PO

Paolo Orsini

NS Nerviano Medical Sciences S.R.L.: 30 patents #1 of 140Top 1%
PS Pharmacia Italia S.P.A.: 3 patents #8 of 70Top 15%
PC Pharmacia & Upjohn Company: 3 patents #145 of 713Top 25%
PS Pharmacia & Upjohn S.P.A.: 3 patents #46 of 170Top 30%
Pfizer: 2 patents #2,078 of 5,153Top 45%
📍 Legnano, IT: #1 of 122 inventorsTop 1%
Overall (All Time): #82,449 of 4,157,543Top 2%
39
Patents All Time

Issued Patents All Time

Showing 1–25 of 39 patents

Patent #TitleCo-InventorsDate
11773064 4-carboxamido-isoindolinone derivatives as selective PARP-1 inhibitors Gianluca Mariano Enrico Papeo, Mikhail Yurievitch Krasavin, Alessandra Scolaro 2023-10-03
11420940 4-carboxamido-isoindolinone derivatives as selective parp-1 inhibitors Gianluca Mariano Enrico Papeo, Mikhail Yurievitch Krasavin, Alessandra Scolaro 2022-08-23
11047217 Safety valve 2021-06-29
10800739 4-carboxamido-isoindolinone derivatives as selective PARP-1 inhibitors Gianluca Mariano Enrico Papeo, Mikhail Yurievitch Krasavin, Alessandra Scolaro 2020-10-13
10556913 Asymmetric process for the preparation of thieno-indoles derivatives Italo Beria, Michele Caruso, Daniele Donati 2020-02-11
10385018 4-carboxamido-isoindolinone derivatives as selective PARP-1 inhibitors Gianluca Mariano Enrico Papeo, Mikhail Yurievitch Krasavin, Alessandra Scolaro 2019-08-20
10266547 Thieno[2,3-e]indole derivatives as new antitumor agents Marina Caldarelli, Michele Caruso 2019-04-23
10174048 Asymmetric process for the preparation of thieno-indoles derivatives Italo Beria, Michele Caruso, Daniele Donati 2019-01-08
10081622 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2018-09-25
10071074 Thieno-indole moieties and methods of treating using the same Italo Beria, Michele Caruso, Vittoria Lupi, Matteo Salsa, Achille Panzeri 2018-09-11
9649306 Treatment of diseases through administration of N-[5-(3,5-difluoro-benzyl)-1H-indazol-3-yl]-4-(4-methyl-piperazin-1-yl)-2-(tetrahydro-pyran-4-ylamino)-benzamide Natale Barbugian, Romualdo Forino, Tiziano Fumagalli 2017-05-16
9616059 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2017-04-11
9561290 Functionalized thieno-indole derivatives for the treatment of cancer Italo Beria, Michele Caruso, Vittoria Lupi, Matteo Salsa 2017-02-07
9527863 Thieno-indole moieties and methods of treating using the same Italo Beria, Michele Caruso, Vittoria Lupi, Matteo Salsa, Achille Panzeri 2016-12-27
9382235 Unsolvated crystalline form 1 of N-[5-(3, 5-difluoro-benzyl)-1H-indazol-3-yl]-4-(4-methyl-piperazin-1-yl)-2-(tetrahydro-pyran-4-ylamino)-benzamide and methods of use thereof Natale Barbugian, Romualdo Forino, Tiziano Fumagalli 2016-07-05
9255087 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2016-02-09
9102662 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2015-08-11
9085558 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2015-07-21
9085565 Process for the preparation of N-[5-(3,5-difluoro-benzyl)-1H-indazol-3-yl]-4-(4-methyl-piperazin-1-yl)-2-(tetrahydro-pyran-4-ylamino)-benzamide Natale Barbugian, Romualdo Forino, Tiziano Fumagalli 2015-07-21
9029356 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2015-05-12
8993594 Isoquinolin-1(2H)-one derivatives as PARP-1 inhibitors Gianluca Mariano Enrico Papeo, Jay Aaron Bertrand, Giovanni Cervi, Barbara Forte, Rosita Lupi +4 more 2015-03-31
8785448 Substituted pyrrolo-pyrazole derivatives as kinase inhibitors Maria Gabriella Brasca, Raffaella Amici, Daniele Fancelli, Marcella Nesi, Fabrizio Orzi +3 more 2014-07-22
8765972 3-oxo-2,3-dihydro-1H-isoindole-4-carboxamides with selective PARP-1 inhibition Gianluca Mariano Enrico Papeo, Alina Anatolievna Busel, Elena Casale, Alexander Khvat, Mikhail Yurievitch Krasavin +2 more 2014-07-01
8673893 Substituted indazole derivatives active as kinase inhibitors Andrea Lombardi Borgia, Maria Menichincheri, Achille Panzeri, Ettore Perrone, Ermes Vanotti +2 more 2014-03-18
8592416 Isoquinolin-1 (2H)-one derivatives as PARP-1 inhibitors Gianluca Mariano Enrico Papeo, Jay Aaron Bertrand, Giovanni Cervi, Barbara Forte, Rosita Lupi +4 more 2013-11-26