. Harris 2016-04-05
9161924 Factor IXa inhibitors William J. Greenlee, Samuel Chackalamannil, Claire M. Lankin 2015-10-20
8907095 Bicyclic heterocycle derivatives and their use as modulators of the activity of GPR119 Yan Xia, William J. Greenlee, Samuel Chackalamannil, Charles Lee Jayne 2014-12-09
8822480 Bicyclic heterocycle derivatives and use thereof as GPR119 modulators Santhosh F. Neelamkavil, Samuel Chackalamannil, William J. Greenlee, Bernard R. Neustadt, Andrew Stamford 2014-09-02
8815876 Bicyclic heterocycle derivatives and methods of use thereof Santhosh F. Neelamkavil, Bernard R. Neustadt, Samuel Chackalamannil, William J. Greenlee 2014-08-26
8604195 Substituted bicyclic piperidinyl- and piperazinyl-sulfonamides useful to inhibit 11β-hydroxysteroid dehydrogenase type-1 Unmesh Shah, Samuel Chackalamannil 2013-12-10
8580807 Bicyclic piperidine and piperazine derivatives as GPCR modulators for the treatment of obesity, diabetes and other metabolic disorders Claire M. Lankin, Unmesh Shah, William J. Greenlee, Samuel Chackalamannil 2013-11-12
8466149 6-substituted sulfonyl azabicyclo[3.2.1]octanes useful to inhibit 11β-hydroxysteroid dehydrogenase type-I Samuel Chackalamannil, Unmesh Shah, Claire M. Lankin 2013-06-18
RE44205 Adenosine A2a receptor antagonists Bernard R. Neustadt, Neil A. Lindo, William J. Greenlee, Deen Tulshian, Lisa S. Silverman +2 more 2013-05-07
8389532 7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(1-propynyl)-7H-pyrazolo-[4,3-E]-[1,2,4]-triazolo-[1,5-C]-pyrimidin-5-amine Samuel Chackalamannil, Unmesh Shah, Jean E. Lachowicz 2013-03-05
8318751 Pyrimidinone derivatives and methods of use thereof Samuel Chackalamannil, Claire M. Lankin, Unmesh Shah, Bernard R. Neustadt, Hong Liu +1 more 2012-11-27
7709492 Pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Bernard R. Neustadt, Jinsong Hao, Hong Liu, Samuel Chackalamannil, Unmesh Shah +2 more 2010-05-04
7572802 7-[2-[4-(6-fluoro-3-methyl-1,2-benzisoxazol-5-yl)-1-piperazinyl]ethyl]-2-(1-propynyl)-7H-pyrazolo-[4,3-e]-[1,2,4]-triazolo-[1,5-C]-pyrimidin-5-amine Samuel Chackalamannil, Unmesh Shah, Jean E. Lachowicz 2009-08-11
7531544 Xanthine phosphodiesterase V inhibitors Samuel Chackalamannil, Yuguang Wang, Andrew Stamford 2009-05-12
7465740 2-heteroaryl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Bernard R. Neustadt, Samuel Chackalamannil, Joel M. Harris, Claire M. Lankin, Hong Liu +2 more 2008-12-16
7368449 2-alkynyl- and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Bernard R. Neustadt, Jinsong Hao, Hong Liu, Samuel Chackalamannil, Unmesh Shah +1 more 2008-05-06
7312223 Metabolite of xanthine Phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction Anima Ghosal, Wei Tong, Swapan Chowdhury, Shmuel Zbaida, Mark A. Wirth +3 more 2007-12-25
7268141 Xanthine phosphodiesterase V inhibitors Samuel Chackalamannil, Yuguang Wang, Andrew Stamford 2007-09-11
7192962 Xanthine phosphodiesterase V inhibitor polymorphs Vilas Hareshwar Dahanukar, Hoa N. Nguyen, Cecilia Orr, Funcheng Zhang, Ilia Zavialov +3 more 2007-03-20
6916811 Adenosine A2a receptor antagonists Samuel Chackalamannil, William J. Greenlee, Unmesh Shah, Yan Xia 2005-07-12
6897217 2-Alkynyl-and 2-alkenyl-pyrazolo-[4,3-e]-1,2,4-triazolo-[1,5-c]-pyrimidine adenosine A2a receptor antagonists Bernard R. Neustadt, Jinsong Hao, Hong Liu, Samuel Chackalamannil, Unmesh Shah +1 more 2005-05-24
6897216 Adenosine A2a receptor antagonists Bernard R. Neustadt, Neil A. Lindo, William J. Greenlee, Deen Tulshian, Lisa S. Silverman +2 more 2005-05-24
6890936 Muscarinic antagonists William J. Greenlee, Samuel Chackalamannil 2005-05-10
6821978 Xanthine phosphodiesterase V inhibitors Samuel Chackalamannil, Yuguang Wang, Andrew Stamford 2004-11-23
6632828 Substituted imidazole neuropeptide Y Y5 receptor antagonists Andrew Stamford, Ying Huang 2003-10-14