| 7781440 |
Use of substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives |
Thierry Gallet, Patrick Lardenois, Alistair Lochead, Severine Marguerie, Mourad Saady +2 more |
2010-08-24 |
$4,085,000 |
| 7585974 |
Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1]octane, their preparation and their therapeutic application |
Frederic Galli, Odile Leclerc, Alistair Lochead |
2009-09-08 |
$46,016,000 |
| 7566720 |
2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives |
Antonio Almario Garcia, Thierry Gallet, Adrien Tak Li, Alistair Lochead, Severine Marguerie +2 more |
2009-07-28 |
$44,543,000 |
| 7465737 |
Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl -6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives |
Alistair Lochead, Mourad Saady, Philippe Yaiche |
2008-12-16 |
$53,376,000 |
| 7462621 |
Use of substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a] pyrimidin-5(1H)one derivatives as therapeutic agents |
Thierry Gallet, Patrick Lardenois, Alistair Lochead, Severine Marguerie, Mourad Saady +2 more |
2008-12-09 |
$12,415,000 |
| 7388005 |
Substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo [1,2-a]pyrimidin-5(1H)one derivatives for neurodegenerative disorders |
Thierry Gallet, Patrick Lardenois, Alistair Lochead, Severine Marguerie, Mourad Saady +2 more |
2008-06-17 |
$12,588,000 |
| 7232827 |
Heteroaryl substituted 2-pyridinyl and 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one derivatives |
Alistair Lochead, Mourad Saady, Philippe Yaiche |
2007-06-19 |
$38,431,000 |
| 7223750 |
Derivatives of 5-(pyridin-3-yl)-1-azabicyclo[3.2.1]octane, the preparation thereof and the application of same in therapeutics |
Frederic Galli, Odile Leclerc, Alistair Lochead |
2007-05-29 |
$10,696,000 |
| 7214682 |
Substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo{1,2-a}pyrimidin-5(1h)one derivatives |
Thierry Gallet, Patrick Lardenois, Alistair Lochead, Severine Marguerie, Mourad Saady +2 more |
2007-05-08 |
$21,052,000 |
| 6987106 |
1,4-diazabicyclo[3.2.2]nonane-4-carboxylates and carboxamide derivates, production and use thereof in therapeutics |
Thierry Gallet, Samir Jegham, Patrick Lardenois, Alistair Lochead |
2006-01-17 |
$40,878,000 |
| 6974819 |
2-pyridinyl-6,7,8,9-tetrahydropyrimido{1,2-a}pyrimidin-4-one and 7-pyridinyl-2,3-dihydoimidazo{1,2-a}pyrimidin-5(1H)one derivatives |
Antonio Almario Garcia, Thierry Gallet, Adrien Tak Li, Alistair Lochead, Severine Marguerie +2 more |
2005-12-13 |
$37,308,000 |
| 6835730 |
4-heteroparyl-1,4-diazabicyclo[3.2.2]nonane, preparation and therapeutic use thereof |
Frederic Galli, Samir Jegham, Odile Leclerc, Alistair Lochead |
2004-12-28 |
$17,501,000 |
| 6635645 |
2,5,-diazabicyclo[2.2.1]heptane derivatives, their preparation and therapeutic uses |
Alistair Lochead, Samir Jegham, Jean Jeunesse, Frederic Galli, Luc Even |
2003-10-21 |
$954,000 |
| 6407095 |
1,4-diazabicylo[3,2,2]nonane derivatives, their preparation and their therapeutic application |
Alistair Lochead, Samir Jegham, Frederic Galli, Jean Jeunesse, Luc Even |
2002-06-18 |
|
| 6255319 |
5-aryl-3-(8-azabicyclo[3.2.1]oct-3-yl)-1,3,4-oxadiazol-2(3H)-one derivatives as 5-ht4 receptor ligands |
Samir Jegham, Alistair Lochead, Frederic Galli, Axelle Samson, Thierry Gallet |
2001-07-03 |
|
| 6057321 |
1,4-diazabicyclo [2.2.2] oct-2-ylmethyl derivatives, their preparation and therapeutic application |
Alistair Lochead, Samir Jegham, Axelle Solignac |
2000-05-02 |
|
| 5929089 |
5-phenyl-3-(piperidin-4-yl)-1,3,4-oxadiazol-2(3H)-one derivatives for use as 5-Ht4 or H3 receptor ligands |
Samir Jegham, Alistair Lochead, Frederic Galli, Axelle Solignac, Laurence De Cruz |
1999-07-27 |
|
| 5663173 |
N-[(1,4-diazabicyclo[2.2.2] oct-2-yl)methyl] benzamide derivatives, their preparations and their application in therapeutics |
Samir Jegham, Jean-Jacques Koenig, Alistair Lochead, Yves Guminski |
1997-09-02 |
|
| 4463004 |
Dioxazabicyclic derivatives |
Patrick G. Guerret, Bernard P. Bucher, Philippe L. Dostert, Gisele C. Mocquet |
1984-07-31 |
|