| 9862704 |
Oxindole derivatives carrying an amine-substituted piperidyl-acetidinyl substituent and use thereof for treating vasopressine-related diseases |
Hervé Geneste, Wilfried Hornberger, Charles W. Hutchins, Katja Jantos, Loic Laplanche +1 more |
2018-01-09 |
$640,201,000 |
| 9840495 |
Oxindole derivatives carrying a piperidyl-substituted azetidinyl substituent and use thereof for treating vasopressine-related diseases |
Hervé Geneste, Wilfried Hornberger, Charles W. Hutchins, Katja Jantos, Loic Laplanche +1 more |
2017-12-12 |
$208,732,000 |
| 9688678 |
Oxindole compounds carrying a nitrogen-bound spiro substituent and use thereof for treating vasopressin-related diseases |
Hervé Geneste, Wilfried Hornberger, Katja Jantos, Marcel van Gaalen |
2017-06-27 |
$159,595,000 |
| 9657002 |
Oxindole derivatives carrying an oxetane substituent and use thereof for treating vassopressin-related diseases |
Katja Jantos, Wilfred Braje, Hervé Geneste, Liliane Unger, Berthold Behl +4 more |
2017-05-23 |
$153,003,000 |
| 9617226 |
Fused heterocyclic or carbocyclic compounds carrying a substituted cycloaliphatic radical and use thereof for treating vasopressin-related diseases |
Wilfried Braje, Jayne Froggett, Hervé Geneste, Wilfried Hornberger, Katja Jantos +1 more |
2017-04-11 |
$236,573,000 |
| 9567325 |
Carboxamide compounds and their use as calpain inhibitors |
Helmut Mack, Katja Jantos, Achim Moeller, Wilfried Hornberger, Charles W. Hutchins |
2017-02-14 |
$158,590,000 |
| 9527811 |
Carboxamide compounds and their use as calpain inhibitors |
Helmut Mack, Katja Jantos, Achim Moeller, Wilfried Hornberger, Charles W. Hutchins |
2016-12-27 |
$303,958,000 |
| 9527856 |
Oxindole compounds carrying a CO-bound spiro substituent and use thereof for treating vasopressin-related diseases |
Wilfried Braje, Hervé Geneste, Wilfried Hornberger, Katja Jantos, Claudia Krack +1 more |
2016-12-27 |
$303,958,000 |
| 9475782 |
Guanidine compounds, and use thereof as binding partners for 5-HT5 receptors |
Astrid Netz, Wilhelm Amberg, Udo Lange, Michael Ochse, Charles W. Hutchins +2 more |
2016-10-25 |
$312,321,000 |
| 9296697 |
Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors |
Wilhelm Amberg, Astrid Netz, Michael Ochse, Udo Lange, Charles W. Hutchins +3 more |
2016-03-29 |
$35,821,000 |
| 9273036 |
Oxindole derivatives carrying an oxetane substituent and use thereof for treating vasopressine-related diseases |
Katja Jantos, Wilfred Braje, Hervé Geneste, Liliane Unger, Berthold Behl +4 more |
2016-03-01 |
$121,077,000 |
| 9150553 |
Carboxamide compounds and their use as calpain inhibitors |
Wilfried Hornberger, Helmut Mack, Achim Moeller, Barbara Vogg, Jürgen Delzer +2 more |
2015-10-06 |
$91,920,000 |
| 9150545 |
Carboxamide compounds and their use as calpain inhibitors V |
Katja Jantos, Helmut Mack, Achim Möller, Wilfried Hornberger, Gisela Backfisch +2 more |
2015-10-06 |
$91,920,000 |
| 9139557 |
Carboxamide compounds and their use as calpain inhibitors |
Wilfried Hornberger, Helmut Mack, Achim Moeller, Volker Nimmrich, Dietmar Seemann +1 more |
2015-09-22 |
$160,450,000 |
| 9096619 |
Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy |
Wilhelm Amberg, Michael Ochse, Udo Lange, Berthold Behl, Wilfried Hornberger +2 more |
2015-08-04 |
$112,867,000 |
| 9067871 |
Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy |
Wilhelm Amberg, Michael Ochse, Udo Lange, Berthold Behl, Wilfried Hornberger +2 more |
2015-06-30 |
$93,334,000 |
| 9062027 |
Carboxamide compounds and their use as calpain inhibitors V |
Katja Jantos, Helmut Mack, Achim Möller, Wilfried Hornberger, Yanbin Lao +2 more |
2015-06-23 |
$83,346,000 |
| 9051304 |
Carboxamide compounds and their use as calpain inhibitors V |
Katja Jantos, Helmut Mack, Achim Möller, Wilfried Hornberger, Gisela Backfisch +2 more |
2015-06-09 |
$60,924,000 |
| 9018206 |
Carboxamide compounds and their use as calpain inhibitors |
Helmut Mack, Katja Jantos, Achim Moeller, Wilfried Hornberger, Charles W. Hutchins |
2015-04-28 |
$111,300,000 |
| 8921406 |
5-ring heteroaromatic compounds and their use as binding partners for 5-HT5 receptors |
Wilhelm Amberg, Astrid Netz, Michael Ochse, Udo Lange, Andreas Haupt +2 more |
2014-12-30 |
$164,094,000 |
| 8906941 |
Carboxamide compounds and their use as calpain inhibitors |
Helmut Mack, Katja Jantos, Achim Moeller, Wilfried Hornberger, Charles W. Hutchins |
2014-12-09 |
$81,481,000 |
| 8686002 |
Heterocyclic compounds and their use as binding partners for 5-HT5 receptors |
Wilhelm Amberg, Astrid Netz, Michael Ochse, Udo Lange, Charles W. Hutchins +2 more |
2014-04-01 |
$86,782,000 |
| 8598211 |
Carboxamide compounds and their use as calpain inhibitors IV |
Katja Jantos, Helmut Mack, Achim Möller, Wilfried Hornberger, Gisela Backfisch +2 more |
2013-12-03 |
$87,921,000 |
| 8563617 |
Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy |
Wilhelm Amberg, Michael Ochse, Udo Lange, Berthold Behl, Wilfried Homberger +2 more |
2013-10-22 |
|
| 8481576 |
Guanidine compounds, and use thereof as binding partners for 5-HT5 receptors |
Astrid Netz, Wilhelm Amberg, Udo Lange, Michael Ochse, Charles W. Hutchins +2 more |
2013-07-09 |
$14,335,000 |