Issued Patents All Time
Showing 1–25 of 31 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12139489 | Polycyclic carbamoylpyridone derivative | Yuto UNOH | 2024-11-12 |
| 12098151 | Arenavirus growth inhibitor comprising polycyclic carbamoyl pyridone derivative | Akihiro Ishii, Akihiko Sato, Makoto Kawai | 2024-09-24 |
| 11814368 | Triazine derivatives having virus replication inhibitory activity and pharmaceutical composition comprising the same | Yuki Tachibana, Shota UEHARA, Yuto UNOH, Kenji NAKAHARA, Yukiko YAMATSU +2 more | 2023-11-14 |
| 11649236 | Polycyclic carbamoylpyridone derivative | Yuto UNOH | 2023-05-16 |
| 11492352 | Arenavirus growth inhibitor comprising polycyclic carbamoylpyridone derivative | Akihiro Ishii, Akihiko Sato, Makoto Kawai | 2022-11-08 |
| 11453669 | Polycyclic pyridone derivative | — | 2022-09-27 |
| 11267823 | Substituted 1,2,3,3a,4,5,7,9,13,13a-decahydropyrido[1′,2′:4,5]pyrazino[1,2-a]pyrrolo[1,2-c]pyrimidines having HIV integrase inhibitory activity | Brian Alvin Johns, Takashi KAWASUJI, Teruhiko TAISHI | 2022-03-08 |
| 10927129 | N-[(2,4-difluorophenyl)methyl]-6-hydroxy-3-methyl-5,7-dioxo-2,3,5,7,11,11a-hexahydro[1,3] oxazolo[3,2-a]pyrido[1,2-d]pyrazine-8-carboxamide having HIV integrase inhibitory activity | Brian Alvin Johns, Takashi KAWASUJI, Teruhiko TAISHI | 2021-02-23 |
| 10202379 | Substituted polycyclic carbamoyl pyridone derivative prodrug | Chika Takahashi, Hidenori Mikamiyama, Toshiyuki Akiyama, Kenji Tomita, Makoto Kawai +2 more | 2019-02-12 |
| 9815835 | Substituted polycyclic carbamolypyridone derivative | Toshiyuki Akiyama, Kenji Takaya, Makoto Kawai, Minako Mikamiyama, Kenji Morimoto +3 more | 2017-11-14 |
| 9758515 | Substituted polycyclic carbamoyl pyridone derivative prodrug | Chika Takahashi, Hindenori Mikamiyama, Toshiyuki Akiyama, Kenji Tomita, Makoto Kawai +3 more | 2017-09-12 |
| 9527840 | Substituted-quinoxaline-type piperidine compounds and the uses thereof | Kouki Fuchino, R. Richard Goehring, Bin Shao, Naoki Tsuno, John William Frank Whitehead +1 more | 2016-12-27 |
| 9469638 | Substituted polycyclic carbamoylpyridone derivative | Toshiyuki Akiyama, Kenji Takaya, Makoto Kawai, Minako Mikamiyama, Kenji Morimoto +3 more | 2016-10-18 |
| 9365587 | Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates | Hiroshi Yoshida, Brian Alvin Johns, Takashi KAWASUJI, Daiki NAGAMATSU | 2016-06-14 |
| 9278967 | Substituted-quinoxaline-type piperidine compounds and the uses thereof | Kouki Fuchino, R. Richard Goehring, Akira Matsumura, Bin Shao, Naoki Tsuno +2 more | 2016-03-08 |
| 9273065 | Substituted pyrido[1',2':4,5]pyrazino[1,2-a]pyrimidines as HIV integrase inhibitors | Brian Alvin Johns, Takashi KAWASUJI, Teruhiko TAISHI | 2016-03-01 |
| 9051337 | Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-a]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides | Brian Alvin Johns, Takashi KAWASUJI, Teruhiko TAISHI | 2015-06-09 |
| 8987441 | Substituted polycyclic carbamoyl pyridone derivative prodrug | Chika Takahashi, Hidenori Mikamiyama, Toshiyuki Akiyama, Kenji Tomita, Makoto Kawai +3 more | 2015-03-24 |
| 8927710 | Substituted polycyclic carbamoylpyridone derivative | Toshiyuki Akiyama, Kenji Takaya, Makoto Kawai, Minako Mikamiyama, Kenji Morimoto +4 more | 2015-01-06 |
| 8846929 | Substituted-quinoxaline-type piperidine compounds and the uses thereof | Kouki Fuchino, R. Richard Goehring, Bin Shao, Naoki Tsuno, John William Frank Whitehead +1 more | 2014-09-30 |
| 8778943 | Substituted 10-hydroxy-9,11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1h-pyrido[1,2-α]pyrrolo[1′,2′:3,4]imidazo[1,2-d]pyrazine-8-carboxamides | Brian Alvin Johns, Takashi KAWASUJI, Teruhiko TAISHI | 2014-07-15 |
| 8754214 | Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates | Hiroshi Yoshida, Brian Alvin Johns, Takashi KAWASUJI, Daiki NAGAMATSU | 2014-06-17 |
| 8691823 | Prodrugs of (4aS, 13ar)-N-[(2,4-difluorophenyl)methyl]-10-hydroxy-9-11-dioxo-2,3,4a,5,9,11,13,13a-octahydro-1H-pyrido[1,2-a]pyrrolo[1′,2′:3:4]imidazo[1,2-d]pyrazine-8-carboxamide and their use in the treatment of HIV infection | Brian Alvin Johns, Jason Gordon Weatherhead, Yasunori Aoyama, Hiroshi Yoshida | 2014-04-08 |
| 8624023 | Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates | Hiroshi Yoshida, Brian Alvin Johns, Takashi KAWASUJI, Daiki NAGAMATSU | 2014-01-07 |
| 8575197 | Pyrolinone derivative and pharmaceutical composition comprising the same | Hiroyuki Kai, Takeshi Endoh, Kentaro Asahi, Hiroyuki Tobinaga | 2013-11-05 |