| 10138246 |
Deuterated triazolopyridazine as a kinase modulator |
Patrick Blasius Furer, Ronaldus Arnodus Hendrika Joseph Gilissen, Ioannnis Nicolaos Houpis, Timothy Pietro Suren Perera, Philip Pye |
2018-11-27 |
| 10087187 |
Imidazopyridazine derivatives as PI3KB inhibitors |
Laurence Anne Mevellec, Sophie Coupa, Virginie Sophie Poncelet, Isabelle Noëlle Constance Pilatte, Elisabeth Therese Jeanne Pasquier +6 more |
2018-10-02 |
| 10077261 |
Imidazolin-5-one derivative useful as FASN inhibitors for the treatment of cancer |
Peter J. Connolly, Gilles Bignan, Tianbao Lu, Michael H. Parker, Donald Ludovici +3 more |
2018-09-18 |
| 10052320 |
Substituted quinoxalines as FGFR kinase inhibitors |
Steven John Woodhead, Christopher William Murray, Valerio Berdini, Gordon Saxty, Gilbert Ebai Besong +2 more |
2018-08-21 |
| 10045982 |
Substituted pyrido[2,3-b]pyrazines as FGFR kinase inhibitors |
Valerio Berdini, Gordon Saxty, Patrick René Angibaud, Olivier Alexis Georges Querolle, Virginie Sophie Poncelet +1 more |
2018-08-14 |
| 10017509 |
Macrocylic pyrimidine derivatives |
Gaston Stanislas Marcella Diels, Bruno Schoentjes, Matthias VERSELE, Didier Jean-Claude Berthelot, Marc Willems +3 more |
2018-07-10 |
| 10000502 |
Substituted thiohydantoin derivatives as androgen receptor antagonists |
Gilles Bignan, Peter J. Connolly, Ian Hickson, Vineet Pande, Zhuming Zhang +3 more |
2018-06-19 |
| 9975899 |
Antifungal 5,6-dihydro-4H-pyrrolo[1,2-a][1,4]benzo-diazepines and 6H-pyrrolo[1,2-a][1,4]benzodiazepines substituted with heterocyclic derivatives |
Louis Jules Roger Marie Maes, Kelly de Wit, Koen Augustyns |
2018-05-22 |