MG

Markus Gude

AP Actelion Pharmaceuticals: 20 patents #13 of 188Top 7%
IP Idorsia Pharmaceuticals: 7 patents #11 of 104Top 15%
PS Pharmacia & Upjohn S.P.A.: 1 patents #98 of 170Top 60%
Overall (All Time): #138,016 of 4,157,543Top 4%
28
Patents All Time

Issued Patents All Time

Showing 25 most recent of 28 patents

Patent #TitleCo-InventorsDate
11040966 Benzimidazole-proline derivatives Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Jodi T. Williams 2021-06-22
10329287 Benzimidazole-proline derivatives Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Jodi T. Williams 2019-06-25
10023560 Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Markus Von Raumer +1 more 2018-07-17
9914721 Use of benzimidazole-proline derivatives Christoph Boss, Catherine Roch, Christine Brotschi, Bibia Heidmann, François Jenck +3 more 2018-03-13
9914720 Crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[D]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone and its use as orexin receptor antagonists Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Markus Von Raumer +1 more 2018-03-13
9790208 Crystalline salt form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Markus Von Raumer +1 more 2017-10-17
9732075 Benzimidazole-proline derivatives Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen, Jodi T. Williams 2017-08-15
9493446 Orexin receptor antagonists which are [ortho bi-(hetero-)aryl]-[2-(meta bi-(hetero-)aryl)-pyrrolidin-1-yl]-methanone derivatives Martin Bolli, Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen +1 more 2016-11-15
9428456 1-[m-carboxamido(hetero)aryl-methyl]-heterocyclyl-carboxamide derivatives Heinz Fretz, Philippe Guerry, Thierry Kimmerlin, Francois Lehembre, Thomas Pfeifer +1 more 2016-08-30
9303023 Pyrazole and imidazole derivatives useful as orexin antagonists Martin Bolli, Christoph Boss, Christine Brotschi, Bibia Heidmann, Thierry Sifferlen +1 more 2016-04-05
9211279 Proline sulfonamide derivatives as orexin receptor antagonists Christoph Boss, Christine Brotschi, John Gatfield, Bibia Heidmann, Thierry Sifferlen +1 more 2015-12-15
9000029 Proline sulfonamide derivatives as orexin receptor antagonists Christoph Boss, Christine Brotschi, John Gatfield, Bibia Heidmann, Thierry Sifferlen +1 more 2015-04-07
8895606 Proline sulfonamide derivatives as orexin receptor antagonists Christoph Boss, Christine Brotschi, John Gatfield, Bibia Heidmann, Thierry Sifferlen +1 more 2014-11-25
8889676 3-ureidoisoquinolin-8-yl derivatives Christian Hubschwerlen, Philippe Panchaud 2014-11-18
8329706 Oxazolidinone derivatives Hamed Aissaoui, Christoph Boss, Christine Brotschi, Romain Siegrist, Thierry Sifferlen +1 more 2012-12-11
8288435 2-aza-bicyclo[3.1.0]hexane derivatives as orexin receptor antagonists Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen, Daniel TRACHSEL 2012-10-16
8288429 2-aza-bicyclo[3.3.0]octane derivatives Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen, Daniel TRACHSEL 2012-10-16
8273740 2-sulfanyl-benzoimidazol-1-yi-acetic acid derivatives as CRTH2 antagonists Heinz Fretz, Kurt Hilpert, Julien Pothier, Markus Riederer, Matthias Steger 2012-09-25
8236964 Thiazolidine derivatives as orexin receptor antagonists Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen 2012-08-07
8188082 5,6,7,8-tetrahydro-imidazo[1,5-α]pyrazine derivatives Hamed Aissaoui, Christoph Boss, Raif Koberstein, Thierry Sifferien 2012-05-29
8133901 3-heteroaryl (amino or amido)-1-(biphenyl or phenylthiazolyl) carbonylpiperidine derivatives as orexin receptor inhibitors Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen 2012-03-13
8114867 Oxazolidinone antibiotic derivatives Christian Hubschwerlen, Georg Rueedi, Jean-Philippe Surivet, Cornelia Zumbrunn-Acklin 2012-02-14
8106215 3-aza-bicyclo[3.3.0]octane compounds Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen 2012-01-31
8063099 Trans-3-aza-bicyclo[3.1.0]hexane derivatives Hamed Aissaoui, Christoph Boss, Ralf Koberstein, David Lehman, Thierry Sifferlen +1 more 2011-11-22
8003654 N-glycinsulfonamide derivatives and uses as orexin receptor antagonists Hamed Aissaoui, Christoph Boss, Ralf Koberstein, Thierry Sifferlen, Cornelia Zumbrunn Acklin 2011-08-23