HE

Harald Engelhardt

BO BOE: 24 patents #785 of 12,373Top 7%
Overall (All Time): #170,617 of 4,157,543Top 5%
24
Patents All Time

Issued Patents All Time

Patent #TitleCo-InventorsDate
12064421 Substituted 1H-pyrazolo[4,3-c]pyridines and derivatives as EGFR inhibitors Mark PETRONCZKI, Juergen Ramharter, Ulrich Reiser, Heinz Stadtmueller, Dirk Scharn +1 more 2024-08-20
11608343 Substituted pyrimido[5,4-d]pyrimidines as HER2 inhibitors Birgit WILDING, Dietrich BOESE, Julian FUCHS, Ralph NEUMUELLER, Mark PETRONCZKI +2 more 2023-03-21
11261184 [1,6]naphthyridine compounds and derivatives as CDK8/CDK19 inhibitors Heribert Arnhof, Sebastian CAROTTA, Marco Hofmann, Marc Kerenyi, Dirk Scharn 2022-03-01
11213520 Phenylpyrazolylacetamide compounds and derivatives as CDK8/CDK19 inhibitors Heribert Arnhof, Sebastian CAROTTA, Marco Hofmann, Marc Kerenyi, Dirk Scharn 2022-01-04
11174245 Benzimidazole compounds and derivatives as EGFR inhibitors Dietrich BOESE, Georg Dahmann, Mark PETRONCZKI, Dirk Scharn 2021-11-16
11077107 Triazolopyrazine Davide Gianni, Christian Alan Paul Smethurst 2021-08-03
10328074 Substituted [1,2,4]triazolo[4,3-a]pyrazines as BRD4 inhibitors Davide Gianni, Christian Alan Paul Smethurst 2019-06-25
9428513 Triazolopyrazine 2016-08-30
9428515 Benzimidazole derivatives 2016-08-30
9422290 Triazolopyridazine Davide Gianni, Dirk Kessler, Ulrich Reiser, Christian Alan Paul Smethurst, Andreas Steffen 2016-08-23
9296748 Pyridinones Laetitia Janine MARTIN, Christian Alan Paul Smethurst 2016-03-29
9266891 Substituted [1,2,4]triazolo[4,3-A]pyrazines that are BRD4 inhibitors Davide Gianni, Christian Alan Paul Smethurst 2016-02-23
9199988 Dihydroquinazolinone analogues Christian Alan Paul Smethurst, Davide Gianni, Ulrich Reiser 2015-12-01
9102684 Indolinone analogues Davide Gianni, Andreas Mantoulidis, Christian Alan Paul Smethurst 2015-08-11
8895581 1H-imidazo[4,5-c]quinolines Darryl McConnell, Christiane Kofink 2014-11-25
8637549 Pyridons as PDK1 inhibitors Guido Boehmelt, Christiane Kofink, Daniel Kuhn, Darryl McConnell, Heinz Stadtmueller 2014-01-28
8575203 Chemical compounds Christiane Kofink, Darryl McConnell 2013-11-05
8404674 Substituted 9H-purin-2-YL compounds, compositions thereof and uses thereof Heinz Stadtmueller, Guido Boehmelt, Ulrich Hirt, Otmar Schaaf, Irene Waizenegger 2013-03-26
8258129 4-heterocycloalkylpyri(mi)dines, process for the preparation thereof and their use as medicaments Gerd Bader, Guido Boehmelt, Ralph Brueckner, Thomas Gerstberger, Maria Impagnatiello +5 more 2012-09-04
8207179 Substituted indolines as tyrosine kinase inhibitors Bodo Betzemeier, Guido Boehmelt, Ulrich Guertler, Thomas Karner, Oliver Kraemer +9 more 2012-06-26
7569561 2,4-diaminopyrimidines useful for treating cell proliferation diseases Heinz Stadtmueller, Anke Baum, Guido Boehmelt, Jens Juergen Quant, Flavio Solca +2 more 2009-08-04
7521457 Pyrimidines as PLK inhibitors Heinz Stadtmueller, Martin Steegmaier, Anke Baum, Ulrich Guertler, Andreas Schoop +6 more 2009-04-21
7371753 Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions Heinz Stadtmueller, Andreas Schoop, Martin Steegmaier, Matthias Hoffmann, Matthias Grauert 2008-05-13
7241769 Pyrimidines as PLK inhibitors Heinz Stadtmueller, Ulrich Reiser, Stephan Karl Zahn, Rudolf Hauptmann, Martin Steegmaier +3 more 2007-07-10