Issued Patents All Time
Showing 1–25 of 74 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12409173 | Repurposing FDA-approved drugs as a novel cancer therapeutic avenue through inhibition of PRMT5 | Tao Lu, Lakshmi Milind PRABHU | 2025-09-09 |
| 12264137 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +4 more | 2025-04-01 |
| 12049466 | Fused bicyclic compounds useful as ubiquitin-specific peptidase 30 inhibitors | Alexandre Joseph Buckmelter | 2024-07-30 |
| 11919839 | Alpha-cinnamide compounds and compositions as HDAC8 inhibitors | Kenneth W. Bair, Nicholas Barczak, Bingsong Han, David R. Lancia, Jr., Cuixian Liu +5 more | 2024-03-05 |
| 11891365 | 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +6 more | 2024-02-06 |
| 11814386 | Fused pyrrolines which act as ubiquitin-specific protease 30 (USP30) inhibitors | Alex J. Buckmelter, Justin Andrew Caravella, Hongbin Li, Steven Mischke, David Richard +1 more | 2023-11-14 |
| 11535618 | Fused pyrrolines which act as ubiquitin-specific protease 30 (USP30) inhibitors | Alex J. Buckmelter, Justin Andrew Caravella, Hongbin Li, Steven Mischke, David Richard +1 more | 2022-12-27 |
| 11535607 | Isoindolines as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Jennifer R. Thomason, Bingsong Han, Aleksandra Rudnitskaya +1 more | 2022-12-27 |
| 11345672 | Methods using HDAC11 inhibitors | Jennifer Lee, Nicholas Barczak, Jaime Escobedo, Chiara Conti, Bingsong Han +6 more | 2022-05-31 |
| 11299484 | Inhibiting fatty acid synthase (FASN) | Mary-Margaret Zablocki, Scot Richard Mente, Christopher J. Dinsmore, Zhongguo Wang, Xiaozhang Zheng | 2022-04-12 |
| 11279681 | 3-alkyl bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +5 more | 2022-03-22 |
| 11274085 | 3-aryl-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +4 more | 2022-03-15 |
| 11274084 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +4 more | 2022-03-15 |
| 11267805 | Solid forms of (4-(2-fluoro-4-(1-methyl-1H-benzo[d]imidazol-5-yl)benzoyl) piperazine-1-yl)(1-hydroxycyclopropyl)methanone | George P. Luke, Stephen Hubbs, Shawn Schiller, Robert Wenslow, Yawei Shi +1 more | 2022-03-08 |
| 11247987 | Inhibiting ubiquitin specific peptidase 30 | Justin Andrew Caravella, Bingsong Han, Cuixian Liu, Stephanos Ioannidis, Alexandre Joseph Buckmelter +3 more | 2022-02-15 |
| 11111229 | Tetrahydroquinoline compositions as BET bromodomain inhibitors | Kenneth W. Bair, Torsten Herbertz, Goss S. Kauffman, Katherine J. Kayser-Bricker, George P. Luke +3 more | 2021-09-07 |
| 11084831 | Benzopiperazine compositions as BET bromodomain inhibitors | Kenneth W. Bair, Torsten Herbertz, Goss S. Kauffman, Katherine J. Kayser-Bricker, George P. Luke +4 more | 2021-08-10 |
| 10995078 | Compounds and compositions for inhibition of FASN | Kenneth W. Bair, David R. Lancia, Jr., Hongbin Li, James Loch, Wei Lu +3 more | 2021-05-04 |
| 10988441 | Alpha-cinnamide compounds and compositions as HDAC8 inhibitors | Kenneth W. Bair, Nicholas Barczak, Bingsong Han, David R. Lancia, Jr., Cuixian Liu +5 more | 2021-04-27 |
| 10988450 | 3-alkyl-4-amido-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +6 more | 2021-04-27 |
| 10875848 | Inhibiting fatty acid synthase (FASN) | Mary-Margaret Zablocki, Scot Richard Mente, Christopher J. Dinsmore, Zhongguo Wang, Xiaozhang Zheng | 2020-12-29 |
| 10829461 | 3-aryl-4-amido-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +4 more | 2020-11-10 |
| 10829462 | 3-alkyl bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +5 more | 2020-11-10 |
| 10822316 | 3-aryl-bicyclic [4,5,0] hydroxamic acids as HDAC inhibitors | Xiaozhang Zheng, Pui Yee Ng, Bingsong Han, Jennifer R. Thomason, Mary-Margaret Zablocki +4 more | 2020-11-03 |
| 10800750 | Compounds and compositions for inhibition of FASN | Kenneth W. Bair, David R. Lancia, Jr., Hongbin Li, James Loch, Wei Lu +3 more | 2020-10-13 |