| 11352360 |
TGF-beta inhibitors |
Todd Kinsella, Marina Gelman, Hui Hong, Ihab Darwish, Rajinder Singh +6 more |
2022-06-07 |
| 10961239 |
TGF beta receptor antagonists |
Robert M. Borzilleri, Upender Velaparthi, Chetan Padmakar Darne, Manjunatha Narayana Rao Kamble, Balaji Seshadri +3 more |
2021-03-30 |
| 10287295 |
TGF-β inhibitors |
Todd Kinsella, Marina Gelman, Hui Hong, Ihab Darwish, Rajinder Singh +6 more |
2019-05-14 |
| 9884868 |
TGF-beta inhibitors |
Todd Kinsella, Marina Gelman, Hui Hong, Ihab Darwish, Rajinder Singh +6 more |
2018-02-06 |
| 9598423 |
Substituted 4,5,6,7-tetrahydropyrazolo[1,5-A]pyrazine derivatives as casein kinase 1 D/E inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Mark D. Wittman, Bradley C. Pearce, Erika M. V. Araujo +13 more |
2017-03-21 |
| 9556179 |
Substituted imidazoles as casein kinase 1 D/E inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Dharmpal S. Dodd, Anthony J. Sampognaro, Mark D. Wittman +3 more |
2017-01-31 |
| 9475817 |
Pyrazole substituted imidazopyrazines as casein kinase 1 d/e inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Dharmpal S. Dodd, Christopher P. Mussari, Mark D. Wittman +2 more |
2016-10-25 |
| 9273058 |
Substituted pyrazolo-piperazines as casein kinase 1 δ/ε inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Mark D. Wittman, Bradley C. Pearce, Erika M. V. Araujo +13 more |
2016-03-01 |
| 9242967 |
Substituted bicyclic heteroaryl compounds |
Upender Velaparthi |
2016-01-26 |
| 9145419 |
Imidazopyridazinyl compounds |
Upender Velaparthi, James Aaron Balog |
2015-09-29 |
| 8592579 |
Pyrrolotriazine kinase inhibitors |
Mark D. Wittman, Harold Mastalerz, Kurt Zimmermann, Mark G. Saulnier, Upender Velaparthi +6 more |
2013-11-26 |
| 8415340 |
Triazine kinase inhibitors |
Upender Velaparthi, Mark D. Wittman, David R. Langley |
2013-04-09 |
| 7879855 |
Pyrrolotriazine kinase inhibitors |
Mark D. Wittman, Harold Mastalerz, Kurt Zimmermann, Mark G. Saulnier, Upender Velaparthi +6 more |
2011-02-01 |
| 7534792 |
Pyrrolotriazine kinase inhibitors |
Mark D. Wittman, Harold Mastalerz, Kurt Zimmermann, Mark G. Saulnier, Upender Velaparthi +6 more |
2009-05-19 |
| 7223757 |
Tyrosine kinase inhibitors |
Mark D. Wittman, Neelakantan Balasubramanian, Upender Velaparthi, Kurt Zimmermann, Mark G. Saulnier +6 more |
2007-05-29 |
| 7081454 |
Tyrosine kinase inhibitors |
Mark D. Wittman, Neelakantan Balasubramanian, Upender Velaparthi, Kurt Zimmermann, Mark G. Saulnier +6 more |
2006-07-25 |
| 6784167 |
17-beta-hydroxysteroid dehydrogenase-II inhibitors |
Jill Wood, Jeremy Lee Baryza, Catherine Brennan, Soongyu Choi, James H. Cook, II +8 more |
2004-08-31 |
| 6353006 |
Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
Brian R. Dixon, Cedo Martin Bagi, Catherine Brennan, David R. Brittelli, William Bullock +11 more |
2002-03-05 |