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Isofuranone compounds useful as HPK1 inhibitors |
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Imidazo-pyridazine derivatives as casein kinase 1 δ/ϵ inhibitors |
Upender Velaparthi, Selvakumar Kumaravel, Arul Mozhi Selvan Subbiah Karupplah, Shilpa Holehatti Maheshwarappa, Chandrasekhar Reddy Rachamreddy |
2018-05-01 |
| 9598423 |
Substituted 4,5,6,7-tetrahydropyrazolo[1,5-A]pyrazine derivatives as casein kinase 1 D/E inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Peiying Liu, Bradley C. Pearce, Erika M. V. Araujo +13 more |
2017-03-21 |
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Substituted imidazoles as casein kinase 1 D/E inhibitors |
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2017-01-31 |
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Pyrazole substituted imidazopyrazines as casein kinase 1 d/e inhibitors |
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2016-10-25 |
| 9273058 |
Substituted pyrazolo-piperazines as casein kinase 1 δ/ε inhibitors |
Upender Velaparthi, Chetan Padmakar Darne, Peiying Liu, Bradley C. Pearce, Erika M. V. Araujo +13 more |
2016-03-01 |
| 8592579 |
Pyrrolotriazine kinase inhibitors |
Harold Mastalerz, Kurt Zimmermann, Mark G. Saulnier, Upender Velaparthi, Dolatrai M. Vyas +6 more |
2013-11-26 |
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Triazine kinase inhibitors |
Upender Velaparthi, Peiying Liu, David R. Langley |
2013-04-09 |
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Thiazolyl compounds useful as kinase inhibitors |
Anne Marinier, Marco Dodier, Stephan Roy, Kurt Zimmermann, Xiaopeng Sang +2 more |
2013-01-01 |
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Pyrrolotriazine kinase inhibitors |
Kurt Zimmermann, Xiaopeng Sang |
2012-09-11 |
| 8198438 |
Pyrrolotriazine kinase inhibitors |
Anthony J. Sampognaro |
2012-06-12 |
| 8148400 |
Thiazolyl compounds useful as kinase inhibitors |
Anne Marinier, Claude A. Quesnelle, Marco Dodier, Stephan Roy, Patrice Gill +1 more |
2012-04-03 |
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Pyrrolotriazine kinase inhibitors |
Harold Mastalerz, Kurt Zimmermann, Mark G. Saulnier, Upender Velaparthi, Dolatrai M. Vyas +6 more |
2011-02-01 |
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Pyrrolotriazine kinase inhibitors |
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2009-05-19 |
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Tyrosine kinase inhibitors |
Francis Beaulieu, Carl Ouellet, Kurt Zimmermann, Upender Velaparthi |
2008-12-30 |
| 7312215 |
Benzimidazole C-2 heterocycles as kinase inhibitors |
Francis Beaulieu, Anne Marinier, Carl Ouellet, Stephan Roy |
2007-12-25 |
| 7232826 |
Tyrosine kinase inhibitors |
Upender Velaparthi |
2007-06-19 |
| 7223757 |
Tyrosine kinase inhibitors |
Neelakantan Balasubramanian, Upender Velaparthi, Kurt Zimmermann, Mark G. Saulnier, Peiying Liu +6 more |
2007-05-29 |
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Tyrosine kinase inhibitors |
Francis Beaulieu, Carl Ouellet, Kurt Zimmermann, Upender Velaparthi |
2007-03-13 |
| 7081454 |
Tyrosine kinase inhibitors |
Neelakantan Balasubramanian, Upender Velaparthi, Kurt Zimmermann, Mark G. Saulnier, Peiying Liu +6 more |
2006-07-25 |
| 6455575 |
Phosphonooxymethyl ethers of taxane derivatives |
Jerzy Golik, Dolatrai M. Vyas, John J. Wright, Henry Wong, John F. Kadow +4 more |
2002-09-24 |
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Taxane anticancer agents |
John F. Kadow, Wendy S. Schwartz, Paul Michael Scola, Qiufen Xue, Mu-Jen Wu |
2002-03-26 |
| 6201140 |
7-0-ethers of taxane derivatives |
Henry Wong |
2001-03-13 |
| 5977386 |
6-thio-substituted paclitaxels |
Andrew J. Staab, John F. Kadow, Dolatrai M. Vyas, Harold Mastalerz |
1999-11-02 |
| 5912264 |
6-halo-or nitrate-substituted paclitaxels |
John F. Kadow |
1999-06-15 |