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1H-indazole carboxamides as receptor-interacting protein kinase 1 inhibitors (RIPK1) |
Junqing Guo, Jie Chen, Carolyn Diane Dzierba, Amy C. Hart, John E. Macor +2 more |
2024-12-24 |
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Aminotriazolopyridines as kinase inhibitors |
Junqing Guo, Amy C. Hart, John E. Macor, Michael E. Mertzman, William J. Pitts +7 more |
2024-12-03 |
| 12110290 |
Triazolopyridinyl compounds as kinase inhibitors |
Jie Chen, Carolyn Diane Dzierba, David B. Frennesson, Junqing Guo, Amy C. Hart +9 more |
2024-10-08 |
| 12065437 |
Biaryl kinase inhibitors |
Carolyn Diane Dzierba, John E. Macor |
2024-08-20 |
| 11767322 |
Triazolopyridinyl compounds as kinase inhibitors |
Jie Chen, Carolyn Diane Dzierba, David B. Frennesson, Junqing Guo, Amy C. Hart +9 more |
2023-09-26 |
| 11618753 |
Aminopyrrolotriazines as kinase inhibitors |
Scott Hunter Watterson, Murugaiah Andappan Murugaiah Subbaiah, Carolyn Diane Dzierba, Hua Gong, Jason M. Guernon +11 more |
2023-04-04 |
| 11440913 |
Aminoimidazopyridazines as kinase inhibitors |
Michael E. Mertzman, Carolyn Diane Dzierba, Jason M. Guernon, Amy C. Hart, John E. Macor +3 more |
2022-09-13 |
| 11053258 |
Pyrimidine carboxamides as GSK-3 inhibitors |
Prasanna Sivaprakasam, Gene M. Dubowchik, John E. Macor |
2021-07-06 |
| 10981910 |
Biaryl kinase inhibitors |
Carolyn Diane Dzierba, John E. Macor |
2021-04-20 |
| 10913738 |
Aminotriazolopyridines as kinase inhibitors |
Junqing Guo, Amy C. Hart, John E. Macor, Michael E. Mertzman, William J. Pitts +7 more |
2021-02-09 |
| 10752609 |
GSK-3 inhibitors |
Richard A. Hartz, Vijay T. Ahuja, Ling Chen, Prasanna Sivaprakasam, Gene M. Dubowchik +2 more |
2020-08-25 |
| 10723734 |
Biaryl kinase inhibitors |
Carolyn Diane Dzierba, John E. Macor |
2020-07-28 |
| 10550080 |
Acyl sulfonamide NaV1.7 inhibitors |
Ling Chen |
2020-02-04 |
| 10544120 |
Biaryl kinase inhibitors |
Joanne J. Bronson, Ling Chen, Jonathan L. Ditta, Carolyn Diane Dzierba, Prasada Rao Jalagam +6 more |
2020-01-28 |
| 10351563 |
Biaryl kinase inhibitors |
— |
2019-07-16 |
| 10246469 |
Biaryl kinase inhibitors |
Joanne J. Bronson, Ling Chen, Jonathan L. Ditta, Carolyn Diane Dzierba, Prasada Rao Jalagam +6 more |
2019-04-02 |
| 10155760 |
Biaryl kinase inhibitors |
Carolyn Diane Dzierba, John E. Macor |
2018-12-18 |
| 9902722 |
Biaryl kinase inhibitors |
Ling Chen, Carolyn Diane Dzierba, Jonathan L. Ditta, John E. Macor, Joanne J. Bronson |
2018-02-27 |
| 9809573 |
Substituted pyridine derivatives useful as GSK-3 inhibitors |
Ling Chen, Gene M. Dubowchik, Swanee E. Jacutin-Porte, Prasanna Sivaprakasam, John E. Macor |
2017-11-07 |
| 9718804 |
GSK-3 inhibitors |
Ling Chen, Gene M. Dubowchik, Swanee E. Jacutin-Porte, Vivekananda M. Vrudhula, Senliang Pan +2 more |
2017-08-01 |
| 8748429 |
CGRP receptor antagonists |
Gene M. Dubowchik, John E. Macor, Ling Chen |
2014-06-10 |
| 8314117 |
CGRP receptor antagonists |
Gene M. Dubowchik, John E. Macor |
2012-11-20 |
| 8143403 |
CGRP receptor antagonists |
David K. Leahy, Yu Fan, Lopa V. Desai, Ronald L. Hanson, Thorsten Rosner |
2012-03-27 |
| 8044043 |
CGRP receptor antagonists |
— |
2011-10-25 |
| 7842808 |
Anti-migraine spirocycles |
Prasad V. Chaturvedula, Ling Chen, Rita Civiello, Andrew P. Degnan, Gene M. Dubowchik +5 more |
2010-11-30 |