Issued Patents All Time
Showing 1–25 of 27 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 9422244 | Synthesis of substituted pyrazoline carboxamidine derivatives | Arnold Van Loevezijn, Gerrit A. Barf, Arnold P. den Hartog | 2016-08-23 |
| 8937184 | 1H-imidazole derivatives as cannabinoid CB2 receptor modulators | Herman H. Van Stuivenberg, Bernard J. Van Vliet | 2015-01-20 |
| 8729101 | 1H-imidazole derivative having CB1, agonistic, CB1 partial agonistic or CB1 antagnistic activity | Cornelis G. Kruse, Arnoldus H. J. Herremans, Herman H. Van Stuivenberg | 2014-05-20 |
| 8575148 | Spiro azepane-oxazolidinones as Kv1.3 potassium channel blockers | Pieter Smid, Michael Mlinaric, Konrad Koehler, Sara Nuñez Garcia, Elmar Wegener | 2013-11-05 |
| 8461184 | Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonists | Cornelis G. Kruse, Bernard J. Vliet Van | 2013-06-11 |
| 8410135 | 4,5 dihydro-(1H)-pyrazole derivatives as cannabinoid CB1 receptor modulators | Hendrik C. Wals, Bernard J. Van Vliet, Mahmut Yildirim | 2013-04-02 |
| 8138174 | Compounds with a combination of cannabinoid CB1 antagonism and serotonin reuptake inhibition | Cornelis G. Kruse | 2012-03-20 |
| 8063062 | Compounds with a combination of cannabinoid-CB1 antagonism and acetylcholinesterase inhibition | Cornelis G. Kruse, Belal Shadid | 2011-11-22 |
| 7928134 | 5-aryl-4,5-dihydro-(1H)-pyrazolines as cannabinoid CB1 receptor agonists | Hicham Zilaout, Bernard J. Van Vliet | 2011-04-19 |
| 7786144 | Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonists | Cornelis G. Kruse, Bernard J. Van Vliet | 2010-08-31 |
| 7745476 | 1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity | Cornelis G. Kruse, Herman H. Van Stuivenberg | 2010-06-29 |
| 7608718 | 4,5-dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity | Cornelis G. Kruse, Jacobus Tipker, Herman H. Van Stuivenberg, Arnoldus H. J. Herremans | 2009-10-27 |
| 7528162 | 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity | Cornelis G. Kruse, Jacobus Tipker, Arnoldus H. J. Herremans, Herman H. Van Stuivenberg | 2009-05-05 |
| 7524867 | Tetrasubstituted imidazole derivatives as cannabinoid CB1 receptor modulators with a high CB1/CB2 receptor subtype selectivity | Henderik C. Wals, Cornelis G. Kruse | 2009-04-28 |
| 7498348 | 1 H-imidazole derivatives as cannabinoid receptor modulators | Cornelis G. Kruse, Herman H. Van Stuivenberg, Hiskias G. Keizer | 2009-03-03 |
| 7495108 | Imidazoline derivatives having CB1-antagonistic activity | Cornelis G. Kruse, Herman H. Van Stuivenberg | 2009-02-24 |
| 7342032 | Thiazole derivatives having CB1-antagonistic, agonistic or partial agonistic activity | Cornelis G. Kruse, Arnoldus H. J. Herremans, Herman H. Van Stuivenberg, Jessica A. R. Dijksman, Andrew McCreary | 2008-03-11 |
| 7319110 | 1H-1,2,4-triazole-3-carboxamide derivatives having cannabinoid-CB1 receptor agonistic, partial agonistic, inverse agonistic or antagonistic activity | Cornelis G. Kruse, Andrew McCreary, Herman H. Van Stuivenberg | 2008-01-15 |
| 7271189 | 1H-imidazole derivatives as cannabinoid receptor modulators | Cornelis G. Kruse, Herman H. Van Stuivenberg, Hiskias G. Keizer | 2007-09-18 |
| 7186741 | Neurotensin active 2,3,diaryl-pyrazolidine derivatives | Roelof Feenstra, Maria L. Pras-Raves, Cornelis G. Kruse, Herman H. Van Stuivenberg, Tinka Tuinstra +1 more | 2007-03-06 |
| 7173044 | Imidazoline derivatives having CB1-antagonistic activity | Cornelis G. Kruse, Herman H. Van Stuivenberg | 2007-02-06 |
| 7109216 | 1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1-antagonistic activity | Cornelis G. Kruse, Arnoldus H. J. Herremans, Herman Stuivenberg | 2006-09-19 |
| 6974810 | 4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity | Cornelis G. Kruse, Jacobus Tipker, Herman H. Van Stuivenberg, Arnoldus H. J. Herremans | 2005-12-13 |
| 6476060 | 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity | Cornelis G. Kruse, Jacobus Tipker, Martinus Th.M. Tulp, Bernard J. Van Vliet | 2002-11-05 |
| 6335326 | Benzisoxazole derivatives having d4-antagonistic activity | Jacobus A. J. den Hartog, Gerben M. Visser, Bartholomeus J. Van Steen, Martinus T. M. Tulp, Eric Ronken +1 more | 2002-01-01 |