Issued Patents All Time
Showing 1–25 of 53 patents
| Patent # | Title | Co-Inventors | Date |
|---|---|---|---|
| 12162849 | Synthesis of 3-methyl-1,2,4-thiadiazole-5-carbohydrazide or of the methyl-d3 deuterated form thereof | Guillaume Dutheuil | 2024-12-10 |
| 11731974 | N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists | Guillaume Dutheuil, Graeme L. Fraser | 2023-08-22 |
| 11478472 | NK-3 receptor antagonists for therapeutic treatment of leptin-related disease | Graeme L. Fraser | 2022-10-25 |
| 11078203 | Deuterated fezolinetant | — | 2021-08-03 |
| 11072582 | Substituted pyrrolidines as G-protein coupled receptor 43 agonists | Didier Schils, Ludivine Zoute, Julien Parcq | 2021-07-27 |
| 10941151 | Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof | Guillaume Dutheuil, Graeme L. Fraser, Marie-Odile Roy, Mohamed El Bousmaqui, Frederic Batt | 2021-03-09 |
| 10836768 | N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists | Guillaume Dutheuil, Graeme L. Fraser | 2020-11-17 |
| 10787458 | Chiral synthesis of N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-A]pyrazines | Guillaume Dutheuil | 2020-09-29 |
| 10781171 | Substituted pyrrolidines as G-protein coupled receptor 43 agonists | Didier Schils, Ludivine Zoute, Julien Parcq | 2020-09-22 |
| 10683295 | Chiral N-acyl-5,6,7(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-A]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof | Guillaume Dutheuil, Graeme L. Fraser, Marie-Odile Roy, Mohamed El Bousmaqui, Frederic Batt | 2020-06-16 |
| 10624890 | NK-3 receptor antagonists for therapeutic or cosmetic treatment of excess body fat | Graeme L. Fraser | 2020-04-21 |
| 10577318 | Substituted pyrrolidines as G-protein coupled receptor 43 agonists | Didier Schils, Ludivine Zoute, Julien Parcq | 2020-03-03 |
| 10544150 | NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders | Marie-Odile Roy, Graeme L. Fraser, Guillaume Dutheuil | 2020-01-28 |
| 10358416 | Substituted pyrrolidines as G-protein coupled receptor 43 agonists | Didier Schils, Ludivine Zoute, Julien Parcq | 2019-07-23 |
| 10258602 | Macrocyclic ghrelin receptor modulators and methods of using the same | Graeme L. Fraser, Kamel Benakli, Eric Marsault, Mark L. Peterson | 2019-04-16 |
| 10214533 | N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders | Guillaume Dutheuil, Graeme L. Fraser | 2019-02-26 |
| 10183948 | N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists | Guillaume Dutheuil, Graeme L. Fraser | 2019-01-22 |
| 10065960 | NK-3 receptor selective antagonist compounds, pharmaceutical composition and methods for use in NK-3 receptors mediated disorders | Marie-Odile Roy, Graeme L. Fraser, Guillaume Dutheuil | 2018-09-04 |
| 10065961 | Chiral N-acyl-5,6,7,(8-substituted)-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor mediated disorders and chiral synthesis thereof | Guillaume Dutheuil, Graeme L. Fraser, Marie-Odile Roy, Mohamed El Bousmaqui, Frederic Batt | 2018-09-04 |
| 10040751 | Intermediates for macrocyclic compounds | Eric Marsault, Kamel Benakli, Mark L. Peterson, Sylvie Beaubien, Luc Ouellet +2 more | 2018-08-07 |
| 10030025 | Substituted [1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists | Guillaume Dutheuil, Graeme L. Fraser | 2018-07-24 |
| 10017468 | Substituted pyrrolidines as G-protein coupled receptor 43 agonists | Didier Schils, Ludivine Zoute, Julien Parcq | 2018-07-10 |
| 9987274 | N-acyl-(3-substituted)-(8-substituted)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists | Guillaume Dutheuil, Graeme L. Fraser | 2018-06-05 |
| 9969745 | N-acyl-(3-substituted)-(8-methyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders | Guillaume Dutheuil, Graeme L. Fraser | 2018-05-15 |
| 9969738 | N-acyl-(3-substituted)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists, pharmaceutical composition, methods for use in NK-3 receptor-mediated disorders | Guillaume Dutheuil, Graeme L. Fraser | 2018-05-15 |