| 11453673 |
Substituted [1,2,4]triazolo[4,3-a]pyrazines as phosphodiesterase inhibitors |
Nicholas Paul Camp, Chafiq Hamdouchi, Jayana Pankaj Lineswala, John Richard Morphy |
2022-09-27 |
$750,369,000 |
| 11401274 |
[1,2,4]Triazolo derivatives as PDE1 inhibitors for the treatment of diabetes |
Michael James Genin, William Glen Holloway, Cynthia Darshini Jesudason |
2022-08-02 |
$1,780,908,000 |
| 11180503 |
[1,2,4]Triazolo[4,3-A]pyrazin-6(5H)-one derivatives |
Michael James Genin, William Glen Holloway, Richard Duane Johnston, John Richard Morphy |
2021-11-23 |
$939,663,000 |
| 10435415 |
Substituted tetrahydrocarbazole and carbazole carboxamide compounds |
Douglas G. Batt, Myra Beaudoin Bertrand, George V. De Lucca, Michael Galella, Soo S. Ko +5 more |
2019-10-08 |
|
| 10214537 |
Bicyclic heteroaryl amine compounds |
Rajeev S. Bhide, Douglas G. Batt, Robert J. Cherney, Lyndon A. M. Cornelius, Qingjie Liu +8 more |
2019-02-26 |
|
| 10138244 |
Triazolopyrazinone derivative useful as a human PDE1 inhibitor |
Mark David Rekhter |
2018-11-27 |
$565,573,000 |
| 10106559 |
Substituted tetrahydrocarbazole and carbazole carboxamide compounds |
Douglas G. Batt, Myra Beaudoin Bertrand, George V. DeLucca, Michael Galella, Soo S. Ko +5 more |
2018-10-23 |
|
| 10023576 |
Heteroaryl substituted pyrrolotriazine amine compounds as PI3K inhibitors |
Rajeev S. Bhide, Zheming Ruan, Robert J. Cherney, Lyndon A. M. Cornelius, T. G. Murali Dhar +5 more |
2018-07-17 |
|
| 9815859 |
Tricyclic sulfones as RORγ modulators |
Jingwu Duan, T. G. Murali Dhar, David Marcoux, Douglas G. Batt, Qingjie Liu +5 more |
2017-11-14 |
|
| 9637495 |
CGRP receptor antagonists |
David Coates, Kevin Charles FORTNER, Richard Duane Johnston, Steven Marc Massey, Jason K. Myers +1 more |
2017-05-02 |
$234,079,000 |
| 9334290 |
Substituted tetrahydrocarbazole and carbazole carboxamide compounds |
Douglas G. Batt, Myra Beaudoin Bertrand, George V. DeLucca, Michael Galella, Soo S. Ko +5 more |
2016-05-10 |
|
| 8586751 |
Nicotinamide compounds useful as kinase modulators |
George V. De Lucca, Chunjian Liu, Jingwu Duan, Andrew J. Tebben |
2013-11-19 |
$194,958,000 |
| 8362065 |
Carbazole carboxamide compounds useful as kinase inhibitors |
Qingjie Liu, Douglas G. Batt, George V. DeLucca, Andrew J. Tebben |
2013-01-29 |
$45,866,000 |
| 8299061 |
Inhibitors of diacylglycerol acyltransferase |
Macklin Brian Arnold, Thomas Beauchamp, Emily J. Canada, Erik James Hembre, Jianliang Lu +2 more |
2012-10-30 |
|
| 8133907 |
Pyridine derivatives as dipeptedyl peptidase inhibitors |
Larry C. Blaszczak, Brian Michael Mathes, Shon Pulley, Michael Alan Robertson, Scott Martin Sheehan +2 more |
2012-03-13 |
$193,239,000 |
| 8106090 |
1-amino linked compounds |
Larry C. Blaszczak, Shon Pulley, Michael Alan Robertson, Scott Martin Sheehan, Michael Robert Wiley |
2012-01-31 |
$97,135,000 |
| 8084620 |
Carbazole carboxamide compounds useful as kinase inhibitors |
Qingjie Liu, Douglas G. Batt, George V. DeLucca, Andrew J. Tebben |
2011-12-27 |
$134,492,000 |
| 8076514 |
Phenyl compounds and their use in the treatment of Type II diabetes |
Larry C. Blaszczak, Shon Pulley, Michael Alan Robertson, Scott Martin Sheehan, Brian Morgan Watson +1 more |
2011-12-13 |
$77,945,000 |
| 7291619 |
Melanocortin receptor agonists |
Christopher Kelly Biggers, Karin Briner, Christopher William Doecke, Matthew Joseph Fisher, Larry W. Hertel +8 more |
2007-11-06 |
$65,050,000 |
| 7186715 |
Piperazine- and piperidine-derivatives as melanocortin receptor agonists |
Karin Briner, Christopher William Doecke, Vincent Mancuso, Michael John Martinelli, Timothy Ivo Richardson +2 more |
2007-03-06 |
$170,937,000 |
| 6906056 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds |
Richard Thompson, Stephen Wilkie, Douglas Richard Stack, Eldon Vanmeter, Thomas C. Britton +9 more |
2005-06-14 |
$111,693,000 |
| 6838455 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
James E. Audia, Warren J. Porter, Richard Thompson, Stephen Wilkie, Douglas Richard Stack |
2005-01-04 |
$316,880,000 |
| 6696438 |
Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting &bgr;-amyloid peptide release and/or its synthesis by use of such compounds |
James E. Audia, Bruce A. Dressman |
2004-02-24 |
$236,890,000 |
| 6569851 |
Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting &bgr;-amyloid peptide release and/or its synthesis by use of such compounds |
Richard Thompson, Stephen Wilkie, Douglas Richard Stack, Eldon Vanmeter, Thomas C. Britton +9 more |
2003-05-27 |
$145,984,000 |
| 6552013 |
Deoxyamino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting &bgr;-amyloid peptide release and/or its synthesis by use of such compounds |
James E. Audia, Warren J. Porter, Richard Thompson, Stephen Wilkie, Douglas Richard Stack |
2003-04-22 |
$103,002,000 |
