Issued Patents All Time
Showing 1–25 of 43 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12037328 | Compounds containing benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of G protein-coupled receptor 119 | Mikhail Chafeev, Mikhail Yudin, Yury Gezentsvey, Aleksandr Nikitin | 2024-07-16 |
| 10906894 | Compounds containing benzo[d][1,3]oxathiole, benzo[d][1,3]oxathiole 3-oxide or benzo[d][1,3]oxathiole 3,3-dioxide and methods/uses thereof as agonists of g protein-coupled receptor 119 | Mikhail Chafeev, Mikhail Yudin, Yury Gezentsvey, Aleksandr Nikitin | 2021-02-02 |
| 10844038 | 1,2-dithiolane compounds useful in neuroprotection, autoimmune and cancer diseases and conditions | Colleen E. Evans | 2020-11-24 |
| 10351540 | 1,2-dithiolane and dithiol compounds useful in treating mutant EGFR-mediated diseases and conditions | — | 2019-07-16 |
| 10246444 | 1,2-dithiolane and dithiol compounds useful in treating mutant EGFR-mediated diseases and conditions | — | 2019-04-02 |
| 10022381 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2018-07-17 |
| 9487535 | Asymmetric syntheses for spiro-oxindole compounds useful as therapeutic agents | Shaoyi Sun, Jianmin Fu, Sultan Chowdhury, Ivan William Hemeon, Michael Edward Grimwood | 2016-11-08 |
| 9174963 | Triazine compounds as PI3 kinase and MTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2015-11-03 |
| 8859542 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2014-10-14 |
| 8748421 | Triazine compounds as P13 kinase and MTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2014-06-10 |
| 8575159 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2013-11-05 |
| 8445486 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2013-05-21 |
| 8217036 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2012-07-10 |
| 8101590 | 9-aminocarbonylsubstituted derivatives of glycylcyclines | Phaik-Eng Sum, David Brian How, Darrin William Hopper, Matthew D. Vera, Joshua James Sabatini +1 more | 2012-01-24 |
| 8039469 | Triazine compounds as PI3 kinase and mTOR inhibitors | Aranapakam Mudumbai Venkatesan, Zecheng Chen, Christoph Martin Dehnhardt, Osvaldo Dos Santos, Efren Guillermo Delos Santos +8 more | 2011-10-18 |
| 7998965 | Glutamate aggrecanase inhibitors | Phaik-Eng Sum, Jerauld S. Skotnicki, Steve Yik-Kai Tam, David Brian How, Joshua James Sabatini +2 more | 2011-08-16 |
| 7812014 | Bicyclic 6-alkylidene-penems as β-lactamase inhibitors | Aranapakam Mudumbai Venkatesan, Takao Abe, Itsuki Yamamura, Tsuyoshi Takasaki, Atul Agarwal +3 more | 2010-10-12 |
| 7812008 | 9-substituted tetracyclines | Phaik-Eng Sum | 2010-10-12 |
| 7691842 | Tricyclic 6-alkylidene-penems as β-lactamase inhibitors | Aranapakam Mudumbai Venkatesan, Takao Abe, Ado Mihira, Atul Agarwal, Hideki Ushirogochi +3 more | 2010-04-06 |
| 7632838 | 11-beta HSD1 inhibitors | Jason Shaoyun Xiang, Eddine Saiah, Steve Y. Tam, John C. McKew, Lihren Chen +10 more | 2009-12-15 |
| 7553873 | Glutamate aggrecanase inhibitors | Phaik-Eng Sum, Jerauld S. Skotnicki, Steve Yik-Kai Tam, David Brian How, Joshua James Sabatini +2 more | 2009-06-30 |
| 7276611 | Process for synthesizing beta-lactamase inhibitor intermediates | Michael W. Winkley, Anita Wai-Yin Chan, Ivo L. Jirkovsky, Kenneth Alfred Martin Kremer, Joseph Zeldis +4 more | 2007-10-02 |
| 7229983 | 4-substituted or unsubstituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as β-lactamase inhibitors | Aranapakam Mudumbai Venkatesan | 2007-06-12 |
| 7112582 | Bicyclic 6-alkylidene-penems as β-lactamase inhibitors | Aranapakam Mudumbai Venkatesan, Takao Abe, Itsuki Yamamura, Tsuyoshi Takasaki, Atul Agarwal +3 more | 2006-09-26 |
| 7018997 | Tricyclic 6-alkylidene-penems as β-lactamase inhibitors | Aranapakam Mudumbai Venkatesan, Takao Abe, Ado Mihira, Atul Agarwal, Hideki Ushirogochi +3 more | 2006-03-28 |