MR

Michael Rowley

Merck: 22 patents #425 of 9,382Top 5%
Overall (All Time): #108,753 of 4,157,543Top 3%
33
Patents All Time

Issued Patents All Time

Showing 25 most recent of 33 patents

Patent #TitleCo-InventorsDate
8314062 Macrocyclic compounds as antiviral agents Benedetta Crescenzi, Monica Donghi, Marco Ferrara, Cristina Gardelli, Steven Harper +2 more 2012-11-20
7968553 Tetrahydro-4H-pyrido[1,2-a] pyrimidines useful as HIV integrase inhibitors Benedetta Crescenzi, Olaf Kinzel, Ester Muraglia, Federica Orvieto, Giovanna Pescatore +1 more 2011-06-28
7863294 Heterocycle derivatives as histone deacetylase (HDAC) inhibitors Barbara Attenni, Federica Ferrigno, Philip Jones, Raffaele Ingenito, Olaf Kinzel +5 more 2011-01-04
7820660 N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase Benedetta Crescenzi, Cristina Gardelli, Ester Muraglia, Emanuela Nizi, Federica Orvieto +6 more 2010-10-26
7795247 Tetracyclic indole derivatives as antiviral agents Immacolata Conte, Caterina Ercolani, Frank Narjes, Marco Pompei, Ian Stansfield 2010-09-14
7781431 Thienopyrroles as antiviral agents Barbara Attenni, Jose Ignacio Martin Hernando, Savina Malancona, Frank Narjes, Jesus Maria Ontoria Ontoria 2010-08-24
7662809 Tetracyclic indole derivatives as antiviral agents Caterina Ercolani, Joerg Habermann, Frank Narjes, Simona Ponzi, Ian Stansfield 2010-02-16
7435734 N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase Benedetta Crescenzi, Cristina Gardelli, Ester Muraglia, Emanuela Nizi, Federica Orvieto +6 more 2008-10-14
7414045 Substituted pyrimido[1,2-a]azepines useful as HIV integrase inhibitors Benedetta Crescenzi, Olaf Kinzel, Ester Muraglia, Federica Orvieto, Giovanna Pescatore +1 more 2008-08-19
7217713 N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase Benedetta Crescenzi, Cristina Gardelli, Ester Muraglia, Emanuela Nizi, Federica Orvieto +6 more 2007-05-15
7169780 N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase Benedetta Crescenzi, Cristina Gardelli, Ester Muraglia, Federica Orvieto, Paola Pace +6 more 2007-01-30
6872731 Imidazo-pyridine derivatives as ligands for GABA receptors James Michael Crawforth, Simon Charles Goodacre, Timothy Harrison, David Hallett, Andrew Pate Owens +1 more 2005-03-29
6723735 Imidazo-pyridine derivatives as ligands for GABA receptors David Hallett 2004-04-20
6608062 Imidazo-triazine derivatives as ligands for GABA receptors William R. Carling, Alexander Richard Guiblin, Kevin W. Moore, Christopher Moyes, Leslie Joseph Street 2003-08-19
6486153 Phenylindole derivatives as 5-HT2A receptor ligands Jose Luis Castro Pineiro, Steven M. Hutchins, Stephen Lewis, Adrian L. Smith, Graeme Irvine Stevenson 2002-11-26
6479480 Phenylindole derivatives as 5-ht2a receptor ligands Christopher Moyes 2002-11-12
6352994 Substituted 1H-pyridinyl-2-ones as GABAA alpha 2/3 ligands Ian Collins, Stephen Robert Fletcher, Timothy Harrison, Paul D. Leeson, Christopher Moyes +3 more 2002-03-05
6337331 Triazolo-pyrimidine as ligands for GABA receptors Howard Barff Broughton, Jose Luis Castro Pineiro, Ian Collins, Karl Richard Gibson, Leslie Joseph Street 2002-01-08
6316468 Phenylindole derivatives as 5-HT2A receptor antagonists Robert Maxey, Monique Bodil Van Niel 2001-11-13
6200982 Substituted 1H-pyridinyl-2-ones as GABAA-.alpha. 2/3 ligands Ian Collins, Stephen Robert Fletcher, Timothy Harrison, Paul D. Leeson, Christopher Moyes +3 more 2001-03-13
6080745 Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands William Barnaby Davey, Paul D. Leeson 2000-06-27
6054456 Substituted piperazine derivatives Tamara Ladduwahetty, Angus Murray MacLeod 2000-04-25
6048878 Substituted piperidine derivatives as selective agonists of 5-HT receptors Jose Luis Castro Pineiro, Ian Collins, Angus Murray MacLeod, Christopher Moyes, Graham Andrew Showell 2000-04-11
5977116 Piperazine, piperidine and tetrahydropyridine derivatives Jose Luis Castro Pineiro, Angus Murray MacLeod, Monique Bodil Van Niel 1999-11-02
5763448 Pyrmidine derivatives William R. Carling, Ian Collins, Paul D. Leeson 1998-06-09