BM

Bruce J. Melancon

VU Vanderbilt University: 12 patents #46 of 1,609Top 3%
📍 Nashville, TN: #121 of 2,243 inventorsTop 6%
🗺 Tennessee: #1,501 of 20,272 inventorsTop 8%
Overall (All Time): #413,842 of 4,157,543Top 10%
12
Patents All Time

Issued Patents All Time

Showing 1–12 of 12 patents

Patent #TitleCo-InventorsDate
10654847 Substituted 2-(4-heterocyclylbenzyl)isoindolin-1-one analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M1 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Corey R. Hopkins, Michael S. Poslusney +1 more 2020-05-19
10189857 Positive allosteric modulators of the muscarinic acetylcholine receptor M4 Craig W. Lindsley, P. Jeffrey Conn, Darren W. Engers, Alison R. Gregro 2019-01-29
9868746 Substituted 5-aminothieno[2,3-C]pyridazine-6-carboxamide analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M4 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, James C. Tarr, James M. Salovich +1 more 2018-01-16
9637498 Substituted thieno[2,3-C]pyridazine-6-carboxamide analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M4 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Michael S. Poslusney, James C. Tarr 2017-05-02
9586964 Substituted 2-(4-heterocyclylbenzyl)isoindolin-1-one analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M1 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Corey R. Hopkins, Michael S. Poslusney +1 more 2017-03-07
9493481 Substituted 5-aminothieno[2,3—C]pyridazine-6-carboxamide analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M4 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, James C. Tarr, James M. Salovich +1 more 2016-11-15
9073935 Substituted benzylspiroindolin-2-one analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M1 Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Corey R. Hopkins, Michael S. Poslusney 2015-07-07
9056876 Substituted 1H-pyrazolo[3′,4′,4,5]thieno[2,3-b]pyridin-3-amine analogs as positive allosteric modulators of the muscarinic acetylcholine receptor M4 Jeffrey P. Conn, Craig W. Lindsley, Michael R. Wood, Corey R. Hopkins, James M. Salovich 2015-06-16
9029563 Substituted 1-benzylindolin-2-one analogs as positive allosteric modulators of muscarinic acetylcholine M1 receptors Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Michael S. Poslusney 2015-05-12
9012445 Substituted 4-(1H-pyrazol-4-yl)benzyl analogues as positive allosteric modulators of mAChR M1 receptors Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Michael S. Poslusney, James C. Tarr 2015-04-21
8697691 Alkyl 3-((2-amidoethyl)amino)-8-azabicyclo[3.2.1]octane-8-carboxylate analogs as selective M1 agonists and methods of making and using same P. Jeffrey Conn, Craig W. Lindsley, Michael R. Wood, Rocco D. Gogliotti, Colleen M. Niswender +1 more 2014-04-15
8697888 Substituted (1-(methylsulfonyl)azetidin-3-yl)(heterocycloalkyl)methanone analogs as antagonists of muscarinic acetylcholine M1 receptors Craig W. Lindsley, P. Jeffrey Conn, Michael R. Wood, Yiu-Yin Cheung 2014-04-15