JA

Jose Alexander

Merck: 22 patents #425 of 9,382Top 5%
Overall (All Time): #186,914 of 4,157,543Top 5%
23
Patents All Time

Issued Patents All Time

Patent #TitleCo-InventorsDate
5733907 Prodrugs of an inhibitor of HIV protease Dilbir S. Bindra, Bruce D. Dorsey, Arnold J. Repta, Joseph P. Vacca 1998-03-31
5684018 Acyloxyisopropyl carbamates as prodrugs for amine drugs 1997-11-04
5466811 Dioxolenylmethyl carbamates pro moieties for amine drugs 1995-11-14
5066648 Pyroglutamic acid esters used as dermal penetration enhancers for drugs Takeru Higuchi 1991-11-19
4973579 Enhancment of absorption of drugs from gastrointestinal tract using choline ester salts Joseph A. Fix 1990-11-27
4970206 Pyroglutamic acid esters used as dermal penetration enhancers for drugs Takeru Higuchi 1990-11-13
4963525 Acylcarnitines as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal compartments Joseph A. Fix, A. J. Repta 1990-10-16
4963556 Choline esters as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal cavities Joseph A. Fix, A. J. Repta 1990-10-16
4916230 Process for preparing novel N-(acyloxy-alkoxy)carbonyl derivatives useful as bioreversible prodrug moieties for primary and secondary amine functions in drugs 1990-04-10
4847250 Pyroglutamic acid esters used as dermal penetration enhancers for drugs Takeru Higuchi 1989-07-11
4847298 Acylcarnitines as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal compartments Joseph A. Fix, A. J. Repta 1989-07-11
4835138 Choline esters as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal cavities A. J. Repta, Joseph A. Fix 1989-05-30
4822773 Enhancement of absorption of drugs from gastrointestinal tract using choline ester salts Joseph A. Fix 1989-04-18
4762851 Pyroglutamic acid esters used as dermal penetration enhancers for drugs Takeru Higuchi 1988-08-09
4760057 (Acyloxyalkoxy)carbonyl derivatives as bioreversible prodrug moieties for primary and secondary amine functions in drugs 1988-07-26
4731360 Acylcarnitines as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal compartments A. J. Repta, Joseph A. Fix 1988-03-15
4729989 Enhancement of absorption of drugs from gastrointestinal tract using choline ester salts Joseph A. Fix 1988-03-08
4692441 Chorine esters as absorption-enhancing agents for drug delivery through mucous membranes of the nasal, buccal, sublingual and vaginal cavities A. J. Repta, Joseph A. Fix 1987-09-08
4537772 Enhancing absorption of drugs from gastrointestinal tract using acylcarnitines Joseph A. Fix 1985-08-27
4495180 Prodrugs of Ara-A an antiviral agent 1985-01-22
4426391 [(Alkoxycarbonyl)oxy]alkyl esters of methyldopa Chung Shih 1984-01-17
4425337 Adjuvants for rectal delivery of drug Joseph A. Fix 1984-01-10
4244880 Anthracycline synthesis Lester A. Mitscher 1981-01-13