Issued Patents All Time
Showing 26–50 of 59 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 10377773 | Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang | 2019-08-13 |
| 10377767 | Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang +1 more | 2019-08-13 |
| 10351571 | Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang | 2019-07-16 |
| 10294206 | Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2019-05-21 |
| 10280150 | Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2019-05-07 |
| 10266495 | Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2019-04-23 |
| 10253015 | Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2019-04-09 |
| 10005734 | Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2018-06-26 |
| 10000495 | Pyrrolotriazinones and imidazotriazinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang | 2018-06-19 |
| RE46856 | Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis | Martin F. Hentemann, Jill Wood, William Scott, Martin Michels, Ann-Marie Bullion +2 more | 2018-05-22 |
| 9938300 | Isothiazolopyrimidinones, pyrazolopyrimidinones, and pyrrolopyrimidinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang | 2018-04-10 |
| 9932351 | Thienopyrimidinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang +1 more | 2018-04-03 |
| 9902728 | Pyrrolo and pyrazolopyrimidines as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang +6 more | 2018-02-27 |
| 9840491 | Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors | Stephanos Ioannidis, Adam Charles Talbot, Bruce Follows, Alexandre Joseph Buckmelter, Minghua Wang +1 more | 2017-12-12 |
| 9834539 | Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2017-12-05 |
| 9815817 | Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R Bruce Diebold +4 more | 2017-11-14 |
| 9771349 | Pyridinyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2017-09-26 |
| 9624216 | Quinolinone five-membered heterocyclic compounds as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2017-04-18 |
| 9624175 | Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors | Jian Lin, Anna Ericsson, Gary Gustafson, Zhongguo Wang, R. Bruce Diebold +4 more | 2017-04-18 |
| 8859538 | Uses of substituted imidazoheterocycles | R. Paul Beckett, Richard Foster, Christelle Henault, Janet L. Ralbovsky, Carla Gauss +3 more | 2014-10-14 |
| 8466283 | Substituted 2,3-dihydroimidazo[1,2-c]quinazoline derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis | Martin F. Hentemann, Jill Wood, William Scott, Martin Michels, Ann-Marie Bullion +2 more | 2013-06-18 |
| 8431565 | Substituted imidazoheterocycles | R. Paul Beckett, Richard Foster, Christelle Henault, Janet L. Ralbovsky, Carla Gauss +4 more | 2013-04-30 |
| 8013166 | Preparation and use of aryl alkyl acid derivatives for the treatment of obesity | Roger Smith, Philip Coish, Miao Dai, Susan Jenkins, Derek Lowe +5 more | 2011-09-06 |
| 7968576 | Preparation and use of aryl alkyl acid derivatives for the treatment of obesity | Roger Smith, Philip Coish, Miao Dai, Susan Jenkins, Derek Lowe +5 more | 2011-06-28 |
| 7759376 | Preparation and use of biphenyl-4-yl-carbonylamino acid derivatives for the treatment of obesity | Roger Smith, Stephen O'Connor, Philip Coish, Derek Lowe, Roger B. Clark +3 more | 2010-07-20 |